JP2009542602A - 2−アミノベンズイミダゾール誘導体及び小コンダクタンスカルシウム依存性カリウムチャネルの調節剤としてのそれらの使用 - Google Patents

2−アミノベンズイミダゾール誘導体及び小コンダクタンスカルシウム依存性カリウムチャネルの調節剤としてのそれらの使用 Download PDF

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JP2009542602A
JP2009542602A JP2009517275A JP2009517275A JP2009542602A JP 2009542602 A JP2009542602 A JP 2009542602A JP 2009517275 A JP2009517275 A JP 2009517275A JP 2009517275 A JP2009517275 A JP 2009517275A JP 2009542602 A JP2009542602 A JP 2009542602A
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pharmaceutically acceptable
acceptable salt
alkyl
aminobenzimidazole
derivative according
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JP2009542602A5 (enExample
Inventor
ソーレンセン、ウルリック、スバン
エリクセン、ビルジット、エル.
ティウバー、レーネ
ペータース、ダン
ストロベイク、ドルテ
ヨハンセン、ティナ、ホルム
クリストファーセン、パレ
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ノイロサーチ アクティーゼルスカブ
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Publication of JP2009542602A5 publication Critical patent/JP2009542602A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
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JP2009517275A 2006-07-07 2007-07-05 2−アミノベンズイミダゾール誘導体及び小コンダクタンスカルシウム依存性カリウムチャネルの調節剤としてのそれらの使用 Abandoned JP2009542602A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81884106P 2006-07-07 2006-07-07
DKPA200600944 2006-07-07
PCT/EP2007/056826 WO2008003752A1 (en) 2006-07-07 2007-07-05 2 -amino benzimidazole derivatives and their use as modulators of small - conductance calcium -act ivated potassium channels

Publications (2)

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JP2009542602A true JP2009542602A (ja) 2009-12-03
JP2009542602A5 JP2009542602A5 (enExample) 2010-07-15

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JP2009517275A Abandoned JP2009542602A (ja) 2006-07-07 2007-07-05 2−アミノベンズイミダゾール誘導体及び小コンダクタンスカルシウム依存性カリウムチャネルの調節剤としてのそれらの使用

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US (1) US20100035951A1 (enExample)
EP (1) EP2041096A1 (enExample)
JP (1) JP2009542602A (enExample)
WO (1) WO2008003752A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010015037A1 (en) * 2008-08-08 2010-02-11 Howard Florey Institute Therapeutic methods and compositions
JP2013532149A (ja) * 2010-06-17 2013-08-15 ノバルティス アーゲー ピペリジニル置換1,3−ジヒドロ−ベンゾイミダゾール−2−イリデンアミン誘導体
CN102947274A (zh) * 2010-06-17 2013-02-27 诺瓦提斯公司 联苯基取代的1,3-二氢-苯并咪唑-2-亚基胺衍生物
CN104744375B (zh) * 2015-02-10 2017-09-19 南开大学 一种胍类ntr1小分子拮抗剂

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3981886A (en) * 1975-01-20 1976-09-21 E. R. Squibb & Sons, Inc. Amino-benzimidazole derivatives
US4004016A (en) * 1975-08-11 1977-01-18 E. R. Squibb & Sons, Inc. Amino-benzimidazole derivatives
DE69924493T2 (de) * 1998-07-02 2005-09-15 Neurosearch A/S Kaliumkanal-blockierende mittel
EP2319512A1 (en) * 2005-01-11 2011-05-11 NeuroSearch AS Novel 2-amino benzimidazole derivatives and their use as modulators of small-conductance calcium-activated potassium channels.
JP4751435B2 (ja) * 2008-10-09 2011-08-17 株式会社東芝 モータ磁極位置検出装置,モータ制御装置,モータ駆動システム及び洗濯機

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US20100035951A1 (en) 2010-02-11
WO2008003752A8 (en) 2008-03-13
WO2008003752A1 (en) 2008-01-10
EP2041096A1 (en) 2009-04-01

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