JP2012140432A5 - - Google Patents
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- Publication number
- JP2012140432A5 JP2012140432A5 JP2012015294A JP2012015294A JP2012140432A5 JP 2012140432 A5 JP2012140432 A5 JP 2012140432A5 JP 2012015294 A JP2012015294 A JP 2012015294A JP 2012015294 A JP2012015294 A JP 2012015294A JP 2012140432 A5 JP2012140432 A5 JP 2012140432A5
- Authority
- JP
- Japan
- Prior art keywords
- heterocyclyl
- cycloalkyl
- alkyl
- heteroaryl
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17094399P | 1999-12-15 | 1999-12-15 | |
| US60/170,943 | 1999-12-15 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001544761A Division JP4990456B2 (ja) | 1999-12-15 | 2000-12-15 | 抗菌剤としてのダプトマイシンアナログ |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2012140432A JP2012140432A (ja) | 2012-07-26 |
| JP2012140432A5 true JP2012140432A5 (US20040106767A1-20040603-C00005.png) | 2013-04-11 |
Family
ID=22621910
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001544761A Expired - Fee Related JP4990456B2 (ja) | 1999-12-15 | 2000-12-15 | 抗菌剤としてのダプトマイシンアナログ |
| JP2012015294A Pending JP2012140432A (ja) | 1999-12-15 | 2012-01-27 | 抗菌剤としてのダプトマイシンアナログ |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001544761A Expired - Fee Related JP4990456B2 (ja) | 1999-12-15 | 2000-12-15 | 抗菌剤としてのダプトマイシンアナログ |
Country Status (13)
Families Citing this family (41)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR0016467A (pt) * | 1999-12-15 | 2002-08-27 | Cubist Pharm Inc | Lipopeptìdeos como agentes antibacterianos |
| US6696412B1 (en) | 2000-01-20 | 2004-02-24 | Cubist Pharmaceuticals, Inc. | High purity lipopeptides, Lipopeptide micelles and processes for preparing same |
| CA2301336A1 (en) * | 2000-03-17 | 2001-09-17 | Michael T. Kelly | Topical treatment of rosacea |
| US20060014674A1 (en) | 2000-12-18 | 2006-01-19 | Dennis Keith | Methods for preparing purified lipopeptides |
| NZ571597A (en) | 2000-12-18 | 2010-05-28 | Cubist Pharm Inc | Method for preparing crystalline and crystal-like forms of purified daptomycin lipopeptides |
| DE60232158D1 (de) * | 2001-08-06 | 2009-06-10 | Cubist Pharm Inc | Lipopeptid-stereoisomere, verfahren zu ihrer herstellung und nützliche zwischenprodukte |
| EP1932853A1 (en) | 2001-08-06 | 2008-06-18 | Cubist Pharmaceutical Inc. | Novel depsipeptides and process for preparing same |
| CA2458644A1 (en) * | 2001-08-28 | 2003-03-13 | Pharmacia Corporation | Crystaline clindamycin free base |
| US6767718B2 (en) | 2002-05-10 | 2004-07-27 | Biosource Pharm, Inc. | Lipodepsipeptide antibiotics and methods of preparation |
| AU2003265241A1 (en) * | 2002-05-23 | 2003-12-12 | Activbiotics, Inc. | Methods of treating bacterial infections and diseases associated therewith |
| AU2003240545A1 (en) | 2002-06-06 | 2003-12-22 | Therapeutics Corporation Genome | Use of ramoplanin to treat diseases associated with the use of antibiotics |
| IL150907A (en) * | 2002-07-25 | 2007-07-04 | Stephan Cherkez | Process for the preparation of stable amorphous calcium pseudomonate |
| ITMI20022076A1 (it) * | 2002-10-01 | 2004-04-02 | Antibioticos Spa | Sali di intermedi del cefdinir. |
| US20040132764A1 (en) * | 2002-10-23 | 2004-07-08 | Morphochem Aktiengesellschaft Fuer Kombinatorische Chemie | Antibiotics for the treatment of infections in acidic environments |
| US20060004185A1 (en) | 2004-07-01 | 2006-01-05 | Leese Richard A | Peptide antibiotics and peptide intermediates for their prepartion |
| CA2587848A1 (en) * | 2004-11-12 | 2006-10-19 | Cubist Pharmaceuticals, Inc. | Antiinfective lipopeptides |
| US20080051326A1 (en) * | 2004-11-12 | 2008-02-28 | Alexander Dylan C | Antiinfective Lipopeptides |
| AU2006242535B2 (en) * | 2005-04-29 | 2012-08-09 | Merck Sharp & Dohme Corp. | Therapeutic compositions |
