IT7820007A0 - Relativo procedimento di nuovi ammino derivati della preparazione. oleandomicina quattro sostituiti e - Google Patents
Relativo procedimento di nuovi ammino derivati della preparazione. oleandomicina quattro sostituiti eInfo
- Publication number
- IT7820007A0 IT7820007A0 IT7820007A IT2000778A IT7820007A0 IT 7820007 A0 IT7820007 A0 IT 7820007A0 IT 7820007 A IT7820007 A IT 7820007A IT 2000778 A IT2000778 A IT 2000778A IT 7820007 A0 IT7820007 A0 IT 7820007A0
- Authority
- IT
- Italy
- Prior art keywords
- oleandomycin
- substitutes
- preparation
- related process
- amino derivatives
- Prior art date
Links
- RZPAKFUAFGMUPI-UHFFFAOYSA-N Oleandomycin Natural products O1C(C)C(O)C(OC)CC1OC1C(C)C(=O)OC(C)C(C)C(O)C(C)C(=O)C2(OC2)CC(C)C(OC2C(C(CC(C)O2)N(C)C)O)C1C RZPAKFUAFGMUPI-UHFFFAOYSA-N 0.000 title 1
- 239000004104 Oleandomycin Substances 0.000 title 1
- 150000001412 amines Chemical class 0.000 title 1
- RZPAKFUAFGMUPI-KGIGTXTPSA-N oleandomycin Chemical compound O1[C@@H](C)[C@H](O)[C@@H](OC)C[C@@H]1O[C@@H]1[C@@H](C)C(=O)O[C@H](C)[C@H](C)[C@H](O)[C@@H](C)C(=O)[C@]2(OC2)C[C@H](C)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C RZPAKFUAFGMUPI-KGIGTXTPSA-N 0.000 title 1
- 229960002351 oleandomycin Drugs 0.000 title 1
- 235000019367 oleandomycin Nutrition 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/765,488 US4085119A (en) | 1977-02-04 | 1977-02-04 | 4-Substituted amino derivatives of oleandomycin |
Publications (2)
Publication Number | Publication Date |
---|---|
IT7820007A0 true IT7820007A0 (it) | 1978-02-03 |
IT1094210B IT1094210B (it) | 1985-07-26 |
Family
ID=25073690
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT20007/78A IT1094210B (it) | 1977-02-04 | 1978-02-03 | Nuovi emmino derivati della oleandomicina quattro sostituiti e relativo procedimento di preparazione |
Country Status (11)
Country | Link |
---|---|
US (2) | US4085119A (it) |
JP (1) | JPS5398983A (it) |
BE (1) | BE863620A (it) |
DE (1) | DE2804517C3 (it) |
DK (1) | DK148035C (it) |
FR (1) | FR2379551A1 (it) |
GB (1) | GB1593644A (it) |
IE (1) | IE46394B1 (it) |
IT (1) | IT1094210B (it) |
LU (1) | LU79005A1 (it) |
NL (1) | NL171588C (it) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4189590A (en) * | 1976-08-06 | 1980-02-19 | Pfizer Inc. | Semi-synthetic oleandomycin derivatives--C8 modifications |
US4124755A (en) * | 1978-01-03 | 1978-11-07 | Pfizer Inc. | 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives |
US4180654A (en) * | 1978-01-03 | 1979-12-25 | Pfizer Inc. | 4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate |
US4133950A (en) * | 1978-01-03 | 1979-01-09 | Pfizer Inc. | 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters |
US4166901A (en) * | 1978-01-03 | 1979-09-04 | Pfizer Inc. | 4"-Deoxy-4"-arylglyoxamido- and aroylthioformamido derivatives of oleandomycin and its esters |
US4316010A (en) * | 1981-01-02 | 1982-02-16 | Pfizer Inc. | Cis-C3 "C4 "-carbonate derivatives of O-demethyloleandomycin and intermediates therefor |
