JP2005538103A - アムロジピンの有機酸塩 - Google Patents
アムロジピンの有機酸塩 Download PDFInfo
- Publication number
- JP2005538103A JP2005538103A JP2004524369A JP2004524369A JP2005538103A JP 2005538103 A JP2005538103 A JP 2005538103A JP 2004524369 A JP2004524369 A JP 2004524369A JP 2004524369 A JP2004524369 A JP 2004524369A JP 2005538103 A JP2005538103 A JP 2005538103A
- Authority
- JP
- Japan
- Prior art keywords
- amlodipine
- camphorsulfonate
- camphor
- acid
- camphor sulfonate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/86—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR1020020044856A KR20040011751A (ko) | 2002-07-30 | 2002-07-30 | 암로디핀의 유기산염 |
PCT/KR2003/001522 WO2004011432A1 (en) | 2002-07-30 | 2003-07-30 | Organic acid salt of amlodipine |
Publications (1)
Publication Number | Publication Date |
---|---|
JP2005538103A true JP2005538103A (ja) | 2005-12-15 |
Family
ID=31185754
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2004524369A Pending JP2005538103A (ja) | 2002-07-30 | 2003-07-30 | アムロジピンの有機酸塩 |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1549616A4 (ko) |
JP (1) | JP2005538103A (ko) |
KR (1) | KR20040011751A (ko) |
CN (1) | CN1678583A (ko) |
AU (1) | AU2003247208A1 (ko) |
BR (1) | BR0313076A (ko) |
MX (1) | MXPA05001241A (ko) |
WO (1) | WO2004011432A1 (ko) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100913791B1 (ko) * | 2006-07-21 | 2009-08-26 | 한미약품 주식회사 | (s)-(-)-암로디핀 캠실레이트 또는 이의 수화물 및 이를함유하는 약학적 조성물 |
KR100821688B1 (ko) | 2006-08-10 | 2008-04-11 | (주)유케이케미팜 | 암로디핀 라셈화물의 입체이성질체의 분리방법과 그의친수성 약물 및 그의 제조방법 |
PL2534153T3 (pl) | 2010-02-12 | 2017-08-31 | Pfizer Inc. | Sole i polimorfy 8-fluoro-2-{4-[(metyloamino}metylo]fenylo}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-onu |
CN101972254B (zh) * | 2010-09-28 | 2012-05-30 | 石药集团欧意药业有限公司 | 一种左旋氨氯地平或其可药用盐固体制剂及其制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK161312C (da) * | 1982-03-11 | 1991-12-09 | Pfizer | Analogifremgangsmaade til fremstilling af 2-aminoalkoxymethyl-4-phenyl-6-methyl-1,4-dihydropyridin-3,5-dicarboxylsyreestere eller syreadditionssalte deraf samt phthalimidoderivater til anvendelse som udgangsmateriale ved fremgangsmaaden |
GB8608335D0 (en) * | 1986-04-04 | 1986-05-08 | Pfizer Ltd | Pharmaceutically acceptable salts |
GB8710493D0 (en) * | 1987-05-02 | 1987-06-03 | Pfizer Ltd | Dihydropyridines |
US6057344A (en) * | 1991-11-26 | 2000-05-02 | Sepracor, Inc. | Methods for treating hypertension, and angina using optically pure (-) amlodipine |
KR100452491B1 (ko) * | 2001-03-29 | 2004-10-12 | 한미약품 주식회사 | 신규한 결정형 암로디핀 캠실레이트 염 및 그의 제조방법 |
-
2002
- 2002-07-30 KR KR1020020044856A patent/KR20040011751A/ko not_active Application Discontinuation
-
2003
- 2003-07-30 WO PCT/KR2003/001522 patent/WO2004011432A1/en active Application Filing
- 2003-07-30 BR BR0313076-2A patent/BR0313076A/pt not_active IP Right Cessation
- 2003-07-30 MX MXPA05001241A patent/MXPA05001241A/es unknown
- 2003-07-30 AU AU2003247208A patent/AU2003247208A1/en not_active Abandoned
- 2003-07-30 EP EP03771480A patent/EP1549616A4/en not_active Withdrawn
- 2003-07-30 CN CNA038208768A patent/CN1678583A/zh active Pending
- 2003-07-30 JP JP2004524369A patent/JP2005538103A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
MXPA05001241A (es) | 2005-06-08 |
KR20040011751A (ko) | 2004-02-11 |
EP1549616A4 (en) | 2006-10-18 |
WO2004011432A1 (en) | 2004-02-05 |
EP1549616A1 (en) | 2005-07-06 |
CN1678583A (zh) | 2005-10-05 |
BR0313076A (pt) | 2005-06-28 |
AU2003247208A1 (en) | 2004-02-16 |
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Legal Events
Date | Code | Title | Description |
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A131 | Notification of reasons for refusal |
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A711 | Notification of change in applicant |
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A131 | Notification of reasons for refusal |
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A02 | Decision of refusal |
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