JP2004522796A - Ｈ＋，ｋ＋−ａｔｐアーゼ阻害剤を含む微粒子の製造方法 - Google Patents
Ｈ＋，ｋ＋−ａｔｐアーゼ阻害剤を含む微粒子の製造方法 Download PDFInfo
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- JP2004522796A JP2004522796A JP2002571030A JP2002571030A JP2004522796A JP 2004522796 A JP2004522796 A JP 2004522796A JP 2002571030 A JP2002571030 A JP 2002571030A JP 2002571030 A JP2002571030 A JP 2002571030A JP 2004522796 A JP2004522796 A JP 2004522796A
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Disintegrating Or Milling (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- General Preparation And Processing Of Foods (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0100822A SE0100822D0 (sv) | 2001-03-09 | 2001-03-09 | Method II to obtain microparticles |
| PCT/SE2002/000400 WO2002072071A1 (en) | 2001-03-09 | 2002-03-06 | Method to obtain microparticles containing a h+, k+ -atp-ase inhibitor |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004522796A true JP2004522796A (ja) | 2004-07-29 |
| JP2004522796A5 JP2004522796A5 (enExample) | 2005-12-22 |
Family
ID=20283293
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002571030A Pending JP2004522796A (ja) | 2001-03-09 | 2002-03-06 | Ｈ＋，ｋ＋−ａｔｐアーゼ阻害剤を含む微粒子の製造方法 |
Country Status (21)
| Country | Link |
|---|---|
| US (2) | US20040101565A1 (enExample) |
| EP (1) | EP1370243B1 (enExample) |
| JP (1) | JP2004522796A (enExample) |
| KR (1) | KR20030081506A (enExample) |
| CN (1) | CN1507343A (enExample) |
| AT (1) | ATE400253T1 (enExample) |
| AU (1) | AU2002235101B8 (enExample) |
| BR (1) | BR0207827A (enExample) |
| CA (1) | CA2440163A1 (enExample) |
| DE (1) | DE60227488D1 (enExample) |
| DK (1) | DK1370243T3 (enExample) |
| ES (1) | ES2307722T3 (enExample) |
| IL (1) | IL157467A0 (enExample) |
| MX (1) | MXPA03007887A (enExample) |
| NO (1) | NO20033966L (enExample) |
| NZ (1) | NZ527997A (enExample) |
| PT (1) | PT1370243E (enExample) |
| SE (1) | SE0100822D0 (enExample) |
| SI (1) | SI1370243T1 (enExample) |
| WO (1) | WO2002072071A1 (enExample) |
| ZA (1) | ZA200306614B (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009534441A (ja) * | 2006-04-24 | 2009-09-24 | メファ・アクチェンゲゼルシャフト | ピリジルメチルスルフィニルベンズイミダゾールのための経口速放医薬製剤 |
| WO2021153525A1 (ja) * | 2020-01-27 | 2021-08-05 | 東和薬品株式会社 | エソメプラゾール経口製剤およびその製造方法 |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20060159756A1 (en) * | 1999-09-10 | 2006-07-20 | Brita Sjoblom | Method to obtain microparticles containing an H+,K+-ATP-ASE inhibitor |
| SE0100823D0 (sv) * | 2001-03-09 | 2001-03-09 | Astrazeneca Ab | Method I to obtain microparticles |
| US8067032B2 (en) | 2000-12-22 | 2011-11-29 | Baxter International Inc. | Method for preparing submicron particles of antineoplastic agents |
| US6977085B2 (en) | 2000-12-22 | 2005-12-20 | Baxter International Inc. | Method for preparing submicron suspensions with polymorph control |
| US6607784B2 (en) | 2000-12-22 | 2003-08-19 | Baxter International Inc. | Microprecipitation method for preparing submicron suspensions |
| US9700866B2 (en) | 2000-12-22 | 2017-07-11 | Baxter International Inc. | Surfactant systems for delivery of organic compounds |
| US6884436B2 (en) | 2000-12-22 | 2005-04-26 | Baxter International Inc. | Method for preparing submicron particle suspensions |
| US6951656B2 (en) | 2000-12-22 | 2005-10-04 | Baxter International Inc. | Microprecipitation method for preparing submicron suspensions |
