JP2004516295A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2004516295A5 JP2004516295A5 JP2002551566A JP2002551566A JP2004516295A5 JP 2004516295 A5 JP2004516295 A5 JP 2004516295A5 JP 2002551566 A JP2002551566 A JP 2002551566A JP 2002551566 A JP2002551566 A JP 2002551566A JP 2004516295 A5 JP2004516295 A5 JP 2004516295A5
- Authority
- JP
- Japan
- Prior art keywords
- ylmethyl
- benzoxazol
- dihydroisoxazol
- piperidin
- fluorobenzyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25783200P | 2000-12-21 | 2000-12-21 | |
| PCT/IB2001/002277 WO2002050070A2 (en) | 2000-12-21 | 2001-11-30 | Piperidine derivatives as subtype selective n-methyl-d-aspartate antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004516295A JP2004516295A (ja) | 2004-06-03 |
| JP2004516295A5 true JP2004516295A5 (enExample) | 2005-06-23 |
Family
ID=22977943
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002551566A Abandoned JP2004516295A (ja) | 2000-12-21 | 2001-11-30 | サブタイプ選択的なｎ−メチル−ｄ−アスパラギン酸拮抗薬としてのピペリジン誘導体 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US6642256B2 (enExample) |
| EP (1) | EP1345935A2 (enExample) |
| JP (1) | JP2004516295A (enExample) |
| AU (1) | AU2002223968A1 (enExample) |
| BR (1) | BR0116311A (enExample) |
| CA (1) | CA2436699A1 (enExample) |
| HN (1) | HN2001000280A (enExample) |
| MX (1) | MXPA03004652A (enExample) |
| PA (1) | PA8535901A1 (enExample) |
| PE (1) | PE20020882A1 (enExample) |
| TN (1) | TNSN01175A1 (enExample) |
| UY (1) | UY27081A1 (enExample) |
| WO (1) | WO2002050070A2 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19952147A1 (de) * | 1999-10-29 | 2001-05-03 | Boehringer Ingelheim Pharma | Neue Cyclopropane, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
| TW200303304A (en) | 2002-02-18 | 2003-09-01 | Astrazeneca Ab | Chemical compounds |
| US7273889B2 (en) * | 2002-09-25 | 2007-09-25 | Innovative Drug Delivery Systems, Inc. | NMDA receptor antagonist formulation with reduced neurotoxicity |
| CA2537185A1 (en) | 2003-08-29 | 2005-03-10 | Ranbaxy Laboratories Limited | Inhibitors of phosphodiesterase type-iv |
| SE0400208D0 (sv) | 2004-02-02 | 2004-02-02 | Astrazeneca Ab | Chemical compounds |
| GT200600042A (es) * | 2005-02-10 | 2006-09-27 | Aventis Pharma Inc | Compuestos de bis arilo y heteroarilo sustituido como antagonistas selectivos de 5ht2a |
| JPWO2006137465A1 (ja) * | 2005-06-24 | 2009-01-22 | 塩野義製薬株式会社 | 含窒素複素環誘導体 |
| US7781460B2 (en) | 2005-09-05 | 2010-08-24 | Ranbaxy Laboratories Limited | Substituted indazoles as inhibitors of phosphodiesterase type-IV |
| EP1934219A1 (en) | 2005-09-16 | 2008-06-25 | Ranbaxy Laboratories Limited | Substituted pyrazolo [3,4-b] pyridines as phosphodiesterase inhibitors |
| CN103497185A (zh) | 2007-03-14 | 2014-01-08 | 兰贝克赛实验室有限公司 | 用作磷酸二酯酶抑制剂的吡唑并(3,4-b)吡啶衍生物 |
| JP5573307B2 (ja) * | 2010-03-31 | 2014-08-20 | Ｊｓｒ株式会社 | 感放射線性樹脂組成物、重合体及び化合物 |
| CA2936749C (en) | 2010-06-11 | 2019-07-09 | Joshua R. Giguere | Transition metal-catalyzed processes for the preparation of n-allyl compounds and use thereof |
| EP2592078A1 (en) | 2011-11-11 | 2013-05-15 | Almirall, S.A. | New cyclohexylamine derivatives having beta2 adrenergic agonist and M3 muscarinic antagonist activities |
| EP2592077A1 (en) | 2011-11-11 | 2013-05-15 | Almirall, S.A. | New cyclohexylamine derivatives having beta2 adrenergic agonist and M3 muscarinic antagonist activities |
| WO2018033853A2 (en) | 2016-08-16 | 2018-02-22 | Beigene, Ltd. | Crystalline form of (s)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra-hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof |
| CN110662541B (zh) * | 2017-03-12 | 2023-02-10 | 王晓冬 | 多环胺作为阿片受体调节剂 |
| KR101798840B1 (ko) | 2017-05-17 | 2017-11-17 | 주식회사 레고켐 바이오사이언스 | 신규 오토탁신 저해 화합물 및 이를 함유하는 약제학적 조성물 |
| CN115135317A (zh) | 2020-01-22 | 2022-09-30 | 西洛斯治疗有限公司 | 减少nmda拮抗剂的副作用 |
