JP2002506036A - 疾患を処置するにおける新規ヌクレオシドアナログおよびその使用 - Google Patents
疾患を処置するにおける新規ヌクレオシドアナログおよびその使用Info
- Publication number
- JP2002506036A JP2002506036A JP2000535350A JP2000535350A JP2002506036A JP 2002506036 A JP2002506036 A JP 2002506036A JP 2000535350 A JP2000535350 A JP 2000535350A JP 2000535350 A JP2000535350 A JP 2000535350A JP 2002506036 A JP2002506036 A JP 2002506036A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- fluoro
- oriented
- deoxyuridine
- evaporated
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Genetics & Genomics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Virology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/038,647 | 1998-03-11 | ||
| US09/038,647 US5939402A (en) | 1995-09-21 | 1998-03-11 | Nucleoside analogs and uses against parasitic infection |
| US09/220,307 | 1998-12-23 | ||
| US09/219,947 | 1998-12-23 | ||
| US09/220,307 US6207649B1 (en) | 1995-09-21 | 1998-12-23 | Nucleoside analogs and uses in treating disease |
| US09/219,947 US6242428B1 (en) | 1995-09-21 | 1998-12-23 | Nucleoside analogs and uses in treating Plasmodium falciparum infection |
| PCT/US1999/005360 WO1999045935A1 (en) | 1998-03-11 | 1999-03-11 | Novel nucleoside analogs and uses in treating disease |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002506036A true JP2002506036A (ja) | 2002-02-26 |
| JP2002506036A5 JP2002506036A5 (https=) | 2006-04-27 |
Family
ID=27365434
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000535350A Pending JP2002506036A (ja) | 1998-03-11 | 1999-03-11 | 疾患を処置するにおける新規ヌクレオシドアナログおよびその使用 |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP1069903A1 (https=) |
| JP (1) | JP2002506036A (https=) |
| AU (1) | AU3080899A (https=) |
| CA (1) | CA2322494A1 (https=) |
| WO (1) | WO1999045935A1 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006516641A (ja) * | 2003-02-03 | 2006-07-06 | シーブイ・セラピューティクス・インコーポレイテッド | アデノシン受容体の完全アゴニストおよび部分アゴニスト |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2004201286B2 (en) * | 1998-08-10 | 2007-06-21 | Centre National De La Recherche Scientifique (Cnrs) | Beta-L-2'-Deoxy Nucleosides for the Treatment of Hepatitis B |
| US6444652B1 (en) | 1998-08-10 | 2002-09-03 | Novirio Pharmaceuticals Limited | β-L-2'-deoxy-nucleosides for the treatment of hepatitis B |
| ES2255295T3 (es) * | 1998-08-10 | 2006-06-16 | Idenix (Cayman) Limited | 2'-deoxi-beta-l-nucleosidos para el tratamiento de la hepatitis b. |
| AU2007216721B2 (en) * | 1998-08-10 | 2011-05-19 | Centre National De La Recherche Scientifique | Beta-L-2'-Deoxy Nucleosides for the Treatment of Hepatitis B |
| US6875751B2 (en) | 2000-06-15 | 2005-04-05 | Idenix Pharmaceuticals, Inc. | 3′-prodrugs of 2′-deoxy-β-L-nucleosides |
| EP1352910A1 (en) | 2002-04-10 | 2003-10-15 | Grünenthal GmbH | New analogs of nitrobenzylthioinosine |
| TWI244393B (en) | 2002-08-06 | 2005-12-01 | Idenix Pharmaceuticals Inc | Crystalline and amorphous forms of beta-L-2'-deoxythymidine |
| GB0400290D0 (en) * | 2004-01-08 | 2004-02-11 | Medivir Ab | dUTPase inhibitors |
| CN106459127A (zh) * | 2014-05-28 | 2017-02-22 | 艾登尼克斯药业有限公司 | 用于治疗癌症的核苷衍生物 |
| JP2017516779A (ja) * | 2014-05-28 | 2017-06-22 | アイデニクス・ファーマシューティカルズ・エルエルシー | 癌治療のためのヌクレオシド誘導体 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5672594A (en) * | 1994-10-24 | 1997-09-30 | Genencor International, Inc. | L-erythrosyl nucleosides |
| US5559101A (en) * | 1994-10-24 | 1996-09-24 | Genencor International, Inc. | L-ribofuranosyl nucleosides |
-
1999
- 1999-03-11 EP EP99912434A patent/EP1069903A1/en not_active Withdrawn
- 1999-03-11 WO PCT/US1999/005360 patent/WO1999045935A1/en not_active Ceased
- 1999-03-11 AU AU30808/99A patent/AU3080899A/en not_active Abandoned
- 1999-03-11 JP JP2000535350A patent/JP2002506036A/ja active Pending
- 1999-03-11 CA CA002322494A patent/CA2322494A1/en not_active Abandoned
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006516641A (ja) * | 2003-02-03 | 2006-07-06 | シーブイ・セラピューティクス・インコーポレイテッド | アデノシン受容体の完全アゴニストおよび部分アゴニスト |
Also Published As
| Publication number | Publication date |
|---|---|
| WO1999045935A1 (en) | 1999-09-16 |
| EP1069903A1 (en) | 2001-01-24 |
| AU3080899A (en) | 1999-09-27 |
| CA2322494A1 (en) | 1999-09-16 |
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