JP2006511491A - 女性の性的欲求および性的反応性を高めるための即放性局所薬学的処方物 - Google Patents
女性の性的欲求および性的反応性を高めるための即放性局所薬学的処方物 Download PDFInfo
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- JP2006511491A JP2006511491A JP2004547084A JP2004547084A JP2006511491A JP 2006511491 A JP2006511491 A JP 2006511491A JP 2004547084 A JP2004547084 A JP 2004547084A JP 2004547084 A JP2004547084 A JP 2004547084A JP 2006511491 A JP2006511491 A JP 2006511491A
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- Prior art keywords
- phosphodiesterase inhibitor
- sexual
- pharmaceutical formulation
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- JOSMPBVYYKRYLG-OLZOCXBDSA-N CN(C1=N[C@H](CCC2)[C@H]2N1c1c2[nH]c(Cc3ccc(C(F)(F)F)cc3)n1)C2=O Chemical compound CN(C1=N[C@H](CCC2)[C@H]2N1c1c2[nH]c(Cc3ccc(C(F)(F)F)cc3)n1)C2=O JOSMPBVYYKRYLG-OLZOCXBDSA-N 0.000 description 1
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/15—Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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- A61K31/28—Compounds containing heavy metals
- A61K31/295—Iron group metal compounds
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- A61K31/4164—1,3-Diazoles
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- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Reproductive Health (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Gynecology & Obstetrics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Dispersion Chemistry (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/279,039 US20040014761A1 (en) | 1997-10-28 | 2002-10-22 | Treatment of female sexual dysfunction with phosphodiesterase inhibitors |
| PCT/US2003/033642 WO2004037262A2 (en) | 2002-10-22 | 2003-10-22 | Immediate release topical pharmaceutical formulation for enhancement of female sexual desire and responsiveness |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006511491A true JP2006511491A (ja) | 2006-04-06 |
| JP2006511491A5 JP2006511491A5 (enExample) | 2006-11-30 |
Family
ID=32174580
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004547084A Pending JP2006511491A (ja) | 2002-10-22 | 2003-10-22 | 女性の性的欲求および性的反応性を高めるための即放性局所薬学的処方物 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20040014761A1 (enExample) |
| EP (1) | EP1562602A2 (enExample) |
| JP (1) | JP2006511491A (enExample) |
| AU (1) | AU2003284877A1 (enExample) |
| CA (1) | CA2503391A1 (enExample) |
| WO (1) | WO2004037262A2 (enExample) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014504592A (ja) * | 2010-12-29 | 2014-02-24 | ストラテジック サイエンス アンド テクノロジーズ, エルエルシー | 勃起不全および他の適応症の処置 |
| US9457092B2 (en) | 2009-06-24 | 2016-10-04 | Strategic Science & Technologies, Llc | Delivery of ibuprofen and other compounds |
| JP2018508585A (ja) * | 2015-03-16 | 2018-03-29 | ミレカ メディシンズ ゲーエムベーハー | cGMPアナログの標的化されたリポソーム送達 |
| WO2023048174A1 (ja) * | 2021-09-22 | 2023-03-30 | テイカ製薬株式会社 | 角膜疾患治療剤 |
| US11684624B2 (en) | 2009-06-24 | 2023-06-27 | Strategic Science & Technologies, Llc | Treatment of erectile dysfunction and other indications |
| US12138268B2 (en) | 2009-06-24 | 2024-11-12 | Strategic Science & Technologies, Llc | Treatment of erectile dysfunction and other indications |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0222522D0 (en) | 2002-09-27 | 2002-11-06 | Controlled Therapeutics Sct | Water-swellable polymers |
| BRPI0406634A (pt) * | 2003-01-23 | 2005-12-06 | Shire Holding Ag | Uso de um anagrelìdeo, anagrelìdeo na forma de base, ou um sal farmaceuticamente aceitável do anagrelìdeo, composição farmacêutica não-oral, e dispositivo médido para administração transdérmica |
| MX347237B (es) | 2004-05-11 | 2017-04-20 | Eb Ip Lybrido B V | Formulaciones farmaceuticas y usos de las mismas en el tratamiento de la disfuncion sexual femenina. |
