JP2003514770A - 抗増殖性医薬の燐脂質プロドラッグ - Google Patents
抗増殖性医薬の燐脂質プロドラッグInfo
- Publication number
- JP2003514770A JP2003514770A JP2001522958A JP2001522958A JP2003514770A JP 2003514770 A JP2003514770 A JP 2003514770A JP 2001522958 A JP2001522958 A JP 2001522958A JP 2001522958 A JP2001522958 A JP 2001522958A JP 2003514770 A JP2003514770 A JP 2003514770A
- Authority
- JP
- Japan
- Prior art keywords
- mtx
- glycero
- stearoyl
- disease
- phosphatidylcholine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IL131887 | 1999-09-14 | ||
| IL13188799A IL131887A0 (en) | 1999-09-14 | 1999-09-14 | Phospholipid prodrugs of anti-proliferative drugs |
| PCT/IL2000/000562 WO2001019320A2 (en) | 1999-09-14 | 2000-09-13 | Phospholipid prodrugs of anti-proliferative drugs |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2003514770A true JP2003514770A (ja) | 2003-04-22 |
| JP2003514770A5 JP2003514770A5 (https=) | 2007-10-11 |
Family
ID=11073248
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001522958A Pending JP2003514770A (ja) | 1999-09-14 | 2000-09-13 | 抗増殖性医薬の燐脂質プロドラッグ |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US6774121B1 (https=) |
| EP (1) | EP1218013A4 (https=) |
| JP (1) | JP2003514770A (https=) |
| AU (1) | AU781507B2 (https=) |
| CA (1) | CA2382633A1 (https=) |
| IL (2) | IL131887A0 (https=) |
| NZ (1) | NZ517522A (https=) |
| WO (1) | WO2001019320A2 (https=) |
| ZA (1) | ZA200201081B (https=) |
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| JP2013525390A (ja) * | 2010-04-30 | 2013-06-20 | テロルメディクス エセアー | リン脂質薬物類似体 |
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| EA014685B1 (ru) | 2003-04-25 | 2010-12-30 | Джилид Сайэнс, Инк. | Фосфонатсодержащие антивирусные соединения (варианты) и фармацевтическая композиция на их основе |
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| AU2005330489B2 (en) | 2004-07-27 | 2011-08-25 | Gilead Sciences, Inc. | Nucleoside phosphonate conjugates as anti HIV agents |
| EP1904183B1 (en) | 2005-07-05 | 2014-10-15 | Purdue Research Foundation | Pharmaceutical composition for the treatment of osteoarthritis |
| DE102006019907A1 (de) * | 2006-04-28 | 2007-10-31 | Müller-Enoch, Dieter, Prof. Dr. | Verwendung von substituierten Glycerinderivaten zur Herstellung einer pharmazeutischen Zubereitung |
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| US20120003298A1 (en) * | 2010-04-30 | 2012-01-05 | Alcide Barberis | Methods for inducing an immune response |
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| US9499800B2 (en) | 2013-12-26 | 2016-11-22 | Regents Of The University Of Minnesota | Methods of making and using chemically self assembled-nanorings |
| CA2968145C (en) * | 2014-11-17 | 2023-06-27 | Cellectar Biosciences, Inc. | Phospholipid ether analogs as cancer-targeting drug vehicles |
| SI3661937T1 (sl) | 2017-08-01 | 2021-11-30 | Gilead Sciences, Inc. | Kristalinične oblike etil((S)-((((2R,5R)-5-(6-amino-9H-purin-9-IL)-4- fluoro-2,5-dihidrofuran-2-IL)oksi)metil)(fenoksi)fosforil)-L-alaninata (GS-9131) za zdravljenje virusnih okužb |
| CN112437674A (zh) * | 2018-04-11 | 2021-03-02 | 新墨西哥科技大学研究园公司 | 用于药物递送的脂质前药 |
| WO2025202629A1 (en) | 2024-03-26 | 2025-10-02 | Coopervision International Limited | Contact lens loaded with a glycerophospholipid |
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- 2000-09-13 WO PCT/IL2000/000562 patent/WO2001019320A2/en not_active Ceased
- 2000-09-13 NZ NZ517522A patent/NZ517522A/en not_active IP Right Cessation
- 2000-09-13 JP JP2001522958A patent/JP2003514770A/ja active Pending
- 2000-09-13 EP EP00960946A patent/EP1218013A4/en not_active Withdrawn
- 2000-09-13 AU AU73093/00A patent/AU781507B2/en not_active Ceased
- 2000-09-13 US US10/088,160 patent/US6774121B1/en not_active Expired - Fee Related
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| JP2013525390A (ja) * | 2010-04-30 | 2013-06-20 | テロルメディクス エセアー | リン脂質薬物類似体 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001019320A3 (en) | 2001-09-27 |
| ZA200201081B (en) | 2003-04-30 |
| NZ517522A (en) | 2003-08-29 |
| CA2382633A1 (en) | 2001-03-22 |
| IL148554A (en) | 2007-10-31 |
| EP1218013A4 (en) | 2004-12-15 |
| AU7309300A (en) | 2001-04-17 |
| EP1218013A2 (en) | 2002-07-03 |
| WO2001019320A2 (en) | 2001-03-22 |
| US6774121B1 (en) | 2004-08-10 |
| IL131887A0 (en) | 2001-03-19 |
| AU781507B2 (en) | 2005-05-26 |
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