IS5240A - Súlfatsalt af HIV próteasa lata sem hefur bætta upptöku um munn og líffræðilega upptöku - Google Patents
Súlfatsalt af HIV próteasa lata sem hefur bætta upptöku um munn og líffræðilega upptökuInfo
- Publication number
- IS5240A IS5240A IS5240A IS5240A IS5240A IS 5240 A IS5240 A IS 5240A IS 5240 A IS5240 A IS 5240A IS 5240 A IS5240 A IS 5240A IS 5240 A IS5240 A IS 5240A
- Authority
- IS
- Iceland
- Prior art keywords
- protease inhibitor
- hiv protease
- sulfate salt
- improved oral
- biological uptake
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Virology (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- AIDS & HIV (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US4795097P | 1997-05-29 | 1997-05-29 | |
| GBGB9714320.0A GB9714320D0 (en) | 1997-07-07 | 1997-07-07 | Hiv protease inhibitor |
| PCT/US1998/010633 WO1998054178A1 (en) | 1997-05-29 | 1998-05-26 | Sulfate salt of an hiv protease inhibitor having an improved oral absorption and bioavailability |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IS5240A true IS5240A (is) | 1999-11-09 |
Family
ID=26311845
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IS5240A IS5240A (is) | 1997-05-29 | 1999-11-09 | Súlfatsalt af HIV próteasa lata sem hefur bætta upptöku um munn og líffræðilega upptöku |
Country Status (22)
| Country | Link |
|---|---|
| EP (1) | EP0986554A1 (is) |
| JP (1) | JP3267632B2 (is) |
| KR (1) | KR20010013042A (is) |
| CN (1) | CN1257497A (is) |
| AU (1) | AU730245B2 (is) |
| BG (1) | BG103923A (is) |
| BR (1) | BR9809498A (is) |
| CA (1) | CA2291086A1 (is) |
| EA (1) | EA199901095A1 (is) |
| EE (1) | EE9900543A (is) |
| HR (1) | HRP980283A2 (is) |
| HU (1) | HUP0004621A3 (is) |
| ID (1) | ID23858A (is) |
| IL (1) | IL132779A0 (is) |
| IS (1) | IS5240A (is) |
| NO (1) | NO995822L (is) |
| PE (1) | PE75099A1 (is) |
| PL (1) | PL336847A1 (is) |
| SK (1) | SK163299A3 (is) |
| TR (1) | TR199902816T2 (is) |
| TW (1) | TW438799B (is) |
| WO (1) | WO1998054178A1 (is) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2391643C (en) | 1999-11-24 | 2010-01-12 | Merck & Co., Inc. | Gamma-hydroxy-2-(fluoroalkylaminocarbonyl)-1-piperazinepentanamides as hiv protease inhibitors |
| US20020082421A1 (en) * | 2000-09-14 | 2002-06-27 | Abdel-Magid Ahmed F. | Novel solid salt forms of N-[2-[4-[2-(1- methylethoxy)phenyl]-1-piperazinyl]-2-oxo-1piperidineacetamide |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUT74681A (en) * | 1993-12-15 | 1997-01-28 | Merck & Co Inc | N-(2-hydroxy-1-indenyl)-2-phenylmethyl-4-hydroxy-5-(2-carboxamido-piperazinyl)-pentaneamide derivatives of hiv protease inhibitor activity and phrmaceutical compositions contining them |
-
1998
- 1998-05-20 TW TW087107834A patent/TW438799B/zh active
- 1998-05-26 EP EP98923741A patent/EP0986554A1/en not_active Withdrawn
- 1998-05-26 KR KR1019997011018A patent/KR20010013042A/ko not_active Application Discontinuation
- 1998-05-26 CN CN98805372A patent/CN1257497A/zh active Pending
- 1998-05-26 SK SK1632-99A patent/SK163299A3/sk unknown
- 1998-05-26 PL PL98336847A patent/PL336847A1/xx unknown
- 1998-05-26 CA CA002291086A patent/CA2291086A1/en not_active Abandoned
- 1998-05-26 ID IDW991462A patent/ID23858A/id unknown
- 1998-05-26 AU AU75959/98A patent/AU730245B2/en not_active Ceased
- 1998-05-26 HU HU0004621A patent/HUP0004621A3/hu unknown
- 1998-05-26 EE EEP199900543A patent/EE9900543A/xx unknown
- 1998-05-26 JP JP50079999A patent/JP3267632B2/ja not_active Expired - Fee Related
- 1998-05-26 TR TR1999/02816T patent/TR199902816T2/xx unknown
- 1998-05-26 IL IL13277998A patent/IL132779A0/xx unknown
- 1998-05-26 EA EA199901095A patent/EA199901095A1/ru unknown
- 1998-05-26 BR BR9809498-0A patent/BR9809498A/pt not_active Application Discontinuation
- 1998-05-26 WO PCT/US1998/010633 patent/WO1998054178A1/en not_active Application Discontinuation
- 1998-05-28 HR HR9714320.0A patent/HRP980283A2/hr not_active Application Discontinuation
- 1998-05-28 PE PE1998000432A patent/PE75099A1/es not_active Application Discontinuation
-
1999
- 1999-11-09 IS IS5240A patent/IS5240A/is unknown
- 1999-11-24 BG BG103923A patent/BG103923A/xx unknown
- 1999-11-26 NO NO995822A patent/NO995822L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| HUP0004621A3 (en) | 2002-04-29 |
| PL336847A1 (en) | 2000-07-17 |
| PE75099A1 (es) | 1999-08-11 |
| HRP980283A2 (en) | 1999-08-31 |
| WO1998054178A1 (en) | 1998-12-03 |
| NO995822L (no) | 2000-01-28 |
| CA2291086A1 (en) | 1998-12-03 |
| HUP0004621A2 (hu) | 2002-03-28 |
| AU730245B2 (en) | 2001-03-01 |
| NO995822D0 (no) | 1999-11-26 |
| KR20010013042A (ko) | 2001-02-26 |
| EP0986554A1 (en) | 2000-03-22 |
| BR9809498A (pt) | 2000-06-20 |
| TW438799B (en) | 2001-06-07 |
| SK163299A3 (en) | 2000-07-11 |
| IL132779A0 (en) | 2001-03-19 |
| TR199902816T2 (xx) | 2000-02-21 |
| CN1257497A (zh) | 2000-06-21 |
| BG103923A (en) | 2000-06-30 |
| AU7595998A (en) | 1998-12-30 |
| JP2000513747A (ja) | 2000-10-17 |
| EA199901095A1 (ru) | 2000-08-28 |
| EE9900543A (et) | 2000-06-15 |
| JP3267632B2 (ja) | 2002-03-18 |
| ID23858A (id) | 2000-05-25 |
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