| US7193084B2 (en) | 2000-12-22 | 2007-03-20 | Baxter International Inc. | Polymorphic form of itraconazole |
| SE0100824D0 (sv) * | 2001-03-09 | 2001-03-09 | Astrazeneca Ab | Method III to obtain microparticles |
| SE0100822D0 (sv) * | 2001-03-09 | 2001-03-09 | Astrazeneca Ab | Method II to obtain microparticles |
| CN1558755A (zh) | 2001-09-26 | 2004-12-29 | ���ع��ʹ�˾ | 通过分散和除去溶剂或液相制备亚微米大小的纳米颗粒 |
| US20060003012A9 (en) | 2001-09-26 | 2006-01-05 | Sean Brynjelsen | Preparation of submicron solid particle suspensions by sonication of multiphase systems |
| US7112340B2 (en) | 2001-10-19 | 2006-09-26 | Baxter International Inc. | Compositions of and method for preparing stable particles in a frozen aqueous matrix |
| CA2518780C (en) | 2003-03-12 | 2014-05-13 | Takeda Pharmaceutical Company Limited | Drug composition having active ingredient adhered at high concentration to spherical core |
| DE10325989A1 (de) * | 2003-06-07 | 2005-01-05 | Glatt Gmbh | Verfahren zur Herstellung von und daraus resultierende Mikropellets sowie deren Verwendung |
| US20050181052A1 (en) * | 2004-02-17 | 2005-08-18 | Patel Satishkumar A. | Lansoprazole microtablets |
| WO2007095376A2 (en) * | 2006-02-15 | 2007-08-23 | Kennametal Inc. | Method and apparatus for coating particulates utilizing physical vapor deposition |
| US20090087569A1 (en) * | 2007-09-27 | 2009-04-02 | Fenchem Enterprises Ltd. | Methods for Preparing Highly Stable Hyaluronic Acid |
| IT1401284B1 (it) * | 2010-08-06 | 2013-07-18 | Valpharma S P A | Nuove formulazioni farmaceutiche idonee per la somministrazione orale di esomeprazolo magnesio diidrato, in forma di compresse mups (multi unit pellets system). |
| WO2017145146A1 (en) | 2016-02-25 | 2017-08-31 | Dexcel Pharma Technologies Ltd. | Compositions comprising proton pump inhibitors |
| US10076494B2 (en) | 2016-06-16 | 2018-09-18 | Dexcel Pharma Technologies Ltd. | Stable orally disintegrating pharmaceutical compositions |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3565475D1 (en) * | 1984-04-07 | 1988-11-17 | Bayer Ag | Process and apparatus for the production of granules |
| IL75400A (en) * | 1984-06-16 | 1988-10-31 | Byk Gulden Lomberg Chem Fab | Dialkoxypyridine methyl(sulfinyl or sulfonyl)benzimidazoles,processes for the preparation thereof and pharmaceutical compositions containing the same |
| GB2189698A (en) * | 1986-04-30 | 1987-11-04 | Haessle Ab | Coated omeprazole tablets |
| DE3909455A1 (de) * | 1989-03-22 | 1990-09-27 | Hoechst Ag | Verfahren zur herstellung von wasserdispergierbaren granulaten |
| WO1996001623A1 (en) * | 1994-07-08 | 1996-01-25 | Astra Aktiebolag | Multiple unit tableted dosage form i |
| FR2725623A1 (fr) * | 1994-10-18 | 1996-04-19 | Flamel Tech Sa | Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os |
| DE19613395A1 (de) * | 1996-04-03 | 1997-10-09 | Basf Ag | Granulate hygroskopischer, wasserlöslicher Produkte |
| DE19733094A1 (de) * | 1997-07-31 | 1999-02-04 | Merck Patent Gmbh | Formulierung auf der Basis von Ascorbinsäure mit verbesserter Farbstabilität |
| WO1999018935A1 (de) * | 1997-10-15 | 1999-04-22 | Merck Patent Gmbh | Herstellung eines direkt verpressbaren tablettierhilfsstoffes |
| US6174548B1 (en) * | 1998-08-28 | 2001-01-16 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
| HUP0100065A2 (hu) * | 1997-12-08 | 2001-08-28 | Byk Gulden Lomberg Chemische Fabrik Gmbh. | Savérzékeny vegyületet tartalmazó új kúp gyógyszerforma |
