JP2004516295A5 - - Google Patents

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Publication number
JP2004516295A5
JP2004516295A5 JP2002551566A JP2002551566A JP2004516295A5 JP 2004516295 A5 JP2004516295 A5 JP 2004516295A5 JP 2002551566 A JP2002551566 A JP 2002551566A JP 2002551566 A JP2002551566 A JP 2002551566A JP 2004516295 A5 JP2004516295 A5 JP 2004516295A5
Authority
JP
Japan
Prior art keywords
ylmethyl
benzoxazol
dihydroisoxazol
piperidin
fluorobenzyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2002551566A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004516295A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2001/002277 external-priority patent/WO2002050070A2/en
Publication of JP2004516295A publication Critical patent/JP2004516295A/ja
Publication of JP2004516295A5 publication Critical patent/JP2004516295A5/ja
Abandoned legal-status Critical Current

Links

JP2002551566A 2000-12-21 2001-11-30 サブタイプ選択的なn−メチル−d−アスパラギン酸拮抗薬としてのピペリジン誘導体 Abandoned JP2004516295A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25783200P 2000-12-21 2000-12-21
PCT/IB2001/002277 WO2002050070A2 (en) 2000-12-21 2001-11-30 Piperidine derivatives as subtype selective n-methyl-d-aspartate antagonists

Publications (2)

Publication Number Publication Date
JP2004516295A JP2004516295A (ja) 2004-06-03
JP2004516295A5 true JP2004516295A5 (enExample) 2005-06-23

Family

ID=22977943

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002551566A Abandoned JP2004516295A (ja) 2000-12-21 2001-11-30 サブタイプ選択的なn−メチル−d−アスパラギン酸拮抗薬としてのピペリジン誘導体

Country Status (13)

Country Link
US (1) US6642256B2 (enExample)
EP (1) EP1345935A2 (enExample)
JP (1) JP2004516295A (enExample)
AU (1) AU2002223968A1 (enExample)
BR (1) BR0116311A (enExample)
CA (1) CA2436699A1 (enExample)
HN (1) HN2001000280A (enExample)
MX (1) MXPA03004652A (enExample)
PA (1) PA8535901A1 (enExample)
PE (1) PE20020882A1 (enExample)
TN (1) TNSN01175A1 (enExample)
UY (1) UY27081A1 (enExample)
WO (1) WO2002050070A2 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19952147A1 (de) * 1999-10-29 2001-05-03 Boehringer Ingelheim Pharma Neue Cyclopropane, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
TW200303304A (en) 2002-02-18 2003-09-01 Astrazeneca Ab Chemical compounds
US7273889B2 (en) * 2002-09-25 2007-09-25 Innovative Drug Delivery Systems, Inc. NMDA receptor antagonist formulation with reduced neurotoxicity
US7825147B2 (en) 2003-08-29 2010-11-02 Ranbaxy Laboratories Limited Inhibitors of phosphodiesterase type-IV
SE0400208D0 (sv) 2004-02-02 2004-02-02 Astrazeneca Ab Chemical compounds
GT200600042A (es) * 2005-02-10 2006-09-27 Aventis Pharma Inc Compuestos de bis arilo y heteroarilo sustituido como antagonistas selectivos de 5ht2a
JPWO2006137465A1 (ja) * 2005-06-24 2009-01-22 塩野義製薬株式会社 含窒素複素環誘導体
EP1928866A1 (en) 2005-09-05 2008-06-11 Ranbaxy Laboratories Limited Substituted indazoles as inhibitors of phosphodiesterase type-iv
US7915286B2 (en) 2005-09-16 2011-03-29 Ranbaxy Laboratories Limited Substituted pyrazolo [3,4-b] pyridines as phosphodiesterase inhibitors
PT2124944E (pt) 2007-03-14 2012-05-17 Ranbaxy Lab Ltd Derivados de pirazolo[3,4-b]piridina como inibidores de fosfodiesterase
JP5573307B2 (ja) * 2010-03-31 2014-08-20 Jsr株式会社 感放射線性樹脂組成物、重合体及び化合物
ES2645725T3 (es) 2010-06-11 2017-12-07 Rhodes Technologies Procesos catalizados por metales de transición para la preparación de compuestos de N-alilo y uso de los mismos
EP2592077A1 (en) 2011-11-11 2013-05-15 Almirall, S.A. New cyclohexylamine derivatives having beta2 adrenergic agonist and M3 muscarinic antagonist activities
EP2592078A1 (en) 2011-11-11 2013-05-15 Almirall, S.A. New cyclohexylamine derivatives having beta2 adrenergic agonist and M3 muscarinic antagonist activities
EP4509183A3 (en) 2016-08-16 2025-05-21 BeiGene Switzerland GmbH Crystalline form of (s)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra-hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof
CN110662541B (zh) * 2017-03-12 2023-02-10 王晓冬 多环胺作为阿片受体调节剂
KR101798840B1 (ko) 2017-05-17 2017-11-17 주식회사 레고켐 바이오사이언스 신규 오토탁신 저해 화합물 및 이를 함유하는 약제학적 조성물
PH12022551856A1 (en) 2020-01-22 2024-01-03 Seelos Therapeutics Inc Reducing side effects of nmda antagonists
CN117466836B (zh) * 2023-11-14 2026-02-06 万华化学集团股份有限公司 一种合成烯丙基叔胺的方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1088062C (zh) * 1994-11-23 2002-07-24 纽罗根公司 某些4-氨基甲基-2-取代的咪唑衍生物2-氨基甲基-4-取代的咪唑衍生物新的一族多巴胺受体亚型特异性配体
DE19531321A1 (de) 1995-08-25 1997-02-27 Merck Patent Gmbh Piperidinylmethyloxazolidinone
ZA9610741B (en) 1995-12-22 1997-06-24 Warner Lambert Co 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610745B (en) 1995-12-22 1997-06-24 Warner Lambert Co 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610736B (en) 1995-12-22 1997-06-27 Warner Lambert Co 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists
DE19739332C1 (de) 1997-09-09 1998-11-26 Merck Patent Gmbh Piperidinylmethyloxazolidinon-Derivat
US6015824A (en) 1998-02-10 2000-01-18 Hoffmann-La Roche Ag Pyrrolidine and piperidine derivatives and treatment of neurodegenerative disorders
DE19812331A1 (de) 1998-03-20 1999-09-23 Merck Patent Gmbh Piperidinderivate
AU2960599A (en) 1998-03-30 1999-10-18 Akira Karasawa Quinazoline derivatives
WO2000018763A2 (en) 1998-09-29 2000-04-06 Neurogen Corporation 2-(2,3-dihydrobenzofuran-5-yl)-4-aminomethylimidazoles: dopamine receptor subtype specific ligands

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