JP2010540649A5 - - Google Patents

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Publication number
JP2010540649A5
JP2010540649A5 JP2010528066A JP2010528066A JP2010540649A5 JP 2010540649 A5 JP2010540649 A5 JP 2010540649A5 JP 2010528066 A JP2010528066 A JP 2010528066A JP 2010528066 A JP2010528066 A JP 2010528066A JP 2010540649 A5 JP2010540649 A5 JP 2010540649A5
Authority
JP
Japan
Prior art keywords
aliphatic
pharmaceutically acceptable
acceptable salt
treating
cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010528066A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010540649A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/078239 external-priority patent/WO2009045992A2/en
Publication of JP2010540649A publication Critical patent/JP2010540649A/ja
Publication of JP2010540649A5 publication Critical patent/JP2010540649A5/ja
Pending legal-status Critical Current

Links

JP2010528066A 2007-10-03 2008-09-30 c−METタンパク質の阻害剤 Pending JP2010540649A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US97730507P 2007-10-03 2007-10-03
PCT/US2008/078239 WO2009045992A2 (en) 2007-10-03 2008-09-30 C-met protein kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2010540649A JP2010540649A (ja) 2010-12-24
JP2010540649A5 true JP2010540649A5 (enExample) 2012-10-18

Family

ID=40512401

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010528066A Pending JP2010540649A (ja) 2007-10-03 2008-09-30 c−METタンパク質の阻害剤

Country Status (12)

Country Link
US (1) US8481524B2 (enExample)
EP (1) EP2205589B1 (enExample)
JP (1) JP2010540649A (enExample)
CN (1) CN101990538A (enExample)
AT (1) ATE502935T1 (enExample)
AU (1) AU2008308900A1 (enExample)
CA (1) CA2701124A1 (enExample)
DE (1) DE602008005786D1 (enExample)
ES (1) ES2361650T3 (enExample)
MX (1) MX2010003563A (enExample)
NZ (1) NZ584311A (enExample)
WO (1) WO2009045992A2 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102317277A (zh) 2008-10-21 2012-01-11 沃泰克斯药物股份有限公司 C-met蛋白激酶抑制剂
ES2534516T3 (es) 2010-01-07 2015-04-23 E.I. Du Pont De Nemours And Company Compuestos heterocíclicos fungicidas
JP2013532627A (ja) 2010-07-01 2013-08-19 武田薬品工業株式会社 cMET阻害剤とHGFおよび/またはcMETに対する抗体との組み合わせ
JP5965499B2 (ja) 2012-12-25 2016-08-03 日本曹達株式会社 ハロゲン化アニリンおよびその製造方法
CN103242216A (zh) * 2013-05-07 2013-08-14 兰州梦唐精细化工有限公司 N- Boc -六氢-5-氧代环戊[C]并吡咯的合成方法
US9896436B2 (en) 2014-09-16 2018-02-20 Celgene Quanticel Research, Inc. Histone demethylase inhibitors
JP6660060B2 (ja) 2014-09-16 2020-03-04 セルジーン クオンティセル リサーチ,インク. ヒストンデメチラーゼ阻害剤
EP3229836B1 (en) 2014-12-09 2019-11-13 Institut National de la Sante et de la Recherche Medicale (INSERM) Human monoclonal antibodies against axl
WO2016135041A1 (en) 2015-02-26 2016-09-01 INSERM (Institut National de la Santé et de la Recherche Médicale) Fusion proteins and antibodies comprising thereof for promoting apoptosis

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1697352B1 (en) * 2003-09-24 2012-06-27 Vertex Pharmceuticals Incorporated 4-azole substituted imidazole compositions useful as inhibitors or c-met receptor tyrosine kinase
US7169781B2 (en) * 2003-10-17 2007-01-30 Hoffmann-La Roche Inc. Imidazole derivatives and their use as pharmaceutical agents
WO2007111904A2 (en) * 2006-03-22 2007-10-04 Vertex Pharmaceuticals Incorporated C-met protein kinase inhibitors for the treatment of proliferative disorders

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