ITRM20050416A1 - Derivati delle benzodiazepine e loro usi in campo medico. - Google Patents
Derivati delle benzodiazepine e loro usi in campo medico.Info
- Publication number
- ITRM20050416A1 ITRM20050416A1 IT000416A ITRM20050416A ITRM20050416A1 IT RM20050416 A1 ITRM20050416 A1 IT RM20050416A1 IT 000416 A IT000416 A IT 000416A IT RM20050416 A ITRM20050416 A IT RM20050416A IT RM20050416 A1 ITRM20050416 A1 IT RM20050416A1
- Authority
- IT
- Italy
- Prior art keywords
- sub
- alkyl
- alkynyl
- alkenyl
- alkoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Priority Applications (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT000416A ITRM20050416A1 (it) | 2005-08-03 | 2005-08-03 | Derivati delle benzodiazepine e loro usi in campo medico. |
EP06756301A EP1910383B1 (en) | 2005-08-03 | 2006-05-26 | Benzodiazepine derivatives and uses thereof in medical field |
PCT/IT2006/000401 WO2007015280A1 (en) | 2005-08-03 | 2006-05-26 | Benzodiazepine derivatives and uses thereof in medical field |
US11/997,689 US20080249080A1 (en) | 2005-08-03 | 2006-05-26 | Benzodiazepine Derivatives and Uses Thereof on Medical Field |
DE602006009276T DE602006009276D1 (de) | 2005-08-03 | 2006-05-26 | Benzodiazepinderivate und anwendungen davon auf dem medizinischen gebiet |
AT06756301T ATE443065T1 (de) | 2005-08-03 | 2006-05-26 | Benzodiazepinderivate und anwendungen davon auf dem medizinischen gebiet |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT000416A ITRM20050416A1 (it) | 2005-08-03 | 2005-08-03 | Derivati delle benzodiazepine e loro usi in campo medico. |
Publications (1)
Publication Number | Publication Date |
---|---|
ITRM20050416A1 true ITRM20050416A1 (it) | 2007-02-04 |
Family
ID=36889076
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT000416A ITRM20050416A1 (it) | 2005-08-03 | 2005-08-03 | Derivati delle benzodiazepine e loro usi in campo medico. |
Country Status (6)
Country | Link |
---|---|
US (1) | US20080249080A1 (it) |
EP (1) | EP1910383B1 (it) |
AT (1) | ATE443065T1 (it) |
DE (1) | DE602006009276D1 (it) |
IT (1) | ITRM20050416A1 (it) |
WO (1) | WO2007015280A1 (it) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3360879A1 (en) | 2009-02-05 | 2018-08-15 | ImmunoGen, Inc. | Benzodiazepine derivatives as cytotoxic agents |
MX346635B (es) | 2011-02-15 | 2017-03-27 | Immunogen Inc | Derivados citotoxicos de la benzodiazepina. |
EP2887965A1 (en) | 2012-08-22 | 2015-07-01 | ImmunoGen, Inc. | Cytotoxic benzodiazepine derivatives |
ES2815353T3 (es) | 2014-09-03 | 2021-03-29 | Immunogen Inc | Derivados de benzodiazepina citotóxicos |
JP2017527562A (ja) | 2014-09-03 | 2017-09-21 | イミュノジェン・インコーポレーテッド | 細胞毒性ベンゾジアゼピン誘導体 |
WO2018195243A1 (en) | 2017-04-20 | 2018-10-25 | Immunogen, Inc. | Cytotoxic benzodiazepine derivatives and conjugates thereof |
WO2019133652A1 (en) | 2017-12-28 | 2019-07-04 | Immunogen, Inc. | Benzodiazepine derivatives |
CN113661172A (zh) | 2019-03-29 | 2021-11-16 | 伊缪诺金公司 | 用于抑制异常细胞生长或治疗增生性疾病的细胞毒性双苯并二氮杂䓬衍生物及其与细胞结合剂的缀合物 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6156746A (en) * | 1998-08-25 | 2000-12-05 | Bristol-Myers Squibb Company | 1,2,5-benzothiadiazepine-1,1-dioxides with n-2 imidazolylalkyl substituents |
-
2005
- 2005-08-03 IT IT000416A patent/ITRM20050416A1/it unknown
-
2006
- 2006-05-26 WO PCT/IT2006/000401 patent/WO2007015280A1/en active Application Filing
- 2006-05-26 DE DE602006009276T patent/DE602006009276D1/de not_active Expired - Fee Related
- 2006-05-26 AT AT06756301T patent/ATE443065T1/de not_active IP Right Cessation
- 2006-05-26 US US11/997,689 patent/US20080249080A1/en not_active Abandoned
- 2006-05-26 EP EP06756301A patent/EP1910383B1/en not_active Not-in-force
Also Published As
Publication number | Publication date |
---|---|
EP1910383A1 (en) | 2008-04-16 |
WO2007015280A8 (en) | 2008-04-10 |
WO2007015280A1 (en) | 2007-02-08 |
ATE443065T1 (de) | 2009-10-15 |
DE602006009276D1 (de) | 2009-10-29 |
EP1910383B1 (en) | 2009-09-16 |
US20080249080A1 (en) | 2008-10-09 |
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