IL93936A - History of 9-dioxo-21,9-epoxy - erythromycin, method of preparation History of 11-oxo and 11-hydroxy, and pharmaceutical preparations containing them - Google Patents
History of 9-dioxo-21,9-epoxy - erythromycin, method of preparation History of 11-oxo and 11-hydroxy, and pharmaceutical preparations containing themInfo
- Publication number
- IL93936A IL93936A IL9393690A IL9393690A IL93936A IL 93936 A IL93936 A IL 93936A IL 9393690 A IL9393690 A IL 9393690A IL 9393690 A IL9393690 A IL 9393690A IL 93936 A IL93936 A IL 93936A
- Authority
- IL
- Israel
- Prior art keywords
- deoxo
- epoxy
- amino
- mmol
- erythromycin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US32947389A | 1989-03-28 | 1989-03-28 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL93936A0 IL93936A0 (en) | 1990-12-23 |
IL93936A true IL93936A (en) | 1994-06-24 |
Family
ID=23285572
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL9393690A IL93936A (en) | 1989-03-28 | 1990-03-28 | History of 9-dioxo-21,9-epoxy - erythromycin, method of preparation History of 11-oxo and 11-hydroxy, and pharmaceutical preparations containing them |
Country Status (14)
Country | Link |
---|---|
US (1) | US5288709A (ja) |
EP (1) | EP0465581B1 (ja) |
JP (1) | JPH04504259A (ja) |
KR (1) | KR920701229A (ja) |
AT (1) | ATE128714T1 (ja) |
AU (1) | AU623764B2 (ja) |
CA (1) | CA2049359A1 (ja) |
DE (1) | DE69022845T2 (ja) |
DK (1) | DK0465581T3 (ja) |
ES (1) | ES2080140T3 (ja) |
GR (1) | GR1000519B (ja) |
IL (1) | IL93936A (ja) |
NZ (1) | NZ233117A (ja) |
WO (1) | WO1990011288A1 (ja) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0549040A1 (en) * | 1991-12-20 | 1993-06-30 | Merck & Co. Inc. | Methods of making 4" derivatives of 9-deoxo-8a-aza-8a-alkyl-8a-homoerythromycin A |
FR2713226B1 (fr) * | 1993-12-03 | 1996-01-05 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
ATE207919T1 (de) * | 1995-08-03 | 2001-11-15 | Dade Behring Inc | Chinidin-konjugate und ihre anwendung in immunoassays |
EP0895999A1 (en) | 1997-08-06 | 1999-02-10 | Pfizer Products Inc. | C-4" substituted macrolide antibiotics |
GB0127349D0 (en) | 2001-11-14 | 2002-01-02 | Glaxo Group Ltd | Macrolides |
CA2483220A1 (en) * | 2002-04-25 | 2003-11-06 | Abbott Laboratories | Oxolide antibacterials |
CN100363359C (zh) * | 2002-08-29 | 2008-01-23 | 菲塞股份有限公司 | 运动内酯化合物 |
GB0310984D0 (en) * | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
PL1628989T3 (pl) * | 2003-05-13 | 2007-05-31 | Glaxo Group Ltd | Nowe związki o 14- i 15- członowym pierścieniu |
GB0310980D0 (en) * | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
GB0310986D0 (en) * | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
CN107365338B (zh) * | 2016-08-12 | 2021-03-19 | 西安世纪盛康药业有限公司 | 一类红霉素a-6,9-9,12-螺缩酮衍生物及其制备方法和应用 |
CN114504585A (zh) * | 2020-11-16 | 2022-05-17 | 中国人民解放军海军军医大学 | 一种大环内酯类衍生物在制备减重降糖药物中的应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1451798A (en) * | 1973-08-02 | 1976-10-06 | Ici Ltd | Prostanoic acid derivatives |
US3963696A (en) * | 1975-02-21 | 1976-06-15 | Abbott Laboratories | 6,6A-AND 6,7-Anhydroerythromycin B and derivatives thereof |
EP0184921A3 (en) * | 1984-12-08 | 1986-10-29 | Beecham Group Plc | Erythromycin derivatives |
US5008249A (en) * | 1985-08-31 | 1991-04-16 | Kitasato Kenkyusho | Therapeutic method of stimulating digestive tract contractile motion in mammals |
SE519436C2 (sv) * | 2001-04-09 | 2003-02-25 | Anoto Ab | Penna med på pennan löstagbart anordnade medel för byte av i pennan anordnat bläckstift, samt förfarande för stiftbyte |
-
1990
- 1990-03-28 IL IL9393690A patent/IL93936A/en not_active IP Right Cessation
- 1990-03-28 ES ES90906030T patent/ES2080140T3/es not_active Expired - Lifetime
- 1990-03-28 AU AU54028/90A patent/AU623764B2/en not_active Ceased
- 1990-03-28 GR GR900100232A patent/GR1000519B/el unknown
- 1990-03-28 NZ NZ233117A patent/NZ233117A/en unknown
- 1990-03-28 CA CA002049359A patent/CA2049359A1/en not_active Abandoned
- 1990-03-28 DK DK90906030.3T patent/DK0465581T3/da active
- 1990-03-28 JP JP2505715A patent/JPH04504259A/ja active Pending
- 1990-03-28 DE DE69022845T patent/DE69022845T2/de not_active Expired - Fee Related
- 1990-03-28 WO PCT/US1990/001658 patent/WO1990011288A1/en active IP Right Grant
- 1990-03-28 EP EP90906030A patent/EP0465581B1/en not_active Expired - Lifetime
- 1990-03-28 US US07/743,424 patent/US5288709A/en not_active Expired - Fee Related
- 1990-03-28 KR KR1019910701206A patent/KR920701229A/ko not_active Application Discontinuation
- 1990-03-28 AT AT90906030T patent/ATE128714T1/de not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DE69022845T2 (de) | 1996-06-13 |
KR920701229A (ko) | 1992-08-11 |
ES2080140T3 (es) | 1996-02-01 |
CA2049359A1 (en) | 1990-09-29 |
EP0465581B1 (en) | 1995-10-04 |
DK0465581T3 (da) | 1996-02-12 |
NZ233117A (en) | 1991-05-28 |
EP0465581A4 (en) | 1992-05-13 |
DE69022845D1 (en) | 1995-11-09 |
EP0465581A1 (en) | 1992-01-15 |
JPH04504259A (ja) | 1992-07-30 |
WO1990011288A1 (en) | 1990-10-04 |
ATE128714T1 (de) | 1995-10-15 |
AU623764B2 (en) | 1992-05-21 |
IL93936A0 (en) | 1990-12-23 |
AU5402890A (en) | 1990-10-22 |
US5288709A (en) | 1994-02-22 |
GR900100232A (en) | 1990-07-31 |
GR1000519B (el) | 1992-08-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
KB | Patent renewed | ||
RH | Patent void |