| US20060030574A1 (en) * | 2004-08-04 | 2006-02-09 | Shire Holdings Ag | Quinazoline derivatives useful for the treatment of peripheral arterial disease and as phosphodiesterase inhibitors |
| US7700608B2 (en) * | 2004-08-04 | 2010-04-20 | Shire Holdings Ag | Quinazoline derivatives and their use in the treatment of thrombocythemia |
| GB0417401D0 (en) | 2004-08-05 | 2004-09-08 | Controlled Therapeutics Sct | Stabilised prostaglandin composition |
| PT1802277E (pt) * | 2004-10-18 | 2010-04-01 | Polymun Scient Immunbio Forsch | Composição lipossomal contendo um ingrediente activo para relaxar a musculatura lisa, produção desta composição e a sua aplicação terapêutica |
| SG155258A1 (en) * | 2004-10-20 | 2009-09-30 | Endorech Inc | Sex steroid precursors alone or in combination with a selective estrogen receptor modulator and/or with estrogens and/or a type 5 cgmp phosphodiesterase inhibitor for the prevention and treatment of vaginal dryness and sexual dysfunction in postmenopausa |
| BRPI0518829A2 (pt) * | 2004-12-06 | 2008-12-09 | Avigen Inc | mÉtodo para o tratamento de dor neuropÁtica e sÍndromes associadas |
| EP1790343A1 (en) * | 2005-11-11 | 2007-05-30 | Emotional Brain B.V. | Pharmaceuticals formulations and uses thereof in the treatment of female sexual dysfunction |
| GB0613333D0 (en) | 2006-07-05 | 2006-08-16 | Controlled Therapeutics Sct | Hydrophilic polyurethane compositions |
| JP2009542648A (ja) * | 2006-07-07 | 2009-12-03 | テバ ファーマシューティカル インダストリーズ リミティド | タダラフィル及び少なくとも1種の担体を含んでなる固体組成物 |
| GB0613638D0 (en) | 2006-07-08 | 2006-08-16 | Controlled Therapeutics Sct | Polyurethane elastomers |
| GB0620685D0 (en) * | 2006-10-18 | 2006-11-29 | Controlled Therapeutics Sct | Bioresorbable polymers |
| EP1925307A1 (en) | 2006-11-03 | 2008-05-28 | Emotional Brain B.V. | Use of 3-alpha-androstanediol in the treatment of sexual dysfunction |
| US8304420B2 (en) | 2006-11-28 | 2012-11-06 | Shire Llc | Substituted quinazolines for reducing platelet count |
| US7910597B2 (en) * | 2006-11-28 | 2011-03-22 | Shire Llc | Substituted quinazolines |
| US20080181876A1 (en) * | 2007-01-30 | 2008-07-31 | Johnson Kirk W | Methods for treating acute and subchronic pain |
| US20080287402A1 (en) * | 2007-05-03 | 2008-11-20 | Johnson Kirk W | Use of a glial attenuator to prevent amplified pain responses caused by glial priming |
| DE102007028869A1 (de) | 2007-06-22 | 2008-12-24 | Ratiopharm Gmbh | Verfahren zur Herstellung eines Arzneimittels enthaltend Tadalafil |
| US8268806B2 (en) * | 2007-08-10 | 2012-09-18 | Endorecherche, Inc. | Pharmaceutical compositions |
| US10561656B2 (en) | 2011-06-10 | 2020-02-18 | Intra-Cellular Therapies, Inc. | Organic compounds |
| ES2395801B1 (es) | 2011-06-23 | 2014-06-06 | María Carmen PARDINA PALLEJÀ | "pentoxifilina por vía transvaginal para el tratamiento de la infertilidad" |
| US20170239175A1 (en) * | 2016-02-19 | 2017-08-24 | FSD Pharma Co, LLC | Topical anorgasmia therapy |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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-
2002
- 2002-10-22 US US10/279,039 patent/US20040014761A1/en not_active Abandoned
-
2003
- 2003-10-22 AU AU2003284877A patent/AU2003284877A1/en not_active Abandoned
- 2003-10-22 CA CA002503391A patent/CA2503391A1/en not_active Abandoned
- 2003-10-22 EP EP03779198A patent/EP1562602A2/en not_active Withdrawn
- 2003-10-22 JP JP2004547084A patent/JP2006511491A/ja active Pending
- 2003-10-22 WO PCT/US2003/033642 patent/WO2004037262A2/en not_active Ceased
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Also Published As
| Publication number | Publication date |
|---|---|
| US20040014761A1 (en) | 2004-01-22 |
| AU2003284877A1 (en) | 2004-05-13 |
| WO2004037262A2 (en) | 2004-05-06 |
| CA2503391A1 (en) | 2004-05-06 |
| EP1562602A2 (en) | 2005-08-17 |
| WO2004037262A3 (en) | 2004-08-12 |
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