IT1402925B1 - Processo per la produzione di aliskiren - Google Patents

Processo per la produzione di aliskiren

Info

Publication number
IT1402925B1
IT1402925B1 ITMI2010A002271A ITMI20102271A IT1402925B1 IT 1402925 B1 IT1402925 B1 IT 1402925B1 IT MI2010A002271 A ITMI2010A002271 A IT MI2010A002271A IT MI20102271 A ITMI20102271 A IT MI20102271A IT 1402925 B1 IT1402925 B1 IT 1402925B1
Authority
IT
Italy
Prior art keywords
aliskiren
production process
production
aliskiren production
Prior art date
Application number
ITMI2010A002271A
Other languages
English (en)
Inventor
Romina Vitale
Luca Banfi
Luca Carcone
Marcello Rasparini
Stephen Roseblade
Elena Cini
Adele Russo
Maurizio Taddei
Antonio Carlo Zanotti-Gerosa
Renata Riva
Original Assignee
Chemo Iberica Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemo Iberica Sa filed Critical Chemo Iberica Sa
Priority to ITMI2010A002271A priority Critical patent/IT1402925B1/it
Priority to TW100118590A priority patent/TW201202178A/zh
Priority to UY0001033425A priority patent/UY33425A/es
Priority to US13/701,440 priority patent/US9346745B2/en
Priority to PCT/EP2011/059196 priority patent/WO2011151442A2/en
Priority to EP11728793.8A priority patent/EP2576500A2/en
Priority to ARP110101938A priority patent/AR081836A1/es
Priority to CA2801126A priority patent/CA2801126A1/en
Publication of ITMI20102271A1 publication Critical patent/ITMI20102271A1/it
Application granted granted Critical
Publication of IT1402925B1 publication Critical patent/IT1402925B1/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/20—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/26—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D307/30—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/32—Oxygen atoms
    • C07D307/33—Oxygen atoms in position 2, the oxygen atom being in its keto or unsubstituted enol form

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ITMI2010A002271A 2010-06-04 2010-12-10 Processo per la produzione di aliskiren IT1402925B1 (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
ITMI2010A002271A IT1402925B1 (it) 2010-12-10 2010-12-10 Processo per la produzione di aliskiren
TW100118590A TW201202178A (en) 2010-06-04 2011-05-27 Process for producing Aliskiren
UY0001033425A UY33425A (es) 2010-06-04 2011-06-02 Proceso para la producción de aliskiren
US13/701,440 US9346745B2 (en) 2010-06-04 2011-06-03 Process for producing Aliskiren
PCT/EP2011/059196 WO2011151442A2 (en) 2010-06-04 2011-06-03 Process for producing aliskiren
EP11728793.8A EP2576500A2 (en) 2010-06-04 2011-06-03 Process for producing aliskiren
ARP110101938A AR081836A1 (es) 2010-06-04 2011-06-03 Proceso para la produccion de aliskiren, procedimiento para la preparacion de intermediarios para su sintesis y compuestos necesarios para obtener estos ultimos
CA2801126A CA2801126A1 (en) 2010-06-04 2011-06-03 Process for producing aliskiren

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI2010A002271A IT1402925B1 (it) 2010-12-10 2010-12-10 Processo per la produzione di aliskiren

Publications (2)

Publication Number Publication Date
ITMI20102271A1 ITMI20102271A1 (it) 2012-06-11
IT1402925B1 true IT1402925B1 (it) 2013-09-27

Family

ID=43736927

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI2010A002271A IT1402925B1 (it) 2010-06-04 2010-12-10 Processo per la produzione di aliskiren

Country Status (1)

Country Link
IT (1) IT1402925B1 (it)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY119161A (en) * 1994-04-18 2005-04-30 Novartis Ag Delta-amino-gamma-hydroxy-omega-aryl-alkanoic acid amides with enzyme especially renin inhibiting activities
ES2220776T3 (es) * 2000-07-25 2004-12-16 Speedel Pharma Ag Proceso para la obtencion de octanoil-amidas sustituidas.
ES2442266T3 (es) * 2007-12-24 2014-02-10 Dsm Ip Assets B.V. Síntesis convergente de inhibidores de renina y compuestos intermedios útiles en la misma

Also Published As

Publication number Publication date
ITMI20102271A1 (it) 2012-06-11

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