JP2006510654A - 糖尿病を処置する方法 - Google Patents
糖尿病を処置する方法 Download PDFInfo
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- JP2006510654A JP2006510654A JP2004558236A JP2004558236A JP2006510654A JP 2006510654 A JP2006510654 A JP 2006510654A JP 2004558236 A JP2004558236 A JP 2004558236A JP 2004558236 A JP2004558236 A JP 2004558236A JP 2006510654 A JP2006510654 A JP 2006510654A
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- Prior art keywords
- alkyl
- fluorophenyl
- imidazole
- aryl
- diabetes
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| WO2007075896A2 (en) * | 2005-12-22 | 2007-07-05 | Kemia, Inc. | Heterocyclic cytokine inhibitors |
| JP2014531425A (ja) * | 2011-09-02 | 2014-11-27 | ザ トラスティーズ オブ コロンビア ユニヴァーシティ イン ザ シティ オブ ニューヨーク | 肥満の代謝異常を治療するためのＣａＭＫＩＩ、ＩＰ３Ｒ、カルシニューリン、ｐ３８、およびＭＫ２／３阻害剤 |
| ES2927715T3 (es) | 2017-10-05 | 2022-11-10 | Fulcrum Therapeutics Inc | Inhibidores de la quinasa p38 reducen la expresión de dux4 y de los genes que le siguen para el tratamiento de la FSHD |
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2003
- 2003-12-05 AU AU2003299652A patent/AU2003299652A1/en not_active Abandoned
- 2003-12-05 US US10/728,665 patent/US20040171659A1/en not_active Abandoned
- 2003-12-05 JP JP2004558236A patent/JP2006510654A/ja active Pending
- 2003-12-05 CA CA002511763A patent/CA2511763A1/en not_active Abandoned
- 2003-12-05 WO PCT/US2003/040140 patent/WO2004053107A2/en not_active Ceased
- 2003-12-05 EP EP03799936A patent/EP1583535A4/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004053107A3 (en) | 2004-10-07 |
| AU2003299652A1 (en) | 2004-06-30 |
| US20040171659A1 (en) | 2004-09-02 |
| EP1583535A2 (en) | 2005-10-12 |
| EP1583535A4 (en) | 2008-03-19 |
| WO2004053107A2 (en) | 2004-06-24 |
| AU2003299652A8 (en) | 2004-06-30 |
| CA2511763A1 (en) | 2004-06-24 |
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