| CN117466836A (zh) * | 2023-11-14 | 2024-01-30 | 万华化学集团股份有限公司 | 一种合成烯丙基叔胺的方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1088062C (zh) * | 1994-11-23 | 2002-07-24 | 纽罗根公司 | 某些4－氨基甲基－2－取代的咪唑衍生物2－氨基甲基－4－取代的咪唑衍生物新的一族多巴胺受体亚型特异性配体 |
| DE19531321A1 (de) | 1995-08-25 | 1997-02-27 | Merck Patent Gmbh | Piperidinylmethyloxazolidinone |
| ZA9610741B (en) | 1995-12-22 | 1997-06-24 | Warner Lambert Co | 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists |
| ZA9610745B (en) | 1995-12-22 | 1997-06-24 | Warner Lambert Co | 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists |
| ZA9610736B (en) | 1995-12-22 | 1997-06-27 | Warner Lambert Co | 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists |
| DE19739332C1 (de) * | 1997-09-09 | 1998-11-26 | Merck Patent Gmbh | Piperidinylmethyloxazolidinon-Derivat |
| US6015824A (en) | 1998-02-10 | 2000-01-18 | Hoffmann-La Roche Ag | Pyrrolidine and piperidine derivatives and treatment of neurodegenerative disorders |
| DE19812331A1 (de) | 1998-03-20 | 1999-09-23 | Merck Patent Gmbh | Piperidinderivate |
| AU2960599A (en) * | 1998-03-30 | 1999-10-18 | Akira Karasawa | Quinazoline derivatives |
| WO2000018763A2 (en) * | 1998-09-29 | 2000-04-06 | Neurogen Corporation | 2-(2,3-dihydrobenzofuran-5-yl)-4-aminomethylimidazoles: dopamine receptor subtype specific ligands |
-
2001
- 2001-11-30 MX MXPA03004652A patent/MXPA03004652A/es not_active Application Discontinuation
- 2001-11-30 EP EP01271104A patent/EP1345935A2/en not_active Withdrawn
- 2001-11-30 CA CA002436699A patent/CA2436699A1/en not_active Abandoned
- 2001-11-30 BR BR0116311-6A patent/BR0116311A/pt not_active IP Right Cessation
- 2001-11-30 WO PCT/IB2001/002277 patent/WO2002050070A2/en not_active Ceased
- 2001-11-30 JP JP2002551566A patent/JP2004516295A/ja not_active Abandoned
- 2001-11-30 US US09/998,479 patent/US6642256B2/en not_active Expired - Fee Related
- 2001-11-30 AU AU2002223968A patent/AU2002223968A1/en not_active Abandoned
- 2001-12-18 PE PE2001001265A patent/PE20020882A1/es not_active Application Discontinuation
- 2001-12-18 UY UY27081A patent/UY27081A1/es not_active Application Discontinuation
- 2001-12-19 HN HN2001000280A patent/HN2001000280A/es unknown
- 2001-12-20 TN TNTNSN01175A patent/TNSN01175A1/fr unknown
- 2001-12-21 PA PA20018535901A patent/PA8535901A1/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2004516295A5 (enExample) | ||
| US9856247B2 (en) | 4-methyl-dihydropyrimidines for the treatment and prophylaxis of Hepatitis B virus infection | |
| US9926285B2 (en) | Allosteric modulators of nicotinic acetylcholine receptors | |
| JP2019077725A5 (enExample) | ||
| US11713312B2 (en) | Substituted bicyclic compounds as farnesoid X receptor modulators | |
| JP2006502134A5 (enExample) | ||
| JP2020516671A5 (enExample) | ||
| US20050043545A1 (en) | 4-(5-Membered)-heteroaryl acyl pyrrolidine derivatives as hcv inhibitors | |
| JP2012502006A5 (enExample) | ||
| JP2020512373A5 (enExample) | ||
| JP2008513515A5 (enExample) | ||
| JP2008513499A5 (enExample) | ||
| JP2007505091A5 (enExample) | ||
| AU782191B2 (en) | Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists | |
| RU2008126398A (ru) | Производные гетероарилзамещенного пиперидина в качестве ингибиторов печеночной карнитин пальмитоилтрансферазы (l-cpti) | |
| JP2007516173A5 (enExample) | ||
| JP2015509510A5 (enExample) | ||
| JP2008500991A (ja) | 医学的使用のためのｃｒｔｈ２レセプターリガンド | |
| JP2009525275A (ja) | 多環式１，２，３，４−テトラヒドロ−イソキノリン誘導体およびｐｐａｒモジュレーターとしてのそれらを含む組成物 | |
| RU2008110949A (ru) | Соединения и композиции-иммуносупрессанты | |
| TW201038586A (en) | Sulfonamide derivatives | |
| KR20090024820A (ko) | 인간 단백질 티로신 포스파타아제 억제제 및 이용 방법 | |
| RU2019132212A (ru) | Селективные ингибиторы hdac6 | |
| JP2006503081A5 (enExample) | ||
| WO2004101529A1 (ja) | 含窒素複素環化合物およびその医薬用途 |