JP2004504320A5 - - Google Patents

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Publication number
JP2004504320A5
JP2004504320A5 JP2002512179A JP2002512179A JP2004504320A5 JP 2004504320 A5 JP2004504320 A5 JP 2004504320A5 JP 2002512179 A JP2002512179 A JP 2002512179A JP 2002512179 A JP2002512179 A JP 2002512179A JP 2004504320 A5 JP2004504320 A5 JP 2004504320A5
Authority
JP
Japan
Prior art keywords
motomeko
compound according
beta
receptor agonist
obesity
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2002512179A
Other languages
English (en)
Japanese (ja)
Other versions
JP4988128B2 (ja
JP2004504320A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2001/016519 external-priority patent/WO2002006276A1/en
Publication of JP2004504320A publication Critical patent/JP2004504320A/ja
Publication of JP2004504320A5 publication Critical patent/JP2004504320A5/ja
Application granted granted Critical
Publication of JP4988128B2 publication Critical patent/JP4988128B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2002512179A 2000-07-13 2001-07-09 β３アドレナリン作動性アゴニスト Expired - Lifetime JP4988128B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US21796500P 2000-07-13 2000-07-13
US60/217,965 2000-07-13
US24161400P 2000-10-19 2000-10-19
US60/241,614 2000-10-19
US29298801P 2001-05-23 2001-05-23
US60/292,988 2001-05-23
PCT/US2001/016519 WO2002006276A1 (en) 2000-07-13 2001-07-09 Beta3 adrenergic agonists

Publications (3)

Publication Number Publication Date
JP2004504320A JP2004504320A (ja) 2004-02-12
JP2004504320A5 true JP2004504320A5 (https=) 2008-08-21
JP4988128B2 JP4988128B2 (ja) 2012-08-01

Family

ID=27396478

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002512179A Expired - Lifetime JP4988128B2 (ja) 2000-07-13 2001-07-09 β３アドレナリン作動性アゴニスト

Country Status (23)

Country Link
US (2) US6730792B2 (https=)
EP (1) EP1303509B1 (https=)
JP (1) JP4988128B2 (https=)
KR (1) KR20030016396A (https=)
CN (1) CN1441800A (https=)
AU (1) AU2001272917A1 (https=)
BR (1) BR0112409A (https=)
CA (1) CA2415331A1 (https=)
CZ (1) CZ2003106A3 (https=)
DK (1) DK1303509T3 (https=)
EA (1) EA200300145A1 (https=)
ES (1) ES2398097T3 (https=)
HR (1) HRP20030018A2 (https=)
HU (1) HUP0301329A2 (https=)
IL (2) IL152528A0 (https=)
MX (1) MXPA03000308A (https=)
NO (1) NO20030098D0 (https=)
PE (1) PE20020195A1 (https=)
PL (1) PL360098A1 (https=)
PT (1) PT1303509E (https=)
SK (1) SK632003A3 (https=)
SV (1) SV2002000522A (https=)
WO (1) WO2002006276A1 (https=)

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EP1303509B1 (en) * 2000-07-13 2012-11-28 Eli Lilly And Company Beta3 adrenergic agonists
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MX354786B (es) 2007-06-04 2018-03-21 Synergy Pharmaceuticals Inc Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos.
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AU2009270833B2 (en) 2008-07-16 2015-02-19 Bausch Health Ireland Limited Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
ES2394349B1 (es) 2012-08-29 2013-11-04 Fundación Centro Nacional De Investigaciones Cardiovasculares Carlos Iii Uso de agonistas selectivos de receptores beta-3 adrenérgicos para el tratamiento de hipertensión pulmonar
AU2014235215A1 (en) 2013-03-15 2015-10-01 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase and their uses
US9346802B2 (en) 2013-03-15 2016-05-24 Epizyme, Inc. CARM1 inhibitors and uses thereof
CA2903813C (en) 2013-03-15 2023-08-29 Epizyme, Inc. Carm1 inhibitors and uses thereof
AU2014235209B2 (en) 2013-03-15 2018-06-14 Bausch Health Ireland Limited Guanylate cyclase receptor agonists combined with other drugs
WO2014144455A1 (en) 2013-03-15 2014-09-18 Epizyme, Inc. 1 -phenoxy-3-(alkylamino)-propan-2-ol derivatives as carm1 inhibitors and uses thereof
BR112015030326A2 (pt) 2013-06-05 2017-08-29 Synergy Pharmaceuticals Inc Agonistas ultrapuros de guanilato ciclase c, método de fabricar e usar os mesmos
CA2996879C (en) 2015-10-05 2020-04-21 Elanco Us Inc. Methods and formulations for reducing ammonia emissions from bovines
CN112255349A (zh) * 2020-10-14 2021-01-22 青岛天祥食品集团有限公司 一种检测食用植物油中缩水甘油及缩水甘油酯的快速检测方法
CN114380811A (zh) * 2021-12-29 2022-04-22 天和药业股份有限公司 一种卢巴贝隆的合成方法

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