JP2006520373A - 炎症の治療に有用なピラゾール化合物 - Google Patents

炎症の治療に有用なピラゾール化合物 Download PDF

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JP2006520373A
JP2006520373A JP2006505952A JP2006505952A JP2006520373A JP 2006520373 A JP2006520373 A JP 2006520373A JP 2006505952 A JP2006505952 A JP 2006505952A JP 2006505952 A JP2006505952 A JP 2006505952A JP 2006520373 A JP2006520373 A JP 2006520373A
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methyl
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JP2006520373A5 (enExample
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アンダース ホールバーグ，
ウェスリー シャール，
マッツ ラーヘド，
クリストファー オロフソン，
ベンジャミン ペルクマン，
アンドレイ サニン，
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Biolipox AB
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Biolipox AB
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Publication of JP2006520373A5 publication Critical patent/JP2006520373A5/ja
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Otolaryngology (AREA)
JP2006505952A 2003-03-14 2004-03-12 炎症の治療に有用なピラゾール化合物 Withdrawn JP2006520373A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0300705A SE0300705D0 (sv) 2003-03-14 2003-03-14 New compounds
US48256303P 2003-06-26 2003-06-26
PCT/GB2004/001054 WO2004080999A1 (en) 2003-03-14 2004-03-12 Pyrazole compounds useful in the treatment of inflammation

Publications (2)

Publication Number Publication Date
JP2006520373A true JP2006520373A (ja) 2006-09-07
JP2006520373A5 JP2006520373A5 (enExample) 2007-04-19

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EP (1) EP1603897A1 (enExample)
JP (1) JP2006520373A (enExample)
WO (1) WO2004080999A1 (enExample)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010536926A (ja) * 2007-08-27 2010-12-02 ビーエーエスエフ ソシエタス・ヨーロピア 無脊椎動物系害虫を防除するためのピラゾール化合物
US8710056B2 (en) 2009-07-06 2014-04-29 Basf Se Pyridazine compounds for controlling invertebrate pests
US8729083B2 (en) 2008-09-24 2014-05-20 Basf Se Pyrazole compounds for controlling invertebrate pests
US9029639B2 (en) 2009-07-06 2015-05-12 Basf Se Pyridazine compounds for controlling invertebrate pests
US9125414B2 (en) 2009-07-24 2015-09-08 Basf Se Pyridine derivatives compounds for controlling invertebrate pests
CN110678456A (zh) * 2017-05-23 2020-01-10 隆德贝克拉荷亚研究中心有限公司 吡唑magl抑制剂

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008513426A (ja) * 2004-09-20 2008-05-01 バイオリポックス エービー 炎症の治療に有用なピラゾール化合物
EP1794130A1 (en) * 2004-09-20 2007-06-13 Biolipox AB Pyrazole compounds useful in the treatment of inflammation
CA2620899A1 (en) * 2005-10-12 2007-04-19 Biolipox Ab Benzoxazoles useful in the treatment of inflammation
WO2007042817A1 (en) * 2005-10-13 2007-04-19 Biolipox Ab Naphthalene-disulfonamides useful for the treatment of inflammation
TW200800911A (en) * 2005-10-20 2008-01-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
EP1943234A1 (en) * 2005-10-31 2008-07-16 Biolipox AB Triazole compounds as lipoxygenase inhibitors
TW200732320A (en) * 2005-10-31 2007-09-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
WO2007052000A1 (en) * 2005-11-01 2007-05-10 Biolipox Ab Pyrazoles useful in the treatment of inflammation
WO2008001079A1 (en) * 2006-06-27 2008-01-03 Biolipox Ab Methods for identifying modulators of eoxin formation
WO2008129276A1 (en) * 2007-04-19 2008-10-30 Boehringer Ingelheim International Gmbh Disulfonamides useful in the treatment of inflammation
WO2008129280A1 (en) * 2007-04-20 2008-10-30 Biolipox Ab Pyrazoles useful in the treatment of inflammation
CA2684105C (en) 2007-05-03 2011-09-06 Pfizer Limited Pyridine derivatives
WO2008135767A1 (en) * 2007-05-07 2008-11-13 Biolipox Ab New triazole compounds useful in the treatment of inflammation
CN102223798A (zh) 2008-09-24 2011-10-19 巴斯夫欧洲公司 用于防治无脊椎动物害虫的吡唑化合物
WO2012031383A1 (zh) * 2010-09-06 2012-03-15 中国科学院广州生物医药与健康研究院 酰胺类化合物
WO2021072487A1 (en) * 2019-10-15 2021-04-22 TroBio Therapeutics Pty Ltd Sulfonamide compounds and the use thereof in the treatment of cancer

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP042397A0 (en) * 1997-11-18 1997-12-11 Fujisawa Pharmaceutical Co., Ltd. 5-arylpyrazole compounds

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010536926A (ja) * 2007-08-27 2010-12-02 ビーエーエスエフ ソシエタス・ヨーロピア 無脊椎動物系害虫を防除するためのピラゾール化合物
US8642597B2 (en) 2007-08-27 2014-02-04 Basf Se Pyrazole compounds for controlling invertebrate pests
US9204647B2 (en) 2007-08-27 2015-12-08 Basf Se Pyrazole compounds for controlling invertebrate pests
US8729083B2 (en) 2008-09-24 2014-05-20 Basf Se Pyrazole compounds for controlling invertebrate pests
US9375008B2 (en) 2008-09-24 2016-06-28 Basf Se Pyrazole compounds for controlling invertebrate pests
US8710056B2 (en) 2009-07-06 2014-04-29 Basf Se Pyridazine compounds for controlling invertebrate pests
US9029639B2 (en) 2009-07-06 2015-05-12 Basf Se Pyridazine compounds for controlling invertebrate pests
US9125414B2 (en) 2009-07-24 2015-09-08 Basf Se Pyridine derivatives compounds for controlling invertebrate pests
CN110678456A (zh) * 2017-05-23 2020-01-10 隆德贝克拉荷亚研究中心有限公司 吡唑magl抑制剂
CN110678456B (zh) * 2017-05-23 2023-05-02 H.隆德贝克有限公司 吡唑magl抑制剂

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