IT8349450A0 - Determinate pirazolo-chinoline sostituite, procedimento per la loro preparazione, preparati farmaceutici contenenti questi composti e loro impiego terapeutico - Google Patents

Determinate pirazolo-chinoline sostituite, procedimento per la loro preparazione, preparati farmaceutici contenenti questi composti e loro impiego terapeutico

Info

Publication number
IT8349450A0
IT8349450A0 IT8349450A IT4945083A IT8349450A0 IT 8349450 A0 IT8349450 A0 IT 8349450A0 IT 8349450 A IT8349450 A IT 8349450A IT 4945083 A IT4945083 A IT 4945083A IT 8349450 A0 IT8349450 A0 IT 8349450A0
Authority
IT
Italy
Prior art keywords
quinolines
compounds
procedure
preparation
pharmaceutical preparations
Prior art date
Application number
IT8349450A
Other languages
English (en)
Other versions
IT1205349B (it
Inventor
Yokoyama Maokata
Original Assignee
Ciba & Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba & Geigy Ag filed Critical Ciba & Geigy Ag
Publication of IT8349450A0 publication Critical patent/IT8349450A0/it
Application granted granted Critical
Publication of IT1205349B publication Critical patent/IT1205349B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents
    • A61P39/02Antidotes
IT49450/83A 1982-12-08 1983-12-06 Determinate pirazolo-chinoline sostituite,procedimento per la loro preparazione,preparati farmaceutici contenenti questi composti e loro impiego terapeutico IT1205349B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/447,825 US4524146A (en) 1982-12-08 1982-12-08 Certain -2-heterocycle substituted pyrazoloquinolines

Publications (2)

Publication Number Publication Date
IT8349450A0 true IT8349450A0 (it) 1983-12-06
IT1205349B IT1205349B (it) 1989-03-15

Family

ID=23777905

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49450/83A IT1205349B (it) 1982-12-08 1983-12-06 Determinate pirazolo-chinoline sostituite,procedimento per la loro preparazione,preparati farmaceutici contenenti questi composti e loro impiego terapeutico

Country Status (9)

Country Link
US (1) US4524146A (it)
JP (1) JPS59110694A (it)
BE (1) BE898383A (it)
CH (1) CH656127A5 (it)
DE (1) DE3343922A1 (it)
FR (1) FR2537584B1 (it)
GB (1) GB2131801B (it)
IT (1) IT1205349B (it)
NL (1) NL8304224A (it)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2549833B1 (fr) * 1983-07-26 1985-11-08 Roussel Uclaf Derives de la pyrazolo /4,3-c/ cinnolin-3-one, leurs sels, procede de preparation, application a titre de medicaments, compositions les renfermant et produits intermediaires
CA1263651A (en) * 1984-07-09 1989-12-05 Ciba-Geigy Ag Certain ring-fused pyrazolo ¬3,4-d|-pyridin-3-one derivatives
US4602014A (en) * 1984-07-09 1986-07-22 Ciba-Geigy Corporation Ring-fused pyrazolo[3,4-d]-pyridin-3-one derivatives as benzodiazepine receptor modulators
PH21213A (en) * 1984-10-26 1987-08-21 Fujisawa Pharmaceutical Co Benzene- and pyrazole- fused heterocyclic compound and pharmaceutical composition comprising the same
JPS61112075A (ja) * 1984-11-05 1986-05-30 Shionogi & Co Ltd チエニルピラゾロキノリン誘導体
US4591589A (en) * 1985-01-16 1986-05-27 Roussel Uclaf 2-aryl pyrazolo[4,3-c]cinnolin-3-ones
US4758427A (en) * 1985-08-08 1988-07-19 Ciba-Geigy Corporation Enhanced absorption of psychoactive 2-aryl-pyrazolo quinolines as a solid molecular dispersion in polyvinylpyrrolidone
US4831013A (en) * 1986-03-20 1989-05-16 Ciba-Geigy Corporation 2-substituted-e-fused-[1,2,4]triazolo[1,5-c]pyrimidines, pharmaceutical compositions, and uses thereof
US4826854A (en) * 1986-11-25 1989-05-02 Ciba-Geigy Corporation Certain cycloalka-(b)-pyrazolo(3,4-d)-pyridin-3-one derivatives
US5192768A (en) * 1990-09-14 1993-03-09 Kyowa Hakko Kogyo Co., Ltd. Pyrazoloquinoline derivatives
US5334595A (en) * 1992-10-23 1994-08-02 Sterling Winthrop Inc. Pyrazoloquinolones as anticancer agents
ID16283A (id) * 1996-03-20 1997-09-18 Astra Pharma Prod Senyawa yang berguna dibidang farmasi
WO2001038329A1 (fr) * 1999-11-24 2001-05-31 Sumika Fine Chemicals Co., Ltd. Cristaux de mirtazapine anhydre et leur procede d'obtention
US7863266B2 (en) * 2007-06-08 2011-01-04 Helicon Therapeutics, Inc. Therapeutic pyrazoloquinoline urea derivatives
WO2009155527A2 (en) * 2008-06-19 2009-12-23 Progenics Pharmaceuticals, Inc. Phosphatidylinositol 3 kinase inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2009079A1 (it) * 1968-05-22 1970-01-30 Sandoz Sa
ATE8629T1 (de) * 1979-06-21 1984-08-15 Ciba-Geigy Ag Pyrazolochinoline, verfahren zu ihrer herstellung, und pharmazeutische praeparate enthaltend diese verbindungen.
US4312870A (en) * 1979-06-21 1982-01-26 Ciba-Geigy Corporation Pyrazoloquinolines

