IT1292438B1 - Derivati peptidomimetici inibitori suicidi della proliferazione del hiv - Google Patents

Derivati peptidomimetici inibitori suicidi della proliferazione del hiv

Info

Publication number
IT1292438B1
IT1292438B1 IT97MI001545A ITMI971545A IT1292438B1 IT 1292438 B1 IT1292438 B1 IT 1292438B1 IT 97MI001545 A IT97MI001545 A IT 97MI001545A IT MI971545 A ITMI971545 A IT MI971545A IT 1292438 B1 IT1292438 B1 IT 1292438B1
Authority
IT
Italy
Prior art keywords
suicide inhibitors
hiv proliferation
peptidomimetic derivatives
peptidomimetic
derivatives
Prior art date
Application number
IT97MI001545A
Other languages
English (en)
Italian (it)
Inventor
Domenico Ungheri
Franco Pellacini
Stefano Romagnano
Jean-Louis Kraus
Jean Claude Chermann
Original Assignee
Zambon Spa
Inst Nat Sante Rech Med
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa, Inst Nat Sante Rech Med filed Critical Zambon Spa
Priority to IT97MI001545A priority Critical patent/IT1292438B1/it
Publication of ITMI971545A0 publication Critical patent/ITMI971545A0/it
Priority to EP98939556A priority patent/EP1001969A1/en
Priority to PCT/EP1998/003970 priority patent/WO1999001470A2/en
Priority to AU88025/98A priority patent/AU8802598A/en
Publication of ITMI971545A1 publication Critical patent/ITMI971545A1/it
Application granted granted Critical
Publication of IT1292438B1 publication Critical patent/IT1292438B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06017Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/0606Dipeptides with the first amino acid being neutral and aliphatic the side chain containing heteroatoms not provided for by C07K5/06086 - C07K5/06139, e.g. Ser, Met, Cys, Thr
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
IT97MI001545A 1997-06-30 1997-06-30 Derivati peptidomimetici inibitori suicidi della proliferazione del hiv IT1292438B1 (it)

Priority Applications (4)

Application Number Priority Date Filing Date Title
IT97MI001545A IT1292438B1 (it) 1997-06-30 1997-06-30 Derivati peptidomimetici inibitori suicidi della proliferazione del hiv
EP98939556A EP1001969A1 (en) 1997-06-30 1998-06-29 Peptidomimetic derivatives suicidal inhibitors of the hiv proliferation
PCT/EP1998/003970 WO1999001470A2 (en) 1997-06-30 1998-06-29 Peptidomimetic derivatives suicidal inhibitors of the hiv proliferation
AU88025/98A AU8802598A (en) 1997-06-30 1998-06-29 Peptidomimetic derivatives suicidal inhibitors of the hiv proliferation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT97MI001545A IT1292438B1 (it) 1997-06-30 1997-06-30 Derivati peptidomimetici inibitori suicidi della proliferazione del hiv

Publications (3)

Publication Number Publication Date
ITMI971545A0 ITMI971545A0 (enrdf_load_stackoverflow) 1997-06-30
ITMI971545A1 ITMI971545A1 (it) 1998-12-30
IT1292438B1 true IT1292438B1 (it) 1999-02-08

Family

ID=11377465

Family Applications (1)

Application Number Title Priority Date Filing Date
IT97MI001545A IT1292438B1 (it) 1997-06-30 1997-06-30 Derivati peptidomimetici inibitori suicidi della proliferazione del hiv

Country Status (4)

Country Link
EP (1) EP1001969A1 (enrdf_load_stackoverflow)
AU (1) AU8802598A (enrdf_load_stackoverflow)
IT (1) IT1292438B1 (enrdf_load_stackoverflow)
WO (1) WO1999001470A2 (enrdf_load_stackoverflow)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU563196B2 (en) * 1982-05-18 1987-07-02 Smithkline Beckman Corporation Peptide prodrug transport system
US5221667A (en) * 1990-01-22 1993-06-22 Warner-Lambert Company Renin inhibiting peptides having an α-heteroatom amino acid at the P3 position
FR2736055B1 (fr) * 1995-06-29 1997-09-12 Laphal Sa Lab Nouveaux thiophenoxy peptides, leur procede de preparation et les compositions pharmaceutiques en renfermant

Also Published As

Publication number Publication date
AU8802598A (en) 1999-01-25
WO1999001470A2 (en) 1999-01-14
WO1999001470A3 (en) 1999-03-25
ITMI971545A1 (it) 1998-12-30
EP1001969A1 (en) 2000-05-24
ITMI971545A0 (enrdf_load_stackoverflow) 1997-06-30

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Legal Events

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