JP2006518328A - 複素環選択的アンドロゲン受容体調節剤及びその使用方法 - Google Patents
複素環選択的アンドロゲン受容体調節剤及びその使用方法 Download PDFInfo
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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/84—Nitriles
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41817302P | 2002-10-15 | 2002-10-15 | |
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| JP2008501800A (ja) * | 2004-06-07 | 2008-01-24 | メルク エンド カムパニー インコーポレーテッド | アンドロゲン受容体調節剤としてのｎ−（２−ベンジル）−２−フェニルブタンアミド |
| JP2014532686A (ja) * | 2011-11-04 | 2014-12-08 | ガルデルマ・リサーチ・アンド・デヴェロップメント | Ｎ−（ピリド−４−イル）アミドおよびｎ−（ピリミジン−４−イル）アミド、ならびにそれらの医薬的および美容的使用関連出願 |
| JP2019522644A (ja) * | 2016-06-10 | 2019-08-15 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
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- 2003-10-14 CA CA002501867A patent/CA2501867A1/en not_active Abandoned
- 2003-10-14 CN CNA2003801061407A patent/CN1726193A/zh active Pending
- 2003-10-14 EP EP03777597A patent/EP1562906A4/en not_active Withdrawn
- 2003-10-14 US US10/683,125 patent/US7214693B2/en not_active Expired - Fee Related
- 2003-10-14 AU AU2003287076A patent/AU2003287076C1/en not_active Ceased
- 2003-10-14 JP JP2004544889A patent/JP2006518328A/ja active Pending
- 2003-10-14 WO PCT/US2003/032510 patent/WO2004035737A2/en not_active Ceased
- 2003-10-15 TW TW092128552A patent/TW200502249A/zh unknown
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2007
- 2007-03-22 US US11/723,957 patent/US20070265290A1/en not_active Abandoned
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| JPS5933250A (ja) * | 1982-07-23 | 1984-02-23 | インペリアル・ケミカル・インダストリ−ズ・ピ−エルシ− | アシルアニリド、その製法及び抗アンドロゲン作用を有する医薬又は獣医薬組成物 |
| JP2002502385A (ja) * | 1997-05-30 | 2002-01-22 | シエーリング アクチエンゲゼルシヤフト | ゲスターゲン及びアンドロゲン混合作用を有する非ステロイド系（複素）環式置換アシルアニリド |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007538094A (ja) * | 2004-05-20 | 2007-12-27 | ユニバーシティ・オブ・テネシー・リサーチ・ファウンデーション | 選択的アンドロゲン受容体調節剤化合物の代謝物及びその使用方法 |
| JP2008501800A (ja) * | 2004-06-07 | 2008-01-24 | メルク エンド カムパニー インコーポレーテッド | アンドロゲン受容体調節剤としてのｎ−（２−ベンジル）−２−フェニルブタンアミド |
| JP4881865B2 (ja) * | 2004-06-07 | 2012-02-22 | メルク・シャープ・エンド・ドーム・コーポレイション | アンドロゲン受容体調節剤としてのｎ−（２−ベンジル）−２−フェニルブタンアミド |
| JP2014532686A (ja) * | 2011-11-04 | 2014-12-08 | ガルデルマ・リサーチ・アンド・デヴェロップメント | Ｎ−（ピリド−４−イル）アミドおよびｎ−（ピリミジン−４−イル）アミド、ならびにそれらの医薬的および美容的使用関連出願 |
| JP2019522644A (ja) * | 2016-06-10 | 2019-08-15 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
| JP2021138780A (ja) * | 2016-06-10 | 2021-09-16 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
| JP7382987B2 (ja) | 2016-06-10 | 2023-11-17 | ユニバーシティ オブ テネシー リサーチ ファウンデーション | 選択的アンドロゲン受容体分解剤（ｓａｒｄ）リガンドおよびその使用方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20070265290A1 (en) | 2007-11-15 |
| AU2003287076C1 (en) | 2010-03-04 |
| CA2501867A1 (en) | 2004-04-29 |
| EP1562906A2 (en) | 2005-08-17 |
| AU2003287076A1 (en) | 2004-05-04 |
| AU2003287076A2 (en) | 2004-05-04 |
| AU2009202683A1 (en) | 2009-07-23 |
| WO2004035737A3 (en) | 2004-09-10 |
| TW200502249A (en) | 2005-01-16 |
| CN1726193A (zh) | 2006-01-25 |
| WO2004035737A2 (en) | 2004-04-29 |
| US7214693B2 (en) | 2007-05-08 |
| US20040138244A1 (en) | 2004-07-15 |
| AU2003287076B2 (en) | 2009-04-02 |
| EP1562906A4 (en) | 2009-12-02 |
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