IT1116846B - Procedimento per la preparazione di derivati di naftalinone con attivita'anti-infiammatoria e prodotto ottenuto - Google Patents

Procedimento per la preparazione di derivati di naftalinone con attivita'anti-infiammatoria e prodotto ottenuto

Info

Publication number
IT1116846B
IT1116846B IT47621/79A IT4762179A IT1116846B IT 1116846 B IT1116846 B IT 1116846B IT 47621/79 A IT47621/79 A IT 47621/79A IT 4762179 A IT4762179 A IT 4762179A IT 1116846 B IT1116846 B IT 1116846B
Authority
IT
Italy
Prior art keywords
naphthalinone
derivatives
procedure
preparation
product obtained
Prior art date
Application number
IT47621/79A
Other languages
English (en)
Other versions
IT7947621A0 (it
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of IT7947621A0 publication Critical patent/IT7947621A0/it
Application granted granted Critical
Publication of IT1116846B publication Critical patent/IT1116846B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT47621/79A 1978-01-30 1979-01-12 Procedimento per la preparazione di derivati di naftalinone con attivita'anti-infiammatoria e prodotto ottenuto IT1116846B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/873,644 US4179558A (en) 1978-01-30 1978-01-30 Naphthalenone derivatives and analogs

Publications (2)

Publication Number Publication Date
IT7947621A0 IT7947621A0 (it) 1979-01-12
IT1116846B true IT1116846B (it) 1986-02-10

Family

ID=25362042

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47621/79A IT1116846B (it) 1978-01-30 1979-01-12 Procedimento per la preparazione di derivati di naftalinone con attivita'anti-infiammatoria e prodotto ottenuto

Country Status (7)

Country Link
US (1) US4179558A (it)
JP (1) JPS54103854A (it)
CA (1) CA1093075A (it)
DE (1) DE2856793A1 (it)
FR (1) FR2415617A1 (it)
GB (1) GB2013178B (it)
IT (1) IT1116846B (it)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT70031A (en) * 1992-11-30 1995-09-28 Sankyo Co Alfa, omega-diarylalkane derivatives, their preparation and pharmaceutical compositions containing them

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3313853A (en) * 1963-10-16 1967-04-11 Upjohn Co 2-(tertiaryaminoalkoxyphenyl)-3, 4-dihydronaphthalenes and 2-(tertiaryaminoalkoxyphenyl) -3, 4- dihydro -1(2h)-naphthalenones
US3506653A (en) * 1966-09-12 1970-04-14 Syntex Corp Non-steroid hormonal agents
US3760007A (en) * 1970-06-11 1973-09-18 Schering Corp Bicyclic benzhydrylidene derivatives
DE2646213A1 (de) * 1975-10-28 1977-05-12 Lilly Co Eli Aroylphenylnaphthaline und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
CA1093075A (en) 1981-01-06
GB2013178A (en) 1979-08-08
IT7947621A0 (it) 1979-01-12
DE2856793A1 (de) 1979-08-02
US4179558A (en) 1979-12-18
JPS54103854A (en) 1979-08-15
FR2415617A1 (fr) 1979-08-24
GB2013178B (en) 1982-04-28

Similar Documents

Publication Publication Date Title
IT1113713B (it) Procedimento per la preparazione di derivati di acidi deidrociclimminici dotati di proprieta' ipotensive e prodotto ottenuto
IT1110885B (it) Procedimento per la preparazione di derivati dello acido ftalazin-4-ilacetico e prodotto ottenuto
IT7850335A0 (it) Procedimento per la preparazione di naftiridinoni sostituiti e prodotto ottenuto
IT1117778B (it) Procedimento per la produzione di derivati di pirimidone e prodotto ottenuto
AR221355A1 (es) Procedimiento para la preparacion de derivados de pirrolidinil y pirrolidinilmetil-benzamidas
IT1105178B (it) Procedimento per la preparazione di copoliammidi aromatiche alifatiche e prodotto ottenuto
IT1121483B (it) Derivati di benzotiepinici e procedimento per la loro preparazione
IT1116858B (it) Procedimento per la preparazione di derivati isopropilenici e prodotto ottenuto
IT1114720B (it) Procedimento per la preparazione di derivati di 2-fenilimmino-imidazolidine composizioni farmaceutiche che li contengono e prodotto ottenuto
IT7948266A0 (it) Procedimento per la preparazione di derivati di bicicloottano e di composizioni farmaceutiche che li con tengono e prodotto ottenuto
IT1120407B (it) Procedimento per la preparazione di derivati di pirrolidincarbossaldeide e piperidincarbossaldeide e prodotto ottenuto
IT8083420A0 (it) Derivati d'amino-14 steroidi e procedimento per la loro preparazione.
IT7949743A0 (it) Procedimento per la preparazione di derivati acetilenici di androst-4ene e composizioni farmaceutiche che li contengono e prodotto ottenuto
IT8049718A0 (it) Derivati imidazoliletossi metilici di 1,3-diossolo chinazoline e procedimento per la loro preparazione
IT1110876B (it) Procedimento per la preparazione di 1-idrossiaporfin derivati e prodotto ottenuto
IT1116846B (it) Procedimento per la preparazione di derivati di naftalinone con attivita'anti-infiammatoria e prodotto ottenuto
IT1157750B (it) Procedimento per la preparazione di derivati di acido 1-idrocarbilpirrolo-2-acetico e prodotto ottenuto
IT1116525B (it) Procedimento per la preparazione di n-imminometil-piperidine sostituite e prodotto ottenuto
IT7947594A0 (it) Procedimento per la preparazione di derivati di acido 1,5-ciclo-esadiencarbossilico sostituito e prodotto ottenuto
IT1162702B (it) Derivati di 11-alcanoil-4"-isonitril-oleandomicina
IT1148788B (it) Derivati dell'amminoisochinolina e procedimento per la loro preparazione
IT7951101A0 (it) Derivati di 7 alfa-metossicefalospo rina e procedimento per produrli
IT1119970B (it) Derivati di 7 alfa metossi cefalosporine e procedimento per la loro preparazione
IT7968018A0 (it) Procedimento per la preparazione stereospecifica di derivati di eteri di imidazolil ossime e di derivati di imidazolil ossime
IT1110883B (it) Procedimento per la preparazione di derivati solfossimmidici farmacolo gicamente attivi e prodotto ottenuto