JP2008513426A5 - - Google Patents

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Publication number
JP2008513426A5
JP2008513426A5 JP2007531830A JP2007531830A JP2008513426A5 JP 2008513426 A5 JP2008513426 A5 JP 2008513426A5 JP 2007531830 A JP2007531830 A JP 2007531830A JP 2007531830 A JP2007531830 A JP 2007531830A JP 2008513426 A5 JP2008513426 A5 JP 2008513426A5
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JP
Japan
Prior art keywords
pharmacology
medicament
inhibition
diseases
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007531830A
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English (en)
Japanese (ja)
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JP2008513426A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/GB2005/003580 external-priority patent/WO2006032851A1/en
Publication of JP2008513426A publication Critical patent/JP2008513426A/ja
Publication of JP2008513426A5 publication Critical patent/JP2008513426A5/ja
Withdrawn legal-status Critical Current

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JP2007531830A 2004-09-20 2005-09-19 炎症の治療に有用なピラゾール化合物 Withdrawn JP2008513426A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US61095204P 2004-09-20 2004-09-20
US61708104P 2004-10-12 2004-10-12
PCT/GB2005/003580 WO2006032851A1 (en) 2004-09-20 2005-09-19 Pyrazole compounds useful in the treatment of inflammation

Publications (2)

Publication Number Publication Date
JP2008513426A JP2008513426A (ja) 2008-05-01
JP2008513426A5 true JP2008513426A5 (https=) 2008-11-20

Family

ID=35149494

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007531830A Withdrawn JP2008513426A (ja) 2004-09-20 2005-09-19 炎症の治療に有用なピラゾール化合物

Country Status (4)

Country Link
US (1) US20070225318A1 (https=)
EP (1) EP1794145A1 (https=)
JP (1) JP2008513426A (https=)
WO (1) WO2006032851A1 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080064682A1 (en) * 2004-07-01 2008-03-13 Daiichi Pharmaceutical Co., Ltd. Pyrazole Derivatives
US20090076275A1 (en) * 2007-09-19 2009-03-19 David Robert Bolin Diacylglycerol acyltransferase inhibitors
UA103272C2 (uk) 2009-12-11 2013-09-25 Ф. Хоффманн-Ля Рош Аг 2-аміно-5,5-дифтор-5,6-дигідро-4h-оксазини як інгібітори bace1 і/або bace2
US8772345B2 (en) 2011-08-03 2014-07-08 Southwest Research Institute Oximes for treatment of peripheral and central nervous system exposure to acetyl cholinesterase inhibitors
EP2628722A1 (en) * 2012-02-16 2013-08-21 Bayer CropScience AG CF3O-containing enaminoketones and their utilization for the preparation of CF3O-containing pyrazoles
EP2935248B1 (en) * 2012-12-21 2018-02-28 Plexxikon Inc. Compounds and methods for kinase modulation, and indications therefor
CN103012428A (zh) 2013-01-08 2013-04-03 中国药科大学 4-(五元杂环并嘧啶/吡啶取代)氨基-1H-3-吡唑甲酰胺类CDK/Aurora双重抑制剂及其用途
US9162983B2 (en) 2013-05-22 2015-10-20 Southwest Research Institute Reactivators of organophosphorous inhibited acetylcholinesterase
WO2016087593A1 (en) * 2014-12-05 2016-06-09 Syngenta Participations Ag Novel fungicidal quinolinylamidines
WO2021007477A1 (en) 2019-07-11 2021-01-14 E-Scape Bio, Inc. Indazoles and azaindazoles as lrrk2 inhibitors
CN115605460A (zh) 2020-04-29 2023-01-13 普莱希科公司（Us） 杂环化合物的合成
ES3048558A1 (es) * 2024-06-07 2025-12-10 Consejo Superior Investigacion Compuestos inhibidores de sgk1 y su uso para el tratamiento de enfermedades neurodegenerativas y/o cardiovasculares

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ATE306481T1 (de) * 1999-05-12 2005-10-15 Ortho Mcneil Pharm Inc Pyrazolecarboxamide zur behandlung von fettleibigkeit und anderen erkrankungen
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
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JP4465133B2 (ja) * 2001-02-08 2010-05-19 クミアイ化学工業株式会社 イソオキサゾリン誘導体及びこれを有効成分とする除草剤
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EP1421077A4 (en) 2001-08-31 2004-11-17 Univ Connecticut NEW PYRAZOLANALOGS ON CANNABINOID RECEPTORS
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TWI263497B (en) * 2002-03-29 2006-10-11 Lilly Co Eli Pyridinoylpiperidines as 5-HT1F agonists
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JP2006512314A (ja) * 2002-11-01 2006-04-13 バーテックス ファーマシューティカルズ インコーポレイテッド Ｊａｋインヒビターおよび他のプロテインキナーゼインヒビターとしての組成物の使用
US7488158B2 (en) * 2002-11-13 2009-02-10 Deka Products Limited Partnership Fluid transfer using devices with rotatable housings
EP1571671A4 (en) * 2002-12-13 2008-04-02 Matsushita Electric Industrial Co Ltd OPTICAL DATA DISTRIBUTION EQUIPMENT
US7429581B2 (en) * 2002-12-23 2008-09-30 Sanofi-Aventis Deutschland Gmbh Pyrazole-derivatives as factor Xa inhibitors
SE0300705D0 (sv) * 2003-03-14 2003-03-14 Biolipox Ab New compounds
EP1603897A1 (en) * 2003-03-14 2005-12-14 Biolipox AB Pyrazole compounds useful in the treatment of inflammation
US7429603B2 (en) * 2003-04-25 2008-09-30 3-Dimensional Pharmaceuticals, Inc. C-fms kinase inhibitors
GB0312609D0 (en) * 2003-06-02 2003-07-09 Astrazeneca Ab Novel compounds
US7659408B2 (en) 2003-08-07 2010-02-09 Merck Sharp & Dhome Corp. Pyrazole carboxamides as inhibitors of 11-β-hydroxysteroid dehydrogenase-1
WO2006032852A1 (en) * 2004-09-20 2006-03-30 Biolipox Ab Pyrazole compounds useful uin the treatment of inflammation
TW200800911A (en) * 2005-10-20 2008-01-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
TW200732320A (en) * 2005-10-31 2007-09-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
WO2007052000A1 (en) * 2005-11-01 2007-05-10 Biolipox Ab Pyrazoles useful in the treatment of inflammation

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