Also Published As

Publication number Publication date
BE898383A (fr) 1984-06-06
DE3343922A1 (de) 1984-06-28
FR2537584B1 (fr) 1987-01-16
GB2131801A (en) 1984-06-27
US4524146A (en) 1985-06-18
NL8304224A (nl) 1984-07-02
CH656127A5 (de) 1986-06-13
GB2131801B (en) 1986-01-22
IT1205349B (it) 1989-03-15
GB8332274D0 (en) 1984-01-11
FR2537584A1 (fr) 1984-06-15
JPS59110694A (ja) 1984-06-26

Similar Documents

Publication Publication Date Title
IT1179029B (it) Preparati farmaceutici ad attivita antimicrobica e procedimento per la loro preparazione
IT1170286B (it) Derivati del labdano, procedimento per la loro preparazione, e composizioni farmaceutiche contenenti derivati del labdano
IT8349450A0 (it) Determinate pirazolo-chinoline sostituite, procedimento per la loro preparazione, preparati farmaceutici contenenti questi composti e loro impiego terapeutico
IT8248970A0 (it) Derivati xantinici, procedimento per la loro preparazione, composizione farmaceutiche che li contengono e loro impiego terapeutico
IT8348734A0 (it) Impiego di derivati dello zucchero per la profilassi e terapia di infezioni da virus e preparati farmaceutici che contengono tali composti
DE3378208D1 (en) Substituted azabicycloalkanes, their use, pharmaceutical preparations containing these compounds and process for preparing these compounds
IT1171361B (it) Amminociclopentanon-ammidi e procedimento per la loro preparazione e formulazione farmaceutica
IT1201523B (it) Eterociclilfenilfomramidine,processi per la loro preparazione e loro uso farmaceutico
IT1194158B (it) Carbacicline,procedimento per la loro preparazione e loro impiego come medicinali
IT8319219A0 (it) Derivati di arilossipropanolamina, procedimento per la loro preparazione composizioni farmaceutiche cheli contengono e loro impiego terapeutico
IT1177980B (it) Composti amminometilici, procetimento per produrli, preparati farmaceutici che li contengono
IT8321721A0 (it) Composti polienici,procedimento per la loro preparazione e preparati farmaceutici che li contengono
IT8349055A0 (it) B-osso-l-carbammoil-pirrolpropionitrile, procedimento per la loro produzione, preparati farmaceutici con tenenti questi composti, nonche' il loro impiego terapeutico
IT1211944B (it) Derivati azolici,procedimento per la loro produzione,preparati farmaceutici che li contengono,e loro impiego
IT8621837A0 (it) Nuovi derivati biciclici del catecolo, procedimento per la loro preparazione e composizioni terapeutiche che li contengono.
IT8349163A0 (it) 5h-dibenz/b,f/azepin-5-carbossamidi loro prodotti intermedi, preparati farmaceutici che le contengono, procedimento per produrle e loro impiego
IT7847545A0 (it) Preparati farmaceutici antidiarroici e procedimento per la loro produzione ed applicazione
IT8567216A0 (it) Composti pteridinici relativi procedimenti di preparazione e preparati farmaceutici che li contengono
IT8348726A0 (it) Composti di amminoimidazolile, procedimenti per la loro produzione e preparati farmaceutici che contengono questi composti
IT1172268B (it) Piperidinoguanidine sostituite,procedimento per la loro preparazione e composizioni farmaceutiche che le contengono
IT8249761A0 (it) Imidazo[4,5-c]chinoline, procedimenti per la loro preparazione, preparati farmaceutici contenenti questi composti nonche' loro impiego terapeutico
IT8321607A0 (it) Preparati farmaceutici topici adattivita' antisettica ed antiinfiammatoria spinta, eprocedimento per la loro preparazione.
HK42585A (en) Novel oxothia compounds,processes for their preparation,pharmaceutical preparations containing these compounds and such compounds for therapeutic use
IT1148712B (it) Derivati della n-acetilcisteina,procedimento per la loro preparazione e preparati farmaceutici che li contengono
IT8222637A0 (it) Eterociclilfenilsolfonil e fosfonilamidine sostituite, procedimento per la loro preparazione e loro uso farmaceutico.