| WO2007127218A2 (en) * | 2006-04-26 | 2007-11-08 | Taro Pharmaceuticals U.S.A., Inc. | Streptomyces-derived antimicrobial compound and method of using same against antibiotic-resistant bacteria |
| CA2659684A1 (en) * | 2006-08-02 | 2008-02-07 | Johannes Gutenberg-Universitaet Mainz | Medicament for lct poisoning |
| US8662086B2 (en) | 2007-02-06 | 2014-03-04 | BBK Tobacco & Foods, LLP | Reclosable package with magnetic clasp for rolling papers used in smoking articles |
| US20080185010A1 (en) * | 2007-02-06 | 2008-08-07 | Kesselman Joshua D | Interleaved Transparent Cellulose Paper with Opaque Adhesive |
| US8584854B2 (en) * | 2007-02-06 | 2013-11-19 | BBK Tobacco & Foods, LLP | Reclosable package with magnetic clasp and detachable tray for rolling papers used in smoking articles |
| US20090020443A1 (en) * | 2007-05-09 | 2009-01-22 | Kesselman Joshua D | Credit Card Carrying Pack for Rolling Papers |
| US9072319B2 (en) | 2007-06-15 | 2015-07-07 | Joshua D. Kesselman | Rolling paper structures for creating smoking articles and gummed, coiled inserts for same |
| US9161572B2 (en) * | 2007-06-15 | 2015-10-20 | Bbk Tobacco & Foods, Inc. | Structures for creating smoking articles and methods of packaging same |
| US20090014342A1 (en) * | 2007-07-14 | 2009-01-15 | Kesselman Joshua D | Rolling papers and methods of packaging same |
| EP2018864A1 (en) | 2007-07-23 | 2009-01-28 | Biomet Deutschland GmbH | Pharmaceutical composition, substrate comprising a pharmaceutical composition, and use of a pharmaceutical composition |
| CA2710602A1 (en) * | 2007-12-26 | 2009-07-09 | Lead Therapeutics, Inc. | Novel semi-synthetic glycopeptides as antibacterial agents |
| US8393332B2 (en) | 2008-08-21 | 2013-03-12 | BBK Tobacco & Foods, LLP | Packaging for rolling papers for smoking articles |
| GB2465863A (en) * | 2008-12-05 | 2010-06-09 | Lead Therapeutics Inc | Semi-synthetic heptapeptidic glycopeptides for the treatment of bacterial infections |
| PL2379580T3 (pl) * | 2008-12-22 | 2014-05-30 | Merck Sharp & Dohme | Nowe środki przeciwbakteryjne do leczenia zakażeń wywołanych bakteriami Gram-dodatnimi |
| NZ593892A (en) | 2008-12-23 | 2013-11-29 | Biosource Pharm Inc | Antibiotic compositions for the treatment of gram negative infections |
| ES2374779B1 (es) * | 2010-03-10 | 2012-12-27 | Universidad De Barcelona | Compuestos péptidicos útiles como agentes antibacterianos. |
| US8415307B1 (en) | 2010-06-23 | 2013-04-09 | Biosource Pharm, Inc. | Antibiotic compositions for the treatment of gram negative infections |
| WO2012011917A1 (en) * | 2010-07-23 | 2012-01-26 | Activbiotics Pharma, Llc | Administration of rifalazil to immunocompromised patients |
| US10072045B1 (en) | 2017-06-26 | 2018-09-11 | Ramapo Pharmaceuticals, Inc. | Antibacterial lipopeptides and methods for their preparation and use |
| US10526343B2 (en) | 2018-03-26 | 2020-01-07 | University Of Sharjah | Heterocyclic systems and pharmaceutical applications thereof |
| CN110577581A (zh) * | 2018-06-07 | 2019-12-17 | 美国蓝博药业公司 | 一种新型的抑菌脂肽化合物、制备方法及其应用 |
| CN109182563B (zh) * | 2018-08-01 | 2020-07-14 | 浙江大学 | 检测20种dfrA类甲氧苄胺嘧啶类药物耐药基因的方法及所用试剂盒 |
| CN113061164B (zh) * | 2021-03-29 | 2023-01-10 | 四川大学 | 环脂肽类化合物及其在抗类风湿关节炎药物中的应用 |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3854480A (en) | 1969-04-01 | 1974-12-17 | Alza Corp | Drug-delivery system |
| USRE32333E (en) | 1978-10-16 | 1987-01-20 | Eli Lilly And Company | A-21978 Antibiotics and process for their production |
| USRE32455E (en) | 1978-10-16 | 1987-07-07 | Eli Lilly And Company | A-21978 antibiotics and process for their production |
| DE3376424D1 (en) | 1982-02-27 | 1988-06-01 | Beecham Group Plc | Antibacterial 1-normon-2-yl-heterocyclic compounds |
| US4399067A (en) | 1982-05-21 | 1983-08-16 | Eli Lilly And Company | Derivatives of A-21978C cyclic peptides |