| SE9903236D0 (sv) * | 1999-09-10 | 1999-09-10 | Astra Ab | Method to obtain microparticles |
| SE0100823D0 (sv) * | 2001-03-09 | 2001-03-09 | Astrazeneca Ab | Method I to obtain microparticles |
| US20060159756A1 (en) * | 1999-09-10 | 2006-07-20 | Brita Sjoblom | Method to obtain microparticles containing an H+,K+-ATP-ASE inhibitor |
| SE0100822D0 (sv) * | 2001-03-09 | 2001-03-09 | Astrazeneca Ab | Method II to obtain microparticles |
| SE0100824D0 (sv) * | 2001-03-09 | 2001-03-09 | Astrazeneca Ab | Method III to obtain microparticles |
-
2001
- 2001-03-09 SE SE0100822A patent/SE0100822D0/xx unknown
-
2002
- 2002-03-06 EP EP02701872A patent/EP1370243B1/en not_active Expired - Lifetime
- 2002-03-06 IL IL15746702A patent/IL157467A0/xx unknown
- 2002-03-06 MX MXPA03007887A patent/MXPA03007887A/es active IP Right Grant
- 2002-03-06 CA CA002440163A patent/CA2440163A1/en not_active Abandoned
- 2002-03-06 NZ NZ527997A patent/NZ527997A/en unknown
- 2002-03-06 SI SI200230729T patent/SI1370243T1/sl unknown
- 2002-03-06 AT AT02701872T patent/ATE400253T1/de not_active IP Right Cessation
- 2002-03-06 ES ES02701872T patent/ES2307722T3/es not_active Expired - Lifetime
- 2002-03-06 BR BR0207827-9A patent/BR0207827A/pt not_active IP Right Cessation
- 2002-03-06 AU AU2002235101A patent/AU2002235101B8/en not_active Ceased
- 2002-03-06 US US10/471,314 patent/US20040101565A1/en not_active Abandoned
- 2002-03-06 DK DK02701872T patent/DK1370243T3/da active
- 2002-03-06 KR KR10-2003-7011781A patent/KR20030081506A/ko not_active Ceased
- 2002-03-06 PT PT02701872T patent/PT1370243E/pt unknown
- 2002-03-06 DE DE60227488T patent/DE60227488D1/de not_active Expired - Fee Related
- 2002-03-06 JP JP2002571030A patent/JP2004522796A/ja active Pending
- 2002-03-06 CN CNA028095987A patent/CN1507343A/zh active Pending
- 2002-03-06 WO PCT/SE2002/000400 patent/WO2002072071A1/en not_active Ceased
-
2003
- 2003-08-25 ZA ZA200306614A patent/ZA200306614B/xx unknown
- 2003-09-08 NO NO20033966A patent/NO20033966L/no not_active Application Discontinuation
-
2007
- 2007-07-16 US US11/778,298 patent/US20080175917A1/en not_active Abandoned
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009534441A (ja) * | 2006-04-24 | 2009-09-24 | メファ・アクチェンゲゼルシャフト | ピリジルメチルスルフィニルベンズイミダゾールのための経口速放医薬製剤 |
| WO2021153525A1 (ja) * | 2020-01-27 | 2021-08-05 | 東和薬品株式会社 | エソメプラゾール経口製剤およびその製造方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| IL157467A0 (en) | 2004-03-28 |
| WO2002072071A1 (en) | 2002-09-19 |
| NO20033966L (no) | 2003-11-03 |
| CA2440163A1 (en) | 2002-09-19 |
| AU2002235101B8 (en) | 2006-08-31 |
| PT1370243E (pt) | 2008-09-16 |
| US20080175917A1 (en) | 2008-07-24 |
| ZA200306614B (en) | 2004-11-25 |
| AU2002235101B2 (en) | 2006-07-13 |
| US20040101565A1 (en) | 2004-05-27 |
| ES2307722T3 (es) | 2008-12-01 |
| NZ527997A (en) | 2005-02-25 |
| SI1370243T1 (sl) | 2008-12-31 |
| EP1370243A1 (en) | 2003-12-17 |
| EP1370243B1 (en) | 2008-07-09 |
| MXPA03007887A (es) | 2003-12-04 |
| HK1059896A1 (en) | 2004-07-23 |
| ATE400253T1 (de) | 2008-07-15 |
| CN1507343A (zh) | 2004-06-23 |
| DK1370243T3 (da) | 2008-10-13 |
| KR20030081506A (ko) | 2003-10-17 |
| NO20033966D0 (no) | 2003-09-08 |
| SE0100822D0 (sv) | 2001-03-09 |
| DE60227488D1 (de) | 2008-08-21 |
| BR0207827A (pt) | 2004-03-02 |
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