IL98691A - Tricyclic macrolides containing heteroatoms their preparation and pharmaceutical compositions containing them - Google Patents

Tricyclic macrolides containing heteroatoms their preparation and pharmaceutical compositions containing them

Info

Publication number
IL98691A
IL98691A IL9869191A IL9869191A IL98691A IL 98691 A IL98691 A IL 98691A IL 9869191 A IL9869191 A IL 9869191A IL 9869191 A IL9869191 A IL 9869191A IL 98691 A IL98691 A IL 98691A
Authority
IL
Israel
Prior art keywords
compound
formula
positions
optionally
hydroxy
Prior art date
Application number
IL9869191A
Other languages
English (en)
Other versions
IL98691A0 (en
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IL98691A0 publication Critical patent/IL98691A0/xx
Publication of IL98691A publication Critical patent/IL98691A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL9869191A 1990-07-02 1991-07-01 Tricyclic macrolides containing heteroatoms their preparation and pharmaceutical compositions containing them IL98691A (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
DE4021191 1990-07-02
DE4034477 1990-10-30
DE4034478 1990-10-30
DE4034480 1990-10-30
DE4034476 1990-10-30
DE4034479 1990-10-30
DE4115132 1991-05-08

Publications (2)

Publication Number Publication Date
IL98691A0 IL98691A0 (en) 1992-07-15
IL98691A true IL98691A (en) 1996-10-16

Family

ID=27561539

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9869191A IL98691A (en) 1990-07-02 1991-07-01 Tricyclic macrolides containing heteroatoms their preparation and pharmaceutical compositions containing them

Country Status (11)

Country Link
EP (1) EP0465426A1 (cs)
JP (1) JPH04230388A (cs)
AU (1) AU648806B2 (cs)
CA (1) CA2045989A1 (cs)
CS (1) CS201191A3 (cs)
FI (1) FI913182L (cs)
HU (1) HUT58338A (cs)
IE (1) IE912297A1 (cs)
IL (1) IL98691A (cs)
MY (1) MY110418A (cs)
NZ (1) NZ238809A (cs)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5708002A (en) * 1991-09-05 1998-01-13 Abbott Laboratories Macrocyclic immunomodulators
EP0642516B1 (en) * 1991-09-05 2002-06-05 Abbott Laboratories Macrocyclic immunomodulators
CA2091194A1 (en) * 1992-04-08 1993-10-09 Richard D. Connell 2-oxo-ethyl derivatives as immunosuppressants
PE52896A1 (es) 1994-10-26 1996-12-12 Novartis Ag Composicion farmaceutica
DE19581804T1 (de) 1994-10-26 1998-01-22 Ciba Geigy Ag Pharmazeutische Zusammensetzungen
AR004480A1 (es) * 1995-04-06 1998-12-16 Amico Derin C D Compuestos de ascomicina que poseen actividad antiinflamatoria, pro cedimiento para prepararlos, uso de dichos compuestos para preparar agentesfarmaceuticos y composiciones farmaceuticas que los incluyen
PT2198858E (pt) 1998-03-26 2011-09-01 Astellas Pharma Inc Composição farmacêutica de libertação constante que contém um macrólido como o tacrolimus
CN1161117C (zh) * 1998-04-27 2004-08-11 藤泽药品工业株式会社 药物组合物
GB9826656D0 (en) 1998-12-03 1999-01-27 Novartis Ag Organic compounds
US7063857B1 (en) 1999-04-30 2006-06-20 Sucampo Ag Use of macrolide compounds for the treatment of dry eye
GB0008785D0 (en) 2000-04-10 2000-05-31 Novartis Ag Organic compounds
US10143682B2 (en) 2014-10-28 2018-12-04 Koushi Yamaguchi Medicine for improving state of pregnancy, and use thereof
WO2020032252A1 (ja) 2018-08-10 2020-02-13 晃史 山口 母体と胎児との関係における液性免疫関連疾患の治療薬
EP3900729A4 (en) 2018-12-18 2022-09-07 Koushi Yamaguchi MEANS OF IMPROVING INFERTILITY, REPEATED MISSORS AND PREGNANCY CONDITIONS

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
EP0346427B1 (en) * 1987-12-09 1995-03-29 FISONS plc Macrocyclic compounds
EP0402931A1 (en) * 1989-06-14 1990-12-19 Sandoz Ltd. Heteroatoms-containing tricyclic compounds
JPH05504944A (ja) * 1989-08-18 1993-07-29 藤沢薬品工業株式会社 巨大環式化合物
EP0427680B1 (en) * 1989-11-09 1995-08-23 Sandoz Ltd. Heteroatoms-containing tricyclic compounds

Also Published As

Publication number Publication date
CS201191A3 (en) 1992-02-19
JPH04230388A (ja) 1992-08-19
AU8010891A (en) 1992-01-02
EP0465426A1 (en) 1992-01-08
IE912297A1 (en) 1992-01-15
HU912107D0 (en) 1991-12-30
AU648806B2 (en) 1994-05-05
IL98691A0 (en) 1992-07-15
NZ238809A (en) 1994-03-25
CA2045989A1 (en) 1992-01-03
HUT58338A (en) 1992-02-28
FI913182A0 (fi) 1991-06-28
MY110418A (en) 1998-05-30
FI913182A7 (fi) 1992-01-03
FI913182L (fi) 1992-01-03

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Legal Events

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FF Patent granted
KB Patent renewed
HC Change of name of proprietor(s)
KB Patent renewed