| USRE32310E (en) | 1982-05-21 | 1986-12-16 | Eli Lilly And Company | Derivatives of A-21978C cyclic peptides |
| US4482487A (en) | 1982-05-21 | 1984-11-13 | Eli Lilly And Company | A-21978C cyclic peptides |
| US4396543A (en) | 1982-05-21 | 1983-08-02 | Eli Lilly And Company | Derivatives of A-21978C cyclic peptides |
| US4524135A (en) | 1982-05-21 | 1985-06-18 | Eli Lilly And Company | A-21978C cyclic peptides |
| USRE32311E (en) | 1982-05-21 | 1986-12-16 | Eli Lilly And Company | Derivatives of A-21978C cyclic peptides |
| IL68700A0 (en) * | 1982-05-21 | 1983-09-30 | Lilly Co Eli | Improvements relating to a-21978c cyclic peptide derivatives and their production |
| US4537717A (en) | 1982-05-21 | 1985-08-27 | Eli Lilly And Company | Derivatives of A-21978C cyclic peptides |
| US4452775A (en) | 1982-12-03 | 1984-06-05 | Syntex (U.S.A.) Inc. | Cholesterol matrix delivery system for sustained release of macromolecules |
| EP0178152B1 (en) | 1984-10-09 | 1991-09-25 | Eli Lilly And Company | Production of a-21978c derivatives |
| US4885243A (en) | 1984-10-09 | 1989-12-05 | Eli Lilly And Company | Process for producing A-21978C derivatives |
| US4874843A (en) | 1987-12-03 | 1989-10-17 | Eli Lilly And Company | Chromatographic purification process |
| ZA883887B (en) | 1987-06-10 | 1990-02-28 | Lilly Co Eli | Chromatographic purification process |
| ES2089133T3 (es) | 1990-06-07 | 1996-10-01 | Lilly Co Eli | Desacilasa de lipopeptidos. |
| JPH04167172A (ja) | 1990-10-31 | 1992-06-15 | Nec Corp | ベクトルプロセッサ |
| EP0712405A1 (en) | 1993-08-13 | 1996-05-22 | Smithkline Beecham Plc | Derivatives of monic acids a and c having antibacterial, antimycoplasmatical, antifungal and herbicidal activity |
| DE4411025A1 (de) | 1994-03-30 | 1995-10-05 | Hoechst Ag | Lipopeptid-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung |
| ATE544851T1 (de) | 1996-03-08 | 2012-02-15 | Astellas Pharma Inc | Verfahren zur deacylierung von zyklischen lipopeptiden |
| DE19807972A1 (de) | 1998-02-25 | 1999-08-26 | Hoechst Marion Roussel De Gmbh | Lipopeptidantibiotika-Calciumsalze, Verfahren zu ihrer Herstellung und Verwendung |
| HU230656B1 (hu) | 1998-09-25 | 2017-06-28 | Cubist Pharmaceuticals Llc | Daptomicin alkalmazása |
| US9393093B2 (en) | 2008-02-18 | 2016-07-19 | Covidien Lp | Clip for implant deployment device |
-
2000
- 2000-12-15 WO PCT/US2000/034118 patent/WO2001044272A2/en active Application Filing
- 2000-12-15 MX MXPA02006029A patent/MXPA02006029A/es unknown
- 2000-12-15 IL IL15022300A patent/IL150223A0/xx unknown
- 2000-12-15 US US09/738,742 patent/US6911525B2/en not_active Expired - Lifetime
- 2000-12-15 EP EP00986444A patent/EP1240181A2/en not_active Withdrawn
- 2000-12-15 BR BR0017026-7A patent/BR0017026A/pt not_active Application Discontinuation
- 2000-12-15 JP JP2001544761A patent/JP4990456B2/ja not_active Expired - Fee Related
- 2000-12-15 EP EP10182947A patent/EP2298790A1/en not_active Withdrawn
- 2000-12-15 CA CA002393907A patent/CA2393907A1/en not_active Abandoned
- 2000-12-15 EP EP10182938A patent/EP2295444A3/en not_active Withdrawn
- 2000-12-15 CN CN00818471A patent/CN1425025A/zh active Pending
- 2000-12-15 EP EP07022686A patent/EP1884520A3/en not_active Withdrawn
- 2000-12-15 KR KR1020027007665A patent/KR20020063227A/ko not_active Application Discontinuation
- 2000-12-15 AU AU22682/01A patent/AU784755B2/en not_active Ceased
-
2002
- 2002-06-13 IL IL150223A patent/IL150223A/en not_active IP Right Cessation
- 2002-06-17 NO NO20022888A patent/NO20022888L/no not_active Application Discontinuation
- 2002-06-25 ZA ZA200205106A patent/ZA200205106B/xx unknown
-
2005
- 2005-05-04 US US11/121,851 patent/US7335725B2/en not_active Expired - Fee Related
-
2012
- 2012-01-27 JP JP2012015294A patent/JP2012140432A/ja active Pending
