MX173421B - Imidazobenzodiazepinas y sus sales y procedimiento para su preparacion - Google Patents
Imidazobenzodiazepinas y sus sales y procedimiento para su preparacionInfo
- Publication number
- MX173421B MX173421B MX012857A MX1285788A MX173421B MX 173421 B MX173421 B MX 173421B MX 012857 A MX012857 A MX 012857A MX 1285788 A MX1285788 A MX 1285788A MX 173421 B MX173421 B MX 173421B
- Authority
- MX
- Mexico
- Prior art keywords
- carbon atoms
- alkyl
- group
- hydrogen
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Child & Adolescent Psychology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención se refiere a compuestos de imidazabenzodiazepinas y sus sales de fórmula 1 en donde R1 representa un grupo fenilo, un grupo cicloalquilo que contiene de 4 a 6 átomos de carbono o un grupo de fórmula (en la cual R4 representa un átomo de hidrógeno o un grupo alquilo que contiene de 1 a 5 átomos de carbono; R5 representa un átomo de hidrógeno o un grupo alquilo que contiene de 1 a 5 átomos de carbono; y R6 representa un átomode hidrógeno, un grupo alquilo que contiene de 1 a 5 átomos de carbono, un grupo fenilo, un átomo de alógeno, un grupo alcoxicarbonilo que contiene de 2 a 5 átomos de carbono, un grupo ciano, un grupo amino o un grupo mono-o di-alquilamido en el que los grupos alquilo contienen de 1 a 5 átomos de carbono); R2 y R3, que puede ser identicos o diferentes, representa cada uno un átomo de hidrógeno, un grupoalquilo que contiene de 1 a 5 átomos de carbono o un grupo de cicloalquilo que contiene de 3 a 5 átomos de carbono, o R2 y R3 representan junto un grupo alquileno que contiene de 3 a 5 átomos de carbono; y X e v, que pueden ser identicos o diferentes, representa cada uno un átomo de hidrógeno, un átomo de halógeno, un grupo nitro, azido, nitrilo o trifluorometilo un grupo alquilo o alcoxi que contiene de 1 a 3 átomos de carbono y sus sales de adición de ácido.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB878720414A GB8720414D0 (en) | 1987-08-28 | 1987-08-28 | Chemical compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX12857A MX12857A (es) | 1993-10-01 |
| MX173421B true MX173421B (es) | 1994-03-03 |
Family
ID=10623016
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX012857A MX173421B (es) | 1987-08-28 | 1988-08-29 | Imidazobenzodiazepinas y sus sales y procedimiento para su preparacion |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US4868176A (es) |
| EP (1) | EP0305298B1 (es) |
| JP (1) | JPS6471880A (es) |
| KR (1) | KR890003765A (es) |
| AT (1) | ATE94878T1 (es) |
| AU (1) | AU608888B2 (es) |
| CA (1) | CA1310638C (es) |
| DE (1) | DE3884319T2 (es) |
| DK (1) | DK470888A (es) |
| ES (1) | ES2059551T3 (es) |
| FI (1) | FI87074C (es) |
| GB (2) | GB8720414D0 (es) |
| HU (1) | HU201764B (es) |
| IL (1) | IL87431A (es) |
| MX (1) | MX173421B (es) |
| NO (1) | NO168178C (es) |
| NZ (1) | NZ225955A (es) |
| PT (1) | PT88338B (es) |
| RU (1) | RU2041225C1 (es) |
| ZA (1) | ZA886209B (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI880814A (fi) * | 1987-03-10 | 1988-09-11 | Hoffmann La Roche | Imidazodiazepin-derivat. |
| GB8909700D0 (en) * | 1989-04-27 | 1989-06-14 | Roussel Lab Ltd | Chemical compounds |
| GB8927928D0 (en) * | 1989-12-11 | 1990-02-14 | Roussel Lab Ltd | Chemical compounds |
| GB9023155D0 (en) * | 1990-10-24 | 1990-12-05 | Roussel Lab Ltd | Chemical compounds |
| RU2636785C1 (ru) * | 2016-11-21 | 2017-12-01 | федеральное государственное автономное образовательное учреждение высшего образования "Южный федеральный университет" | Гидрогалогенид 1-(3,4-диметоксифенил)-2-(7,8-диметил-2,3,4,5-тетрагидро[1,3]диазепино[1,2-а]бензимидазол-11-ил)этанона, обладающий обезболивающей и анксиолитической активностью |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1143728A (en) * | 1979-10-04 | 1983-03-29 | Max Gerecke | Imidazodiazepine derivatives |
| MC1528A1 (fr) * | 1982-07-21 | 1984-04-13 | Hoffmann La Roche | Imidazobenzodiazepines |
| DK174086D0 (da) * | 1986-04-16 | 1986-04-16 | Ferrosan As | Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme |
| YU136287A (en) * | 1986-07-25 | 1990-06-30 | Boehringer Kg | Process for preparing new 1,4 benzodiazepines |
-
1987
- 1987-08-28 GB GB878720414A patent/GB8720414D0/en active Pending
-
1988
- 1988-08-08 NO NO883522A patent/NO168178C/no unknown
- 1988-08-12 IL IL87431A patent/IL87431A/xx not_active IP Right Cessation
- 1988-08-22 ZA ZA886209A patent/ZA886209B/xx unknown
- 1988-08-23 DK DK470888A patent/DK470888A/da not_active Application Discontinuation
- 1988-08-24 JP JP63208496A patent/JPS6471880A/ja active Pending
- 1988-08-25 PT PT88338A patent/PT88338B/pt not_active IP Right Cessation
- 1988-08-26 FI FI883965A patent/FI87074C/fi not_active IP Right Cessation
- 1988-08-26 DE DE88402166T patent/DE3884319T2/de not_active Expired - Fee Related
- 1988-08-26 KR KR1019880010852A patent/KR890003765A/ko not_active Application Discontinuation
- 1988-08-26 NZ NZ225955A patent/NZ225955A/xx unknown
- 1988-08-26 AU AU21553/88A patent/AU608888B2/en not_active Ceased
- 1988-08-26 AT AT88402166T patent/ATE94878T1/de not_active IP Right Cessation
- 1988-08-26 US US07/237,508 patent/US4868176A/en not_active Expired - Fee Related
- 1988-08-26 HU HU884466A patent/HU201764B/hu not_active IP Right Cessation
- 1988-08-26 EP EP88402166A patent/EP0305298B1/fr not_active Expired - Lifetime
- 1988-08-26 GB GB8820356A patent/GB2209165B/en not_active Expired - Lifetime
- 1988-08-26 ES ES88402166T patