JP2006500315A5 - - Google Patents
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- Publication number
- JP2006500315A5 JP2006500315A5 JP2003559504A JP2003559504A JP2006500315A5 JP 2006500315 A5 JP2006500315 A5 JP 2006500315A5 JP 2003559504 A JP2003559504 A JP 2003559504A JP 2003559504 A JP2003559504 A JP 2003559504A JP 2006500315 A5 JP2006500315 A5 JP 2006500315A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- hydrogen
- heterocyclic
- alkylcarbonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 *c(c(*)c1*)c(*)c(**C2(P)IN(*)*)c1C2=* Chemical compound *c(c(*)c1*)c(*)c(**C2(P)IN(*)*)c1C2=* 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/043,848 US20030134835A1 (en) | 2002-01-11 | 2002-01-11 | Histamine-3 receptor ligands for diabetes conditions |
| US10/326,546 US20030153548A1 (en) | 2002-01-11 | 2002-12-23 | Histamine-3 receptor ligands for diabetic conditions |
| PCT/US2003/000733 WO2003059342A1 (en) | 2002-01-11 | 2003-01-10 | Histamine-3 receptor ligands for diabetic conditions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006500315A JP2006500315A (ja) | 2006-01-05 |
| JP2006500315A5 true JP2006500315A5 (https=) | 2006-02-16 |
Family
ID=26720877
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003559504A Pending JP2006500315A (ja) | 2002-01-11 | 2003-01-10 | 糖尿病状態に用いるヒスタミン−３受容体リガンド |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20050113435A1 (https=) |
| EP (1) | EP1474132A1 (https=) |
| JP (1) | JP2006500315A (https=) |
| AU (1) | AU2003235687A1 (https=) |
| CA (1) | CA2473232C (https=) |
| MX (1) | MXPA04006777A (https=) |
| PL (1) | PL373586A1 (https=) |
| WO (1) | WO2003059342A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6620839B2 (en) * | 2000-07-13 | 2003-09-16 | Abbott Laboratories | 1,3-disubstituted and 1,3,3-trisubstituted pyrrolidines as histamine-3 receptor ligands and their therapeutic applications |
| US6822101B2 (en) | 2002-09-16 | 2004-11-23 | Abbott Laboratories | Process for preparing amine-substituted benzofurans |
| WO2004024707A2 (en) * | 2002-09-16 | 2004-03-25 | Abbott Laboratories | Process for preparing amine type substituted benzofurans |
| WO2005009471A1 (en) * | 2003-07-28 | 2005-02-03 | Osaka Industrial Promotion Organization | Composition for lowering blood-sugar level |
| US7435837B2 (en) | 2003-10-24 | 2008-10-14 | Wyeth | Dihydrobenzofuranyl alkanamine derivatives and methods for using same |
| EP1717233A1 (en) * | 2005-04-29 | 2006-11-02 | Bioprojet | Histamine H3-receptor ligands and their therapeutic application |
| EP1717234A1 (en) * | 2005-04-29 | 2006-11-02 | Bioprojet | Phenoxypropylpiperidines and -pyrrolidines and their use as histamine H3-receptor ligands |
| EP1717235A3 (en) * | 2005-04-29 | 2007-02-28 | Bioprojet | Phenoxypropylpiperidines and -pyrrolidines and their use as histamine H3-receptor ligands |
| FR2903904A1 (fr) * | 2006-07-21 | 2008-01-25 | Bioprojet Soc Civ Ile | Association de modafinil et d'un antagoniste ou agoniste inverse du recepteur h3 |
| JP2010520199A (ja) * | 2007-03-02 | 2010-06-10 | シェーリング コーポレイション | ピペリジン誘導体およびその使用方法 |
| WO2008108958A2 (en) * | 2007-03-02 | 2008-09-12 | Schering Corporation | Benzimidazole derivatives and methods of use thereof |
| WO2022113008A1 (en) | 2020-11-27 | 2022-06-02 | Richter Gedeon Nyrt. | Histamine h3 receptor antagonists/inverse agonists for the treatment of autism spectrum disorder |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4096331A (en) * | 1976-12-28 | 1978-06-20 | A. H. Robins Company, Incorporated | 1-Substituted-3-aminoethoxypyrrolidines |
| GB2056441B (en) * | 1979-07-26 | 1983-07-06 | Kyowa Hakko Kogyo Kk | Derivatives of benzo(b)furan and pharmaceutical compositions containing them |
| US4452986A (en) * | 1982-06-08 | 1984-06-05 | The Upjohn Company | Imidazolyl-substituted benzofurans |
| US4447620A (en) * | 1982-06-08 | 1984-05-08 | The Upjohn Company | Imidazolyl-substituted benzothiophenes |
| NZ270418A (en) * | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
| EP0977753A1 (en) * | 1997-12-02 | 2000-02-09 | Dr. Reddy's Research Foundation | Azolidinediones useful for the treatment of diabetes, dyslipidemia and hypertension |
| US6136559A (en) * | 1998-10-07 | 2000-10-24 | Ortho Pharmaceutical Corporation | DNA encoding as human histamine receptor of the H3 subtype |
| AU3957600A (en) * | 1999-04-26 | 2000-11-10 | Boehringer Ingelheim International Gmbh | Piperidyl-imidazole derivatives, their preparations and therapeutic uses |
| US6437147B1 (en) * | 2000-03-17 | 2002-08-20 | Novo Nordisk | Imidazole compounds |
| AU2001244087A1 (en) * | 2000-03-17 | 2001-09-24 | Boehringer Ingelheim International G.M.B.H | Condensed imidazoles as histamine h3 receptor ligands |
| US6620839B2 (en) * | 2000-07-13 | 2003-09-16 | Abbott Laboratories | 1,3-disubstituted and 1,3,3-trisubstituted pyrrolidines as histamine-3 receptor ligands and their therapeutic applications |
| US6316475B1 (en) * | 2000-11-17 | 2001-11-13 | Abbott Laboratories | Aminoalkoxybiphenylcarboxamides as histamine-3 receptor ligands and their therapeutic applications |
| CN101444496B (zh) * | 2001-06-12 | 2011-04-13 | 维尔斯达医疗公司 | 用于治疗代谢失调的化合物 |
| CN1642599A (zh) * | 2002-02-27 | 2005-07-20 | 辉瑞产品公司 | Acc抑制剂 |
-
2003
- 2003-01-10 EP EP03729628A patent/EP1474132A1/en not_active Withdrawn
- 2003-01-10 JP JP2003559504A patent/JP2006500315A/ja active Pending
- 2003-01-10 AU AU2003235687A patent/AU2003235687A1/en not_active Abandoned
- 2003-01-10 PL PL03373586A patent/PL373586A1/xx not_active Application Discontinuation
- 2003-01-10 MX MXPA04006777A patent/MXPA04006777A/es active IP Right Grant
- 2003-01-10 CA CA2473232A patent/CA2473232C/en not_active Expired - Fee Related
- 2003-01-10 WO PCT/US2003/000733 patent/WO2003059342A1/en not_active Ceased
-
2004
- 2004-10-06 US US10/959,799 patent/US20050113435A1/en not_active Abandoned
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