JP2001501170A5 - - Google Patents

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Publication number
JP2001501170A5
JP2001501170A5 JP1997537864A JP53786497A JP2001501170A5 JP 2001501170 A5 JP2001501170 A5 JP 2001501170A5 JP 1997537864 A JP1997537864 A JP 1997537864A JP 53786497 A JP53786497 A JP 53786497A JP 2001501170 A5 JP2001501170 A5 JP 2001501170A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1997537864A
Other languages
English (en)
Japanese (ja)
Other versions
JP2001501170A (ja
JP4215822B2 (ja
Filing date
Publication date
Priority claimed from GBGB9608457.9A external-priority patent/GB9608457D0/en
Priority claimed from GBGB9616115.3A external-priority patent/GB9616115D0/en
Priority claimed from GBGB9624584.0A external-priority patent/GB9624584D0/en
Application filed filed Critical
Priority claimed from PCT/GB1997/001157 external-priority patent/WO1997040065A2/en
Publication of JP2001501170A publication Critical patent/JP2001501170A/ja
Publication of JP2001501170A5 publication Critical patent/JP2001501170A5/ja
Application granted granted Critical
Publication of JP4215822B2 publication Critical patent/JP4215822B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP53786497A 1996-04-24 1997-04-24 タンパク質分解酵素の基質および阻害剤 Expired - Fee Related JP4215822B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB9608457.9 1996-04-24
GBGB9608457.9A GB9608457D0 (en) 1996-04-24 1996-04-24 Inhibitors of proteolytic enzymes
GBGB9616115.3A GB9616115D0 (en) 1996-07-31 1996-07-31 Substrate and inhibitors of proteolytic enzymes
GB9616115.3 1996-07-31
GB9624584.0 1996-11-27
GBGB9624584.0A GB9624584D0 (en) 1996-11-27 1996-11-27 Substances and inhibitors of proteolytic enzymes
PCT/GB1997/001157 WO1997040065A2 (en) 1996-04-24 1997-04-24 Substrates and inhibitors of proteolytic enzymes

Publications (3)

Publication Number Publication Date
JP2001501170A JP2001501170A (ja) 2001-01-30
JP2001501170A5 true JP2001501170A5 (https=) 2005-01-13
JP4215822B2 JP4215822B2 (ja) 2009-01-28

Family

ID=27268257

Family Applications (2)

Application Number Title Priority Date Filing Date
JP53786497A Expired - Fee Related JP4215822B2 (ja) 1996-04-24 1997-04-24 タンパク質分解酵素の基質および阻害剤
JP09539622A Abandoned JP2000512979A (ja) 1996-04-24 1997-04-24 自己デコンボリューション法によるコンビナトリアルライブラリー

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP09539622A Abandoned JP2000512979A (ja) 1996-04-24 1997-04-24 自己デコンボリューション法によるコンビナトリアルライブラリー

Country Status (10)

