IT1216772B - INDOLATION DERIVATIVES, PROCEDURE TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM FOR THE TREATMENT OF Migraine - Google Patents

INDOLATION DERIVATIVES, PROCEDURE TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM FOR THE TREATMENT OF Migraine

Info

Publication number
IT1216772B
IT1216772B IT8747506A IT4750687A IT1216772B IT 1216772 B IT1216772 B IT 1216772B IT 8747506 A IT8747506 A IT 8747506A IT 4750687 A IT4750687 A IT 4750687A IT 1216772 B IT1216772 B IT 1216772B
Authority
IT
Italy
Prior art keywords
indolation
migraine
derivatives
prepare
procedure
Prior art date
Application number
IT8747506A
Other languages
Italian (it)
Other versions
IT8747506A0 (en
Inventor
Mills Keith
Coates Ian Harold
David Edmund Bays
Colin Frederick Webb
Michael Dennis Dowle
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of IT8747506A0 publication Critical patent/IT8747506A0/en
Application granted granted Critical
Publication of IT1216772B publication Critical patent/IT1216772B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
IT8747506A 1986-01-08 1987-01-08 INDOLATION DERIVATIVES, PROCEDURE TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM FOR THE TREATMENT OF Migraine IT1216772B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868600398A GB8600398D0 (en) 1986-01-08 1986-01-08 Chemical compounds

Publications (2)

Publication Number Publication Date
IT8747506A0 IT8747506A0 (en) 1987-01-08
IT1216772B true IT1216772B (en) 1990-03-14

Family

ID=10591075

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8747506A IT1216772B (en) 1986-01-08 1987-01-08 INDOLATION DERIVATIVES, PROCEDURE TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM FOR THE TREATMENT OF Migraine

Country Status (11)

Country Link
JP (1) JPS62228057A (en)
AT (1) AT386197B (en)
AU (1) AU597324B2 (en)
BE (1) BE1000072A4 (en)
CH (1) CH671017A5 (en)
DE (1) DE3700407A1 (en)
FR (1) FR2595352B1 (en)
GB (2) GB8600398D0 (en)
IT (1) IT1216772B (en)
NL (1) NL8700027A (en)
ZA (1) ZA87104B (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
GB8819024D0 (en) * 1988-08-10 1988-09-14 Glaxo Group Ltd Chemical compounds
RU2160736C2 (en) * 1990-06-07 2000-12-20 Зенека Лимитед Indole derivatives and physiologically acceptable salts and solvates thereof, methods of preparing thereof, drug for treatment or prophylaxes of clinical states for which administration of 5-ht1-like receptor agonist, and method of preparing thereof
GB9012672D0 (en) * 1990-06-07 1990-08-01 Wellcome Found Therapeutic heterocyclic compounds
TW263508B (en) * 1991-02-12 1995-11-21 Pfizer
US5206377A (en) * 1991-12-05 1993-04-27 Whitby Research, Inc. Compounds useful as antiproliferative agents
GB9201038D0 (en) * 1992-01-16 1992-03-11 Glaxo Group Ltd Chemical compounds
US5409941A (en) * 1992-02-03 1995-04-25 Pfizer Inc. 5-heteroyl indole derivatives
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
US5496957A (en) * 1993-09-01 1996-03-05 Virginia Commonwealth University Tryptamine analogs with 5-HT1D selectivity
WO1995006638A1 (en) * 1993-09-01 1995-03-09 Allelix Biopharmaceuticals Inc. Tryptamine analogs with 5-ht1d selectivity
CN1729174B (en) * 2002-12-20 2015-10-21 西巴特殊化学品控股有限公司 The synthesis of amine and the intermediate for the synthesis of amine

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB147107A (en) * 1915-04-06 1921-10-07 Zeiss Carl Improvements in finders for photographic apparatus
GB145459A (en) * 1917-03-24 1921-04-21 Anschuetz & Co Gmbh Improvements in indicators for the turning of aircraft about a vertical axis
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds
AU550010B2 (en) * 1980-08-12 1986-02-27 Glaxo Group Limited 5-tryptaminoacetamides, carbamates and ureas
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
FR2903394B1 (en) * 2006-07-05 2008-09-19 Pierre Marcelli EXPANDABLE CHUCK REEL FOR SPOOL
BRPI0808952A2 (en) * 2007-04-06 2014-08-26 Gaiasoft Ip Ltd "CONTENT DELIVERY SYSTEM, INTERMEDIATE CONTENT MECHANISM, RELIABLE PROFILE DATA MECHANISM AND METHOD FOR DELIVERING CONTENT"

Also Published As

Publication number Publication date
AU6741887A (en) 1987-07-09
DE3700407A1 (en) 1987-07-09
AT386197B (en) 1988-07-11
GB8600398D0 (en) 1986-02-12
BE1000072A4 (en) 1988-02-02
NL8700027A (en) 1987-08-03
FR2595352B1 (en) 1990-07-13
ZA87104B (en) 1987-12-30
IT8747506A0 (en) 1987-01-08
ATA2487A (en) 1987-12-15
GB8700381D0 (en) 1987-02-11
GB2186874A (en) 1987-08-26
CH671017A5 (en) 1989-07-31
FR2595352A1 (en) 1987-09-11
JPS62228057A (en) 1987-10-06
AU597324B2 (en) 1990-05-31
GB2186874B (en) 1990-02-07

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