JP2010523596A5 - - Google Patents

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Publication number
JP2010523596A5
JP2010523596A5 JP2010502341A JP2010502341A JP2010523596A5 JP 2010523596 A5 JP2010523596 A5 JP 2010523596A5 JP 2010502341 A JP2010502341 A JP 2010502341A JP 2010502341 A JP2010502341 A JP 2010502341A JP 2010523596 A5 JP2010523596 A5 JP 2010523596A5
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JP
Japan
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substituted
unsubstituted
alkylenyl
conr
cycloalkyl
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JP2010502341A
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English (en)
Japanese (ja)
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JP2010523596A (ja
JP5347164B2 (ja
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Priority claimed from PCT/US2008/059505 external-priority patent/WO2008124651A2/en
Publication of JP2010523596A publication Critical patent/JP2010523596A/ja
Publication of JP2010523596A5 publication Critical patent/JP2010523596A5/ja
Application granted granted Critical
Publication of JP5347164B2 publication Critical patent/JP5347164B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2010502341A 2007-04-05 2008-04-04 ニトロ−イミダゾール低酸素造影剤 Expired - Fee Related JP5347164B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US92193207P 2007-04-05 2007-04-05
US60/921,932 2007-04-05
US96425407P 2007-08-10 2007-08-10
US60/964,254 2007-08-10
PCT/US2008/059505 WO2008124651A2 (en) 2007-04-05 2008-04-04 Nitro-imidazole hypoxia imaging agents

Publications (3)

Publication Number Publication Date
JP2010523596A JP2010523596A (ja) 2010-07-15
JP2010523596A5 true JP2010523596A5 (OSRAM) 2011-05-12
JP5347164B2 JP5347164B2 (ja) 2013-11-20

Family

ID=39831553

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010502341A Expired - Fee Related JP5347164B2 (ja) 2007-04-05 2008-04-04 ニトロ−イミダゾール低酸素造影剤

Country Status (7)

Country Link
US (2) US7807394B2 (OSRAM)
EP (1) EP2132200B1 (OSRAM)
JP (1) JP5347164B2 (OSRAM)
KR (1) KR101523257B1 (OSRAM)
CN (1) CN101652360B (OSRAM)
CA (1) CA2683433C (OSRAM)
WO (1) WO2008124651A2 (OSRAM)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2683433C (en) * 2007-04-05 2016-10-11 Siemens Medical Solutions Usa, Inc. Nitro-imidazole hypoxia imaging agents
CN101709060B (zh) * 2009-12-02 2013-05-01 北京师范大学 一种f-三唑环-聚乙二醇-甲硝唑化合物及其制备方法
PT2534136T (pt) 2010-02-08 2017-12-15 Lantheus Medical Imaging Inc Métodos para sintetizar agentes de imagiologia, e seus intermediários
US10639608B2 (en) 2010-04-08 2020-05-05 Siemens Medical Solutions Usa, Inc. System, device and method for preparing tracers and transferring materials during radiosynthesis
WO2011127345A1 (en) 2010-04-08 2011-10-13 Siemens Medical Solutions Usa, Inc. Synthesis of 18f-labeled tracers in hydrous organic solvents
CN101921263A (zh) * 2010-04-16 2010-12-22 兰州大学 2-硝基咪唑衍生物及其用途和制备方法
CA3041113C (en) 2010-05-11 2022-01-18 Lantheus Medical Imaging, Inc. Compositions, methods, and systems for the synthesis and use of imaging agents
ES2731471T3 (es) 2011-09-09 2019-11-15 Lantheus Medical Imaging Inc Composiciones, métodos y sistemas para la síntesis y el uso de agentes de obtención de imágenes
CN103945901A (zh) * 2011-10-14 2014-07-23 住友重机械工业株式会社 带电粒子束照射系统以及带电粒子束照射计划方法
EP2793871A4 (en) * 2011-12-23 2015-07-22 Auckland Uniservices Ltd COMPOUNDS AND METHODS FOR SELECTIVE IMAGING AND / OR ABLATION
US9278124B2 (en) 2012-10-16 2016-03-08 Halozyme, Inc. Hypoxia and hyaluronan and markers thereof for diagnosis and monitoring of diseases and conditions and related methods
WO2015104589A1 (en) 2014-01-13 2015-07-16 Shanghai Lawring Biomedical Co., Ltd Dendrimer compositions, methods of synthesis, and uses thereof
WO2016047424A1 (ja) * 2014-09-25 2016-03-31 日本メジフィジックス株式会社 腎イメージング剤
US10695446B2 (en) 2015-05-01 2020-06-30 Vanderbilt University Composition and method for detecting hypoxia
US10695450B2 (en) 2016-07-26 2020-06-30 Laboratoires Cyclopharma Synthesis of a radioactive agent composition
CN106977501A (zh) * 2017-03-20 2017-07-25 华东师范大学 一种基于2‑硝基咪唑‑1‑烷基醇的低氧激活前药
FR3068695B1 (fr) * 2017-07-05 2019-08-16 Centre National De La Recherche Scientifique Composes utiles comme agent d'imagerie de l'hypoxie
US20200216486A1 (en) * 2017-09-19 2020-07-09 The Governors Of The University Of Alberta Markers, conjugates, compositions and methods for hypoxia imaging, mapping, and therapy
CN111372940A (zh) * 2017-09-19 2020-07-03 阿尔伯塔大学理事会 生物还原活化的化合物、其前药、放射性药物、组合物及其在包括癌症在内的低氧疾病的多模式治疗控制中的应用
CN115210229A (zh) 2020-01-03 2022-10-18 博格有限责任公司 多环酰胺作为治疗癌症的ube2k调节剂
CN111233821B (zh) * 2020-01-20 2022-12-27 上海交通大学医学院附属仁济医院 含3-羟基苯甲酸基团的新抗霉素衍生物及其制备方法和应用
CN114478489B (zh) * 2022-01-18 2023-04-28 中国科学院精密测量科学与技术创新研究院 一种氟-19修饰的硝基咪唑化合物及其衍生物的制备方法和应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5674693A (en) * 1994-03-18 1997-10-07 Natural Pharmacia International Inc. Derivatives of 2-nitro-imidazoles as hypoxic cell markers
US5721265A (en) * 1994-08-05 1998-02-24 Sri International Fluorinated 2-nitroimidazole analogs for detecting hypoxic tumor cells
DE60022058T2 (de) 1999-08-11 2006-06-01 Universite Catholique De Louvain Verfahren zur herstellung von [18f] radiomarkierten nitroimidazol-derivaten zum nachweis zellulärer hypoxie
CA2683433C (en) * 2007-04-05 2016-10-11 Siemens Medical Solutions Usa, Inc. Nitro-imidazole hypoxia imaging agents

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