JP2011520991A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2011520991A5 JP2011520991A5 JP2011510782A JP2011510782A JP2011520991A5 JP 2011520991 A5 JP2011520991 A5 JP 2011520991A5 JP 2011510782 A JP2011510782 A JP 2011510782A JP 2011510782 A JP2011510782 A JP 2011510782A JP 2011520991 A5 JP2011520991 A5 JP 2011520991A5
- Authority
- JP
- Japan
- Prior art keywords
- ethoxy
- compound
- pharmaceutical composition
- compound according
- pyridazinyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims 9
- 239000008194 pharmaceutical composition Substances 0.000 claims 5
- 241000430519 Human rhinovirus sp. Species 0.000 claims 4
- 208000005155 Picornaviridae Infections Diseases 0.000 claims 4
- 239000003814 drug Substances 0.000 claims 3
- -1 6- {2- [1- (6-Methyl-3-pyridazinyl) -4-piperidinyl] ethoxy} -3-ethoxy-1,2-benzisoxazole bis-phosphate dihydrogen salt Chemical class 0.000 claims 2
- NBIIXXVUZAFLBC-UHFFFAOYSA-N Phosphoric acid Chemical compound OP(O)(O)=O NBIIXXVUZAFLBC-UHFFFAOYSA-N 0.000 claims 2
- 238000004519 manufacturing process Methods 0.000 claims 2
- DKSVBVKHUICELN-UHFFFAOYSA-N 3-ethoxy-6-[2-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]ethoxy]-1,2-benzoxazole Chemical compound C=1C=C2C(OCC)=NOC2=CC=1OCCC(CC1)CCN1C1=CC=C(C)N=N1 DKSVBVKHUICELN-UHFFFAOYSA-N 0.000 claims 1
- WQZGKKKJIJFFOK-GASJEMHNSA-N Glucose Natural products OC[C@H]1OC(O)[C@H](O)[C@@H](O)[C@@H]1O WQZGKKKJIJFFOK-GASJEMHNSA-N 0.000 claims 1
- 229910000147 aluminium phosphate Inorganic materials 0.000 claims 1
- 239000003937 drug carrier Substances 0.000 claims 1
- 125000001301 ethoxy group Chemical group [H]C([H])([H])C([H])([H])O* 0.000 claims 1
- 239000008103 glucose Substances 0.000 claims 1
- 238000000034 method Methods 0.000 claims 1
- 239000000203 mixture Substances 0.000 claims 1
- 239000000843 powder Substances 0.000 claims 1
- 239000012453 solvate Substances 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5634108P | 2008-05-27 | 2008-05-27 | |
| US61/056,341 | 2008-05-27 | ||
| PCT/AU2009/000663 WO2009143571A1 (en) | 2008-05-27 | 2009-05-27 | Antiviral salts |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011520991A JP2011520991A (ja) | 2011-07-21 |
| JP2011520991A5 true JP2011520991A5 (https=) | 2012-07-05 |
| JP5469662B2 JP5469662B2 (ja) | 2014-04-16 |
Family
ID=41376478
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011510782A Expired - Fee Related JP5469662B2 (ja) | 2008-05-27 | 2009-05-27 | 抗ウイルス剤の塩 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US8580791B2 (https=) |
| EP (1) | EP2297141B1 (https=) |
| JP (1) | JP5469662B2 (https=) |
| KR (1) | KR20110019759A (https=) |
| CN (1) | CN102046621B (https=) |
| AU (1) | AU2009253738B2 (https=) |
| BR (1) | BRPI0912038A2 (https=) |
| CA (1) | CA2725618C (https=) |
| CO (1) | CO6280534A2 (https=) |
| EA (1) | EA020455B1 (https=) |
| MX (1) | MX2010013019A (https=) |
| NZ (1) | NZ590286A (https=) |
| WO (1) | WO2009143571A1 (https=) |
| ZA (1) | ZA201009284B (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ603040A (en) * | 2010-04-15 | 2015-03-27 | Biota Scient Management | Compound for treatment of respiratory condition or disease |
| EP2585067B1 (en) | 2010-06-25 | 2017-08-09 | Biota Scientific Management Pty Ltd | Compound for the treatment of enteroviruses |
| CN102617462B (zh) * | 2012-02-28 | 2014-02-12 | 南京大学 | 特异性抑制肌肉微小核糖核酸的化合物及其合成方法和应用 |
| EA201692549A1 (ru) * | 2014-06-20 | 2017-08-31 | Эвайраджен Терепьютикс, Инк. | Безводная кристаллическая форма свободного основания 6-{2-[1-(6-метил-3-пиридазинил)-4-пиперидинил]этокси}-3-этокси-1,2-бензизоксазола |
| US20250281519A1 (en) * | 2021-05-05 | 2025-09-11 | Emory University | Nucleotide and nucleoside therapeutic compositions, combinations and uses related thereto |
| WO2024192151A2 (en) * | 2023-03-13 | 2024-09-19 | Altesa BioSciences, Inc. | Method of dosing vapendavir to treat enterovirus infections |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1170387B (it) | 1982-06-07 | 1987-06-03 | Glaxo Group Ltd | Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono |
| GB2162522B (en) | 1984-08-01 | 1988-02-24 | Glaxo Group Ltd | An indole derivative |
| GB9026998D0 (en) | 1990-12-12 | 1991-01-30 | Glaxo Group Ltd | Medicaments |
| US5514778A (en) * | 1993-07-01 | 1996-05-07 | Eli Lilly And Company | Anti-picornaviral agents |
| US5693661A (en) * | 1995-06-07 | 1997-12-02 | Eli Lilly And Company | Anti-viral compounds |
| US5545653A (en) * | 1995-06-07 | 1996-08-13 | Eli Lilly And Company | Anti-viral compounds |
| US5891874A (en) * | 1996-06-05 | 1999-04-06 | Eli Lilly And Company | Anti-viral compound |
| US5821242A (en) * | 1996-06-06 | 1998-10-13 | Eli Lilly And Company | Anti-viral compounds |
| AU6031898A (en) * | 1997-01-22 | 1998-08-07 | Eli Lilly And Company | Anti-viral compounds |
| CA2293508A1 (en) * | 1997-06-04 | 1998-12-10 | Louis Nickolaus Jungheim | Anti-viral compounds |
| CZ289425B6 (cs) * | 1998-05-20 | 2002-01-16 | Eli Lilly And Company | Imidazo[1,2-a] pyridinové sloučeniny, jejich pouľití a farmaceutický přípravek s jejich obsahem |
| US6358971B1 (en) * | 1998-05-20 | 2002-03-19 | Eli Lilly And Company | Anti-viral compounds |
| AUPR213700A0 (en) | 2000-12-18 | 2001-01-25 | Biota Scientific Management Pty Ltd | Antiviral agents |
-
2009
- 2009-05-27 CA CA2725618A patent/CA2725618C/en not_active Expired - Fee Related
- 2009-05-27 AU AU2009253738A patent/AU2009253738B2/en not_active Ceased
- 2009-05-27 EA EA201001835A patent/EA020455B1/ru not_active IP Right Cessation
- 2009-05-27 US US12/994,633 patent/US8580791B2/en active Active
- 2009-05-27 NZ NZ590286A patent/NZ590286A/en not_active IP Right Cessation
- 2009-05-27 CN CN200980120191.2A patent/CN102046621B/zh not_active Expired - Fee Related
- 2009-05-27 EP EP09753335.0A patent/EP2297141B1/en not_active Not-in-force
- 2009-05-27 JP JP2011510782A patent/JP5469662B2/ja not_active Expired - Fee Related
- 2009-05-27 WO PCT/AU2009/000663 patent/WO2009143571A1/en not_active Ceased
- 2009-05-27 BR BRPI0912038A patent/BRPI0912038A2/pt not_active IP Right Cessation
- 2009-05-27 KR KR1020107029303A patent/KR20110019759A/ko not_active Ceased
- 2009-05-27 MX MX2010013019A patent/MX2010013019A/es active IP Right Grant
-
2010
- 2010-11-25 CO CO10148308A patent/CO6280534A2/es not_active Application Discontinuation
- 2010-12-23 ZA ZA2010/09284A patent/ZA201009284B/en unknown
-
2013
- 2013-09-10 US US14/023,280 patent/US9206171B2/en not_active Expired - Fee Related
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2011520991A5 (https=) | ||
| UA90545C2 (ru) | Твердая фармацевтическая лекарственная форма для перорального введения с быстрым высвобождением ингибитора фактора ха свертывания крови | |
| WO2007127635A3 (en) | Diketo-piperazine and piperidine derivatives as antiviral agents | |
| NZ593712A (en) | Intermediates for synthesising nucleoside aryl phosphoramidates | |
| JP2008538115A5 (https=) | ||
| JP2011507977A5 (https=) | ||
| WO2009080705A3 (en) | Bis-thiazole derivatives, process for their preparation and their use as medicaments | |
| MX2008013212A (es) | 4-anilinquinolina-3-carboxamidas como inhibidores de la cinsa csf-1r. | |
| JP2009506014A5 (https=) | ||
| NZ596820A (en) | Trans-4-[[(5s)-5-[[[3,5-bis(trifluoromethyl)phenyl]methyl] (2-methyl-2h-tetrazol-5-yl)amino]-2,3,4,5-tetrahydro-7,9-dimethyl-1h-1-benzazepin-1-yl]methyl]-cyclohexanecarboxylic acid | |
| JP2010518061A5 (https=) | ||
| JP2014503593A5 (https=) | ||
| WO2008009639A2 (en) | New indications for direct thrombin inhibitors | |
| NZ596154A (en) | Cyclic compound having substituted phenyl group | |
| CN115315423A (zh) | 取代芳基类化合物 | |
| JP2008534453A5 (https=) | ||
| JP2011527687A5 (https=) | ||
| NO20044571L (no) | Isokinolinderivater | |
| JP2010521516A5 (https=) | ||
| SG179031A1 (en) | Hsl inhibitors useful in the treatment of diabetes | |
| JP2012508256A5 (https=) | ||
| JP2009513604A5 (https=) | ||
| JP2010500284A5 (https=) | ||
| JP2011519873A5 (https=) | ||
| JP2012504584A5 (https=) |