IT1169013B (it) | 1981-01-09 | 1987-05-20 | Pierrel Spa | Composti macrolidici ad attivita' antibiotica, procedimento e microorganismo per la loro preparazione e relative composizioni farmaceutiche |
US4336368A (en) * | 1981-04-20 | 1982-06-22 | Pfizer Inc. | 4 Deoxy-4-methylene oleandomycin and derivatives thereof |
US4427663A (en) | 1982-03-16 | 1984-01-24 | Merck & Co., Inc. | 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof |
US4808590A (en) * | 1987-07-17 | 1989-02-28 | Harbor Branch Oceanographic Institution, Inc. | Antiviral, antitumor and antifungal compositions and their methods of use |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2870138A (en) * | 1953-08-13 | 1959-01-20 | Upjohn Co | Erythromycin salts |
US3357999A (en) * | 1965-12-23 | 1967-12-12 | Abbott Lab | Anhydrotriacetylerythronolide b |
US3842068A (en) * | 1972-06-15 | 1974-10-15 | Abbott Lab | 8-epi-erythromycins |
US3836519A (en) * | 1973-05-04 | 1974-09-17 | Abbott Lab | Sulfonyl derivatives of erythromycin |
US3928387A (en) * | 1974-02-04 | 1975-12-23 | Hoffmann La Roche | Antibiotic 1745A/X and methods for the production thereof |
US3963696A (en) * | 1975-02-21 | 1976-06-15 | Abbott Laboratories | 6,6A-AND 6,7-Anhydroerythromycin B and derivatives thereof |
US4036853A (en) * | 1976-08-06 | 1977-07-19 | Pfizer Inc. | Semi-synthetic oleandomycin derivatives-C8 modifications |
-
1977
- 1977-02-04 US US05/765,488 patent/US4085119A/en not_active Expired - Lifetime
-
1978
- 1978-01-17 US US05/870,160 patent/US4140848A/en not_active Expired - Lifetime
- 1978-02-02 DE DE2804517A patent/DE2804517C3/de not_active Expired
- 1978-02-02 GB GB4166/78A patent/GB1593644A/en not_active Expired
- 1978-02-03 BE BE184872A patent/BE863620A/xx not_active IP Right Cessation
- 1978-02-03 FR FR7803067A patent/FR2379551A1/fr active Granted
- 1978-02-03 DK DK51678A patent/DK148035C/da not_active IP Right Cessation
- 1978-02-03 IT IT20007/78A patent/IT1094210B/it active
- 1978-02-03 LU LU79005A patent/LU79005A1/xx unknown
- 1978-02-03 JP JP1135178A patent/JPS5398983A/ja active Granted
- 1978-02-03 IE IE234/78A patent/IE46394B1/en unknown
- 1978-02-03 NL NLAANVRAGE7801261,A patent/NL171588C/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DE2804517B2 (de) | 1980-09-25 |
LU79005A1 (fr) | 1979-09-06 |
NL171588C (nl) | 1983-04-18 |
DE2804517A1 (de) | 1978-08-10 |
FR2379551A1 (fr) | 1978-09-01 |
NL7801261A (nl) | 1978-08-08 |
DE2804517C3 (de) | 1981-05-07 |
DK51678A (da) | 1978-08-05 |
IT1094210B (it) | 1985-07-26 |
DK148035B (da) | 1985-02-11 |
DK148035C (da) | 1985-07-15 |
GB1593644A (en) | 1981-07-22 |
FR2379551B1 (it) | 1980-08-29 |
BE863620A (fr) | 1978-08-03 |
US4140848A (en) | 1979-02-20 |
JPS5628918B2 (it) | 1981-07-04 |
US4085119A (en) | 1978-04-18 |
IE46394B1 (en) | 1983-06-01 |
JPS5398983A (en) | 1978-08-29 |
IE780234L (en) | 1978-08-04 |
NL171588B (nl) | 1982-11-16 |
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