IT1052111B - Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati - Google Patents

Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati

Info

Publication number
IT1052111B
IT1052111B IT48628/72A IT4862872A IT1052111B IT 1052111 B IT1052111 B IT 1052111B IT 48628/72 A IT48628/72 A IT 48628/72A IT 4862872 A IT4862872 A IT 4862872A IT 1052111 B IT1052111 B IT 1052111B
Authority
IT
Italy
Prior art keywords
carboxyls
indazol
benzyl
derivatives
acids
Prior art date
Application number
IT48628/72A
Other languages
English (en)
Italian (it)
Original Assignee
Acraf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Acraf filed Critical Acraf
Priority to IT48628/72A priority Critical patent/IT1052111B/it
Priority to US330902A priority patent/US3895026A/en
Priority to GB780673A priority patent/GB1381422A/en
Priority to IN389/CAL/73A priority patent/IN139264B/en
Priority to CA164,360A priority patent/CA994347A/en
Priority to NLAANVRAGE7302669,A priority patent/NL179729C/xx
Priority to HUAI224A priority patent/HU165172B/hu
Priority to FR7307055A priority patent/FR2181773B1/fr
Priority to DE2310031A priority patent/DE2310031C3/de
Application granted granted Critical
Publication of IT1052111B publication Critical patent/IT1052111B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT48628/72A 1972-02-29 1972-02-29 Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati IT1052111B (it)

Priority Applications (9)

Application Number Priority Date Filing Date Title
IT48628/72A IT1052111B (it) 1972-02-29 1972-02-29 Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati
US330902A US3895026A (en) 1972-02-29 1973-02-09 Substituted 1-benzyl-1h-indazole-3-carboxylic acids and derivatives thereof
GB780673A GB1381422A (en) 1972-02-29 1973-02-16 Substituted 1-benzyl-indazole-3-carboxylic acids
IN389/CAL/73A IN139264B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1972-02-29 1973-02-21
CA164,360A CA994347A (en) 1972-02-29 1973-02-22 Substituted 1-benzyl-indazole-3-carboxylic acids
NLAANVRAGE7302669,A NL179729C (nl) 1972-02-29 1973-02-26 Werkwijze ter bereiding van farmaceutische preparaten op basis van 1h-indazool-3-carbonzuurderivaten alsmede werkwijze ter bereiding van deze 1h-indazool-3-carbonzuurderivaten.
HUAI224A HU165172B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1972-02-29 1973-02-27
FR7307055A FR2181773B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1972-02-29 1973-02-28
DE2310031A DE2310031C3 (de) 1972-02-29 1973-02-28 1 -Benzyl-1 H-indazol-3-carbonsäuren, -amide und -ester

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT48628/72A IT1052111B (it) 1972-02-29 1972-02-29 Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati

Publications (1)

Publication Number Publication Date
IT1052111B true IT1052111B (it) 1981-06-20

Family

ID=11267725

Family Applications (1)

Application Number Title Priority Date Filing Date
IT48628/72A IT1052111B (it) 1972-02-29 1972-02-29 Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati

Country Status (9)

Country Link
US (1) US3895026A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA994347A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE2310031C3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2181773B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1381422A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HU165172B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IN (1) IN139264B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IT (1) IT1052111B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL179729C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1050741B (it) * 1975-12-01 1981-03-20 Acraf Utilizzazione degli acidi i benzil ih indazol 3 carbossilici sostituiti e loro derivati nel campo della contraccezione femminile
US5229408A (en) * 1988-07-15 1993-07-20 Ici Pharma 4-carbamoyl-1,2-dihydro-3H-indazol-3-one derivatives
US5914405A (en) * 1997-10-07 1999-06-22 Eli Lilly And Company Process for preparing 3-substituted indazoles
US6001865A (en) * 1999-05-04 1999-12-14 Angelini Pharmaceuticals Inc. 3-substituted 1-benzyl-1H-indazole derivatives as antifertility agents
KR100424341B1 (ko) * 2001-10-23 2004-03-24 하나제약 주식회사 1-메틸인다졸-3-카르복실산의 제조방법
CA2513572A1 (en) * 2003-01-17 2004-08-05 Threshold Pharmaceuticals, Inc. Treatment of benign prostatic hyperplasia
EP1599196A4 (en) * 2003-01-17 2006-05-31 Threshold Pharmaceuticals Inc COMBINATION THERAPIES FOR CANCER TREATMENT
US7452997B2 (en) * 2004-03-24 2008-11-18 Janssen Pharmaceutica, N.V. Tetrahydro-indazole cannabinoid modulators
WO2005120498A2 (en) * 2004-06-03 2005-12-22 Threshold Pharmaceuticals, Inc. Method for synthesis of lonidamine and related indazole derivatives
WO2006010077A2 (en) * 2004-07-08 2006-01-26 Threshold Pharmaceuticals, Inc. Prodrugs of lonidamine and lonidamine analogs
US7514463B2 (en) * 2004-08-20 2009-04-07 University Of Kansas Lonidamine analogues and their use in male contraception and cancer treatment
CN101735151B (zh) * 2005-08-17 2012-07-04 杭州民生药业有限公司 氯尼达明的结晶形式i、其制备方法和含有所述结晶形式i的组合物
CN101759644B (zh) * 2005-08-17 2011-11-02 杭州民生药业有限公司 氯尼达明的结晶形式iii、其制备方法和含有所述结晶形式iii的组合物
KR20120069658A (ko) * 2009-07-06 2012-06-28 유니버시티 오브 캔사스 생식력 제어를 위한 로니다민 유사체
ES2894919T3 (es) 2015-06-12 2022-02-16 Vettore Llc Inhibidores de MCT4 para el tratamiento de enfermedades
WO2018111904A1 (en) 2016-12-12 2018-06-21 Vettore, LLC Heterocyclic inhibitors of mct4
WO2022061008A2 (en) * 2020-09-17 2022-03-24 Escient Pharmaceuticals, Inc. Modulators of mas-related g-protein receptor x4 and related products and methods

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3007938A (en) * 1959-04-17 1961-11-07 Sterling Drug Inc 1-(3-indazolecarbonyl)-hydrazines and their preparation
US3145215A (en) * 1961-12-19 1964-08-18 Sterling Drug Inc Indazole derivatives
IL28032A (en) * 1966-08-29 1971-08-25 Acraf Indazol-3-yl-oxyalkanoic acids and process for the preparation thereof
US3567721A (en) * 1968-11-29 1971-03-02 Geigy Chem Corp Indazolecarboxylic acids and derivatives thereof
DE1948793A1 (de) * 1969-09-26 1971-04-01 Rhein Chemie Rheinau Gmbh Verfahren zur Herstellung von 4,5,6,7-Tetrahydroindazolen

Also Published As

Publication number Publication date
FR2181773A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1973-12-07
HU165172B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1974-07-27
NL179729C (nl) 1986-11-03
IN139264B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-05-29
DE2310031A1 (de) 1973-09-20
DE2310031C3 (de) 1980-07-31
CA994347A (en) 1976-08-03
DE2310031B2 (de) 1979-11-15
US3895026A (en) 1975-07-15
FR2181773B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1975-12-26
NL7302669A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1973-08-31
GB1381422A (en) 1975-01-22
NL179729B (nl) 1986-06-02

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Legal Events

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ITCP Complementary protection certificate

Free format text: CCP 12

MEDA Supplementary protection certificate for pharmaceutical products: examined

Free format text: CCP 12, 19920115; AZIENDE CHIMICHE RIUNITE ANGELINI F RANCESCO(A.C.R.A.F)S.P.A.