IL87431A - 3-acyl-5,6-dihydro-4h-imidazo(1,5-a)(1,4)benzodiazepin-6-ones and related compounds,their preparation and pharmaceutical compositions comprising them - Google Patents

3-acyl-5,6-dihydro-4h-imidazo(1,5-a)(1,4)benzodiazepin-6-ones and related compounds,their preparation and pharmaceutical compositions comprising them

Info

Publication number
IL87431A
IL87431A IL87431A IL8743188A IL87431A IL 87431 A IL87431 A IL 87431A IL 87431 A IL87431 A IL 87431A IL 8743188 A IL8743188 A IL 8743188A IL 87431 A IL87431 A IL 87431A
Authority
IL
Israel
Prior art keywords
carbon atoms
alkyl
group
hydrogen
preparation
Prior art date
Application number
IL87431A
Other languages
English (en)
Other versions
IL87431A0 (en
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IL87431A0 publication Critical patent/IL87431A0/xx
Publication of IL87431A publication Critical patent/IL87431A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL87431A 1987-08-28 1988-08-12 3-acyl-5,6-dihydro-4h-imidazo(1,5-a)(1,4)benzodiazepin-6-ones and related compounds,their preparation and pharmaceutical compositions comprising them IL87431A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB878720414A GB8720414D0 (en) 1987-08-28 1987-08-28 Chemical compounds

Publications (2)

Publication Number Publication Date
IL87431A0 IL87431A0 (en) 1989-01-31
IL87431A true IL87431A (en) 1992-11-15

Family

ID=10623016

Family Applications (1)

Application Number Title Priority Date Filing Date
IL87431A IL87431A (en) 1987-08-28 1988-08-12 3-acyl-5,6-dihydro-4h-imidazo(1,5-a)(1,4)benzodiazepin-6-ones and related compounds,their preparation and pharmaceutical compositions comprising them

Country Status (20)

Country Link
US (1) US4868176A (ko)
EP (1) EP0305298B1 (ko)
JP (1) JPS6471880A (ko)
KR (1) KR890003765A (ko)
AT (1) ATE94878T1 (ko)
AU (1) AU608888B2 (ko)
CA (1) CA1310638C (ko)
DE (1) DE3884319T2 (ko)
DK (1) DK470888A (ko)
ES (1) ES2059551T3 (ko)
FI (1) FI87074C (ko)
GB (2) GB8720414D0 (ko)
HU (1) HU201764B (ko)
IL (1) IL87431A (ko)
MX (1) MX173421B (ko)
NO (1) NO168178C (ko)
NZ (1) NZ225955A (ko)
PT (1) PT88338B (ko)
RU (1) RU2041225C1 (ko)
ZA (1) ZA886209B (ko)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI880814A (fi) * 1987-03-10 1988-09-11 Hoffmann La Roche Imidazodiazepin-derivat.
GB8909700D0 (en) * 1989-04-27 1989-06-14 Roussel Lab Ltd Chemical compounds
GB8927928D0 (en) * 1989-12-11 1990-02-14 Roussel Lab Ltd Chemical compounds
GB9023155D0 (en) * 1990-10-24 1990-12-05 Roussel Lab Ltd Chemical compounds
RU2636785C1 (ru) * 2016-11-21 2017-12-01 федеральное государственное автономное образовательное учреждение высшего образования "Южный федеральный университет" Гидрогалогенид 1-(3,4-диметоксифенил)-2-(7,8-диметил-2,3,4,5-тетрагидро[1,3]диазепино[1,2-а]бензимидазол-11-ил)этанона, обладающий обезболивающей и анксиолитической активностью

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1143728A (en) * 1979-10-04 1983-03-29 Max Gerecke Imidazodiazepine derivatives
MC1528A1 (fr) * 1982-07-21 1984-04-13 Hoffmann La Roche Imidazobenzodiazepines
DK174086D0 (da) * 1986-04-16 1986-04-16 Ferrosan As Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme
YU136287A (en) * 1986-07-25 1990-06-30 Boehringer Kg Process for preparing new 1,4 benzodiazepines

Also Published As

Publication number Publication date
EP0305298A3 (en) 1990-07-11
DE3884319D1 (de) 1993-10-28
GB8820356D0 (en) 1988-09-28
AU2155388A (en) 1989-03-02
DK470888D0 (da) 1988-08-23
NO883522D0 (no) 1988-08-08
FI883965A0 (fi) 1988-08-26
GB2209165A (en) 1989-05-04
GB2209165B (en) 1991-08-14
NO168178C (no) 1992-01-22
ATE94878T1 (de) 1993-10-15
FI87074B (fi) 1992-08-14
HUT50474A (en) 1990-02-28
MX12857A (es) 1993-10-01
NZ225955A (en) 1990-08-28
KR890003765A (ko) 1989-04-17
HU201764B (en) 1990-12-28
PT88338A (pt) 1989-06-30
JPS6471880A (en) 1989-03-16
PT88338B (pt) 1995-05-04
EP0305298B1 (fr) 1993-09-22
FI883965A (fi) 1989-03-01
NO883522L (no) 1989-03-01
MX173421B (es) 1994-03-03
US4868176A (en) 1989-09-19
GB8720414D0 (en) 1987-10-07
NO168178B (no) 1991-10-14
CA1310638C (en) 1992-11-24
ES2059551T3 (es) 1994-11-16
EP0305298A2 (fr) 1989-03-01
FI87074C (fi) 1992-11-25
AU608888B2 (en) 1991-04-18
DE3884319T2 (de) 1994-02-17
RU2041225C1 (ru) 1995-08-09
IL87431A0 (en) 1989-01-31
ZA886209B (en) 1989-11-29
DK470888A (da) 1989-03-01

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Legal Events

Date Code Title Description
RH Patent void
MM9K Patent not in force due to non-payment of renewal fees