JP2011503081A - グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用 - Google Patents

グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用 Download PDF

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JP2011503081A
JP2011503081A JP2010533163A JP2010533163A JP2011503081A JP 2011503081 A JP2011503081 A JP 2011503081A JP 2010533163 A JP2010533163 A JP 2010533163A JP 2010533163 A JP2010533163 A JP 2010533163A JP 2011503081 A JP2011503081 A JP 2011503081A
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alkyl
disease
hydrogen
inhibitor
substituted
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JP2011503081A5 (https=
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ティ・ジー・ムラリ・ダー
ハイ−ユン・シャオ
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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JP2010533163A 2007-11-01 2008-10-30 グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用 Withdrawn JP2011503081A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US98451507P 2007-11-01 2007-11-01
PCT/US2008/081702 WO2009058944A2 (en) 2007-11-01 2008-10-30 Nonsteroidal compounds useful as modulators of glucocorticoid receptor ap-1 and /or nf- kappa b activity and use thereof

Publications (2)

Publication Number Publication Date
JP2011503081A true JP2011503081A (ja) 2011-01-27
JP2011503081A5 JP2011503081A5 (https=) 2011-04-07

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JP2010533163A Withdrawn JP2011503081A (ja) 2007-11-01 2008-10-30 グルココルチコイド受容体、ＡＰ−１および／またはＮＦ−κＢ活性の調節剤として有用な非ステロイド性化合物、並びにその使用

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US (1) US8309730B2 (https=)
EP (1) EP2209780B1 (https=)
JP (1) JP2011503081A (https=)
CN (1) CN101910171A (https=)
ES (1) ES2448839T3 (https=)
WO (1) WO2009058944A2 (https=)

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JP7789561B2 (ja) 2019-02-22 2025-12-22 コーセプト セラピューティクス， インコーポレイテッド レラコリラント、ヘテロアリール－ケトン縮合アザデカリングルココルチコイド受容体調節物質の治療用途
JP7569492B2 (ja) 2019-12-11 2024-10-18 コーセプト セラピューティクス， インコーポレイテッド 抗精神病薬誘発性体重増加のミリコリラントによる治療方法
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EP2209780A2 (en) 2010-07-28
WO2009058944A3 (en) 2009-07-02
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US20110263494A1 (en) 2011-10-27
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