JP2012012417A5 - - Google Patents

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Publication number
JP2012012417A5
JP2012012417A5 JP2011227135A JP2011227135A JP2012012417A5 JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5 JP 2011227135 A JP2011227135 A JP 2011227135A JP 2011227135 A JP2011227135 A JP 2011227135A JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5
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JP
Japan
Prior art keywords
compound
independently
occurrence
optionally substituted
nrco
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011227135A
Other languages
English (en)
Japanese (ja)
Other versions
JP2012012417A (ja
Filing date
Publication date
Priority claimed from PCT/US2005/011358 external-priority patent/WO2005103050A2/en
Application filed filed Critical
Publication of JP2012012417A publication Critical patent/JP2012012417A/ja
Publication of JP2012012417A5 publication Critical patent/JP2012012417A5/ja
Pending legal-status Critical Current

Links

JP2011227135A 2004-06-30 2011-10-14 タンパク質キナーゼのインヒビターとして有用なアザインドール Pending JP2012012417A (ja)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US60/584,383 2004-06-30
US58472104P 2004-07-01 2004-07-01
US60/584,721 2004-07-01
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
USPCT/US05/11358 2005-04-04
US11/098,751 2005-04-04
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2007519460A Division JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013001760A Division JP2013064015A (ja) 2004-06-30 2013-01-09 タンパク質キナーゼのインヒビターとして有用なアザインドール

Publications (2)

Publication Number Publication Date
JP2012012417A JP2012012417A (ja) 2012-01-19
JP2012012417A5 true JP2012012417A5 (https=) 2013-02-28

Family

ID=37801682

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007519460A Expired - Fee Related JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール
JP2011227135A Pending JP2012012417A (ja) 2004-06-30 2011-10-14 タンパク質キナーゼのインヒビターとして有用なアザインドール

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2007519460A Expired - Fee Related JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール

Country Status (4)

Country Link
JP (2) JP5122280B2 (https=)
IL (1) IL180303A0 (https=)
MX (1) MX2007000092A (https=)
NO (1) NO20070502L (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.
CA2575466A1 (en) * 2004-08-13 2006-02-23 Genentech, Inc. Thiazole based inhibitors of atp-utilizing enzymes
DE102008038221A1 (de) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-Azaindolderivate
DE102009058280A1 (de) * 2009-12-14 2011-06-16 Merck Patent Gmbh Thiazolderivate
AU2011239966B2 (en) 2010-04-16 2014-05-08 Ac Immune S.A. Novel compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
MX2013000103A (es) * 2010-06-23 2013-06-13 Vertex Pharma Derivados de pirrolo-pirazina utiles como inhibidores de cinasa art.
DE102011105469A1 (de) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-Azaindolderivate
SG11201407919WA (en) * 2012-05-31 2014-12-30 Phenex Pharmaceuticals Ag Carboxamide or sulfonamide substituted thiazoles and related derivatives as modulators for the orphan nuclear receptor ror[gamma]
TR201820925T4 (tr) 2014-02-04 2019-01-21 Taiho Pharmaceutical Co Ltd Azaindol türevi.
MX2023003996A (es) * 2020-10-05 2023-06-15 Enliven Inc Compuestos de 7-azaindol para la inhibicion de tirosina cinasas bcr-abl.
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
JP2003525291A (ja) * 2000-03-01 2003-08-26 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ２，４−二置換チアゾリル誘導体
SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
AR049333A1 (es) * 2004-04-02 2006-07-19 Vertex Pharma Azaindoles inhibidores de proteinquinasas rock y otras proteinas quinasas. composiciones farmaceuticas.
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.

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