MX2007000092A - Azaindoles utiles como inhibidores de proteinas cinasas. - Google Patents

Azaindoles utiles como inhibidores de proteinas cinasas.

Info

Publication number
MX2007000092A
MX2007000092A MX2007000092A MX2007000092A MX2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A
Authority
MX
Mexico
Prior art keywords
compound according
optionally substituted
nitrogen
sulfur
oxygen
Prior art date
Application number
MX2007000092A
Other languages
English (en)
Spanish (es)
Inventor
Guy Brenchley
Michael Mortimore
Francoise Pierad
Juan Miguel Jimenez
Ronald Kengtel
Francesca Mazzei
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2005/011358 external-priority patent/WO2005103050A2/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Priority claimed from PCT/US2005/023429 external-priority patent/WO2006004984A1/en
Publication of MX2007000092A publication Critical patent/MX2007000092A/es

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
MX2007000092A 2004-06-30 2005-06-29 Azaindoles utiles como inhibidores de proteinas cinasas. MX2007000092A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US58472104P 2004-07-01 2004-07-01
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
PCT/US2005/023429 WO2006004984A1 (en) 2004-06-30 2005-06-29 Azaindoles useful as inhibitors of protein kinases

Publications (1)

Publication Number Publication Date
MX2007000092A true MX2007000092A (es) 2007-03-07

Family

ID=37801682

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007000092A MX2007000092A (es) 2004-06-30 2005-06-29 Azaindoles utiles como inhibidores de proteinas cinasas.

Country Status (4)

Country Link
JP (2) JP5122280B2 (https=)
IL (1) IL180303A0 (https=)
MX (1) MX2007000092A (https=)
NO (1) NO20070502L (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.
SG155222A1 (en) * 2004-08-13 2009-09-30 Genentech Inc Thiazole based inhibitors of atp-utilizing enzymes
DE102008038221A1 (de) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-Azaindolderivate
DE102009058280A1 (de) * 2009-12-14 2011-06-16 Merck Patent Gmbh Thiazolderivate
PH12012502079A1 (en) 2010-04-16 2013-02-11 Ac Immune Sa Novel compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
CA2803802A1 (en) * 2010-06-23 2011-12-29 Vertex Pharmaceuticals Incorporated Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase
DE102011105469A1 (de) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-Azaindolderivate
CN107007597A (zh) * 2012-05-31 2017-08-04 菲尼克斯药品股份公司 作为孤儿核受体RORγ调节物的经甲酰胺或磺酰胺取代的噻唑及相关衍生物的制药用途
TR201820925T4 (tr) * 2014-02-04 2019-01-21 Taiho Pharmaceutical Co Ltd Azaindol türevi.
EP4225741A4 (en) * 2020-10-05 2024-10-30 Enliven Inc. 7-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
AU2001237401B2 (en) * 2000-03-01 2006-11-09 Janssen Pharmaceutica N.V. 2,4-disubstituted thiazolyl derivatives
SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
KR20070002081A (ko) * 2004-04-02 2007-01-04 버텍스 파마슈티칼스 인코포레이티드 Rock 및 기타 단백질 키나아제의 억제제로서 유용한아자인돌
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.

Also Published As

Publication number Publication date
JP5122280B2 (ja) 2013-01-16
JP2012012417A (ja) 2012-01-19
IL180303A0 (en) 2007-06-03
NO20070502L (no) 2007-01-26
JP2008513352A (ja) 2008-05-01

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