Country Link
US (2) US6528275B1 (https=)
EP (2) EP0906333B1 (https=)
JP (2) JP4215822B2 (https=)
AT (1) ATE203545T1 (https=)
AU (2) AU706855B2 (https=)
CA (2) CA2252408A1 (https=)
DE (1) DE69705838T2 (https=)
DK (1) DK0906333T3 (https=)
ES (1) ES2162277T3 (https=)
WO (2) WO1997042216A1 (https=)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6042789A (en) * 1996-10-23 2000-03-28 Glaxo Group Limited System for parallel synthesis of organic compounds
US6149869A (en) * 1996-10-23 2000-11-21 Glaxo Wellcome Inc. Chemical synthesizers
US6617114B1 (en) 1996-10-31 2003-09-09 Karo Bio Ab Identification of drug complementary combinatorial libraries
CA2270394A1 (en) * 1996-10-31 1998-05-07 Novalon Pharmaceutical Corporation Identification of drugs using complementary combinatorial libraries
US6083761A (en) * 1996-12-02 2000-07-04 Glaxo Wellcome Inc. Method and apparatus for transferring and combining reagents
US6054325A (en) * 1996-12-02 2000-04-25 Glaxo Wellcom Inc. Method and apparatus for transferring and combining distinct chemical compositions with reagents
GB9722818D0 (en) * 1997-10-30 1997-12-24 Peptide Therapeutics Ltd A method for mapping the active sites bound by enzymes that covalently modify substrate molecules
JP2001524457A (ja) * 1997-11-26 2001-12-04 メディヴァー ユーケイ リミテッド アミド結合固着による混成ライブラリー調製のための固相技術
US6083682A (en) 1997-12-19 2000-07-04 Glaxo Group Limited System and method for solid-phase parallel synthesis of a combinatorial collection of compounds
MY153569A (en) 1998-01-20 2015-02-27 Mitsubishi Tanabe Pharma Corp Inhibitors of ?4 mediated cell adhesion
US6569636B2 (en) 1998-05-29 2003-05-27 Hawaii Biotechnology Group, Inc. Assay for modulators of metallo-enzyme activity
DE19925402C2 (de) * 1999-06-02 2001-12-20 Molecular Machines & Ind Gmbh Screening von Target-Ligand-Wechselwirkungen
US20020076741A1 (en) 2000-02-11 2002-06-20 Tencza Sarah Burroughs Peptide biosensors for anthrax protease
JP2002250730A (ja) * 2001-02-27 2002-09-06 Shinwa Kako Kk 分子センサー及びその製造方法
MY140707A (en) 2002-02-28 2010-01-15 Mitsubishi Tanabe Pharma Corp Process for preparing a phenylalanine derivative and intermediates thereof
AU2003265398A1 (en) * 2002-08-09 2004-02-25 Transtech Pharma, Inc. Aryl and heteroaryl compounds and methods to modulate coagulation
US7501538B2 (en) 2003-08-08 2009-03-10 Transtech Pharma, Inc. Aryl and heteroaryl compounds, compositions and methods of use
US7208601B2 (en) * 2003-08-08 2007-04-24 Mjalli Adnan M M Aryl and heteroaryl compounds, compositions, and methods of use
US8015064B2 (en) * 2005-04-20 2011-09-06 At&T Intellectual Property I, Lp System and method of providing advertisements to cellular devices
ATE442438T1 (de) * 2005-07-26 2009-09-15 Council Scient Ind Res Verfahren zur identifizierung von die stresstoleranz in hefe erhíhenden genen sowie verwendung dieser gene zur verbesserung von hefestämmen
DK2364366T3 (da) 2008-11-05 2014-03-31 Morphosys Ag Affoldningsmetode
JP5798487B2 (ja) * 2008-11-20 2015-10-21 ネーデルランドセ・オルガニサティ・フォール・トゥーヘパスト−ナトゥールウェテンスハッペライク・オンデルズーク・テーエヌオー Fretに基づく病原体の迅速診断
EP2189536A1 (en) * 2008-11-20 2010-05-26 Nederlandse Organisatie voor toegepast-natuurwetenschappelijk Onderzoek TNO Rapid FRET based anthrax diagnosis
KR102668696B1 (ko) * 2012-01-12 2024-05-29 예일 유니버시티 E3 유비퀴틴 리가아제에 의한 표적 단백질 및 다른 폴리펩티드의 증진된 분해를 위한 화합물 및 방법
GB201311891D0 (en) 2013-07-03 2013-08-14 Glaxosmithkline Ip Dev Ltd Novel compound
GB201311888D0 (en) 2013-07-03 2013-08-14 Glaxosmithkline Ip Dev Ltd Novel compounds
US20180228907A1 (en) 2014-04-14 2018-08-16 Arvinas, Inc. Cereblon ligands and bifunctional compounds comprising the same
BR112018008918A8 (pt) 2015-11-02 2019-02-26 Univ Yale compostos de quimera proteólise dirigida e métodos para preparação e uso dos mesmos

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0428000A1 (en) 1989-11-03 1991-05-22 Abbott Laboratories Fluorogenic substrates for the detection of proteolytic enzyme activity
US5011910A (en) * 1989-12-28 1991-04-30 Washington University Reagent and method for determining activity of retroviral protease
US5164300A (en) 1989-12-28 1992-11-17 Washington University Method for determining activity of retroviral protease
DK93990D0 (da) * 1990-04-17 1990-04-17 Carlsberg As Fluorogene peptider og deres anvendelse ved bestemmelse af enzymatisk aktivitet
HU9201687D0 (en) 1992-05-21 1992-08-28 Arpad Furka Preparation of sets from peptid mixtures with polycomponents and their use for the identification of biologically active peptides
US5585275A (en) * 1992-09-02 1996-12-17 Arris Pharmaceutical Corporation Pilot apparatus for peptide synthesis and screening
AU7552394A (en) 1993-12-15 1995-07-03 Combichem, Inc. Combinatorial libraries and methods for their use
US5506115A (en) 1994-04-29 1996-04-09 G. D. Searle & Co. Reagent and method for determining activity of herpes protease
US5738996A (en) 1994-06-15 1998-04-14 Pence, Inc. Combinational library composition and method
EP1019528B1 (en) 1996-01-04 2003-10-29 Nederlandse Organisatie Voor Toegepast-Natuurwetenschappelijk Onderzoek Tno Method for assaying proteolytic enzymes using fluorescence-quenched substrates
US7135288B2 (en) * 2002-09-27 2006-11-14 Ut-Battelle, Llc Combinatorial synthesis of ceramic materials

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