IT1182089B - INDOLATION DERIVATIVES, PROCEDURE, TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

INDOLATION DERIVATIVES, PROCEDURE, TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
IT1182089B
IT1182089B IT48921/85A IT4892185A IT1182089B IT 1182089 B IT1182089 B IT 1182089B IT 48921/85 A IT48921/85 A IT 48921/85A IT 4892185 A IT4892185 A IT 4892185A IT 1182089 B IT1182089 B IT 1182089B
Authority
IT
Italy
Prior art keywords
indolation
derivatives
prepare
procedure
pharmaceutical compositions
Prior art date
Application number
IT48921/85A
Other languages
Italian (it)
Other versions
IT8548921A0 (en
Inventor
David Edmund Bays
Colin Frederick Webb
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of IT8548921A0 publication Critical patent/IT8548921A0/en
Application granted granted Critical
Publication of IT1182089B publication Critical patent/IT1182089B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
IT48921/85A 1984-12-13 1985-12-12 INDOLATION DERIVATIVES, PROCEDURE, TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IT1182089B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB848431426A GB8431426D0 (en) 1984-12-13 1984-12-13 Chemical compounds

Publications (2)

Publication Number Publication Date
IT8548921A0 IT8548921A0 (en) 1985-12-12
IT1182089B true IT1182089B (en) 1987-09-30

Family

ID=10571103

Family Applications (1)

Application Number Title Priority Date Filing Date
IT48921/85A IT1182089B (en) 1984-12-13 1985-12-12 INDOLATION DERIVATIVES, PROCEDURE, TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (11)

Country Link
JP (1) JPS61151172A (en)
AU (1) AU579687B2 (en)
BE (1) BE903846A (en)
CH (1) CH667454A5 (en)
DE (1) DE3543982A1 (en)
FR (1) FR2574793B1 (en)
GB (2) GB8431426D0 (en)
IT (1) IT1182089B (en)
NL (1) NL8503424A (en)
SE (1) SE8505887L (en)
ZA (1) ZA859520B (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds
GB8607824D0 (en) * 1986-03-27 1986-04-30 Glaxo Group Ltd Chemical compounds
GB8614287D0 (en) * 1986-06-12 1986-07-16 Glaxo Group Ltd Chemical compounds
US4894386A (en) * 1987-04-15 1990-01-16 Ici Americas Inc. Aliphatic carboxamides
GB8719167D0 (en) * 1987-08-13 1987-09-23 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
MC2210A1 (en) * 1990-06-07 1992-11-26 Wellcome Found THERAPEUTIC HETEROCYCLIC COMPOUNDS, THEIR USE AND PROCESS FOR PREPARING THEM
GB9209882D0 (en) * 1992-05-07 1992-06-24 Glaxo Lab Sa Compositions
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
GB9216009D0 (en) * 1992-07-28 1992-09-09 Almirall Lab New indol derivatives
ES2056025B1 (en) * 1992-10-08 1995-05-01 Almirall Lab NEW DERIVATIVES OF INDOL.
FR2707639B1 (en) * 1993-06-30 1995-10-13 Pf Medicament New indole compounds derived from arylamines as selective ligands for the 5HT1D and 5HT1B receptors.
CA2508290C (en) * 2002-12-20 2017-02-28 Ciba Specialty Chemicals Holding Inc. Synthesis of amines and intermediates for the synthesis thereof
WO2005118551A2 (en) 2004-05-28 2005-12-15 Ligand Pharmaceuticals Inc. Thrombopoietin activity modulating compounds and methods
BRPI0516883A (en) 2004-10-25 2008-09-23 Ligand Pharm Inc compounds and methods for modulating thrombopoietin activity
RU2009139931A (en) 2007-03-29 2011-05-10 Асубио Фарма Ко., Лтд. (Jp) DERIVATIVES OF INDOLA WITH INHIBITING ACTIVITY WITH RESPECT TO СPLA2, AND METHODS FOR PRODUCING THEM

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
DE3542698A1 (en) * 1984-12-04 1986-06-05 Glaxo Group Ltd., London INDOLDER DERIVATIVES, METHOD FOR THEIR PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds

Also Published As

Publication number Publication date
GB2168347B (en) 1988-02-03
ZA859520B (en) 1986-08-27
AU579687B2 (en) 1988-12-01
GB2168347A (en) 1986-06-18
IT8548921A0 (en) 1985-12-12
FR2574793A1 (en) 1986-06-20
FR2574793B1 (en) 1988-10-14
GB8431426D0 (en) 1985-01-23
BE903846A (en) 1986-06-12
CH667454A5 (en) 1988-10-14
NL8503424A (en) 1986-07-01
AU5115185A (en) 1986-06-19
JPS61151172A (en) 1986-07-09
SE8505887L (en) 1986-06-14
SE8505887D0 (en) 1985-12-12
GB8530591D0 (en) 1986-01-22
DE3543982A1 (en) 1986-06-19

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