JP2002114786A5 - - Google Patents
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- Publication number
- JP2002114786A5 JP2002114786A5 JP2001288509A JP2001288509A JP2002114786A5 JP 2002114786 A5 JP2002114786 A5 JP 2002114786A5 JP 2001288509 A JP2001288509 A JP 2001288509A JP 2001288509 A JP2001288509 A JP 2001288509A JP 2002114786 A5 JP2002114786 A5 JP 2002114786A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrogen
- lower alkyl
- compound according
- halogen
- sulfamoyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 229910052739 hydrogen Inorganic materials 0.000 claims 21
- 239000001257 hydrogen Substances 0.000 claims 21
- 125000000217 alkyl group Chemical group 0.000 claims 19
- 150000001875 compounds Chemical class 0.000 claims 12
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 11
- 150000002431 hydrogen Chemical class 0.000 claims 10
- 125000003545 alkoxy group Chemical group 0.000 claims 8
- -1 cyano, nitro, amino Chemical group 0.000 claims 8
- 229910052736 halogen Inorganic materials 0.000 claims 8
- 150000002367 halogens Chemical class 0.000 claims 8
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims 7
- 125000004414 alkyl thio group Chemical group 0.000 claims 7
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 claims 7
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 7
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 claims 7
- 125000004663 dialkyl amino group Chemical group 0.000 claims 7
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 7
- RSSRTDPSDFGXCU-UHFFFAOYSA-N C=1(NC=CC2=CC=C3C(C=12)=CC=N3)C(=O)O Chemical compound C=1(NC=CC2=CC=C3C(C=12)=CC=N3)C(=O)O RSSRTDPSDFGXCU-UHFFFAOYSA-N 0.000 claims 4
- 150000001408 amides Chemical class 0.000 claims 4
- 150000002148 esters Chemical class 0.000 claims 4
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 4
- 239000000651 prodrug Substances 0.000 claims 4
- 229940002612 prodrug Drugs 0.000 claims 4
- 150000003839 salts Chemical class 0.000 claims 4
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 4
- 125000003710 aryl alkyl group Chemical group 0.000 claims 3
- 125000003118 aryl group Chemical group 0.000 claims 3
- 125000001072 heteroaryl group Chemical group 0.000 claims 3
- 125000004446 heteroarylalkyl group Chemical group 0.000 claims 3
- 208000018737 Parkinson disease Diseases 0.000 claims 1
- 239000003085 diluting agent Substances 0.000 claims 1
- 239000003814 drug Substances 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
- 239000000546 pharmaceutical excipient Substances 0.000 claims 1
- 229940124597 therapeutic agent Drugs 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23482600P | 2000-09-22 | 2000-09-22 | |
| US60/234826 | 2000-09-22 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002114786A JP2002114786A (ja) | 2002-04-16 |
| JP2002114786A5 true JP2002114786A5 (https=) | 2004-12-24 |
Family
ID=22882987
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001288509A Pending JP2002114786A (ja) | 2000-09-22 | 2001-09-21 | Ｍ４選択性アザアントラセンムスカリンレセプター拮抗薬としてインドールを含む縮合環系 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US6500837B2 (https=) |
| EP (1) | EP1191027A1 (https=) |
| JP (1) | JP2002114786A (https=) |
| BR (1) | BR0104169A (https=) |
| CA (1) | CA2357306A1 (https=) |
| MX (1) | MXPA01009550A (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002072549A1 (en) * | 2001-03-12 | 2002-09-19 | Millennium Pharmaceuticals, Inc. | Functionalized heterocycles as modulators of chemokine receptor function and methods of use therefor |
| CN113613650B (zh) * | 2019-03-25 | 2024-12-10 | 冷泉港实验室 | 治疗贫血的毒蕈碱乙酰胆碱受体亚型4拮抗剂 |
-
2001
- 2001-09-14 CA CA002357306A patent/CA2357306A1/en not_active Abandoned
- 2001-09-14 US US09/952,735 patent/US6500837B2/en not_active Expired - Fee Related
- 2001-09-18 EP EP01122280A patent/EP1191027A1/en not_active Withdrawn
- 2001-09-20 BR BR0104169-0A patent/BR0104169A/pt not_active IP Right Cessation
- 2001-09-21 JP JP2001288509A patent/JP2002114786A/ja active Pending
- 2001-09-21 MX MXPA01009550A patent/MXPA01009550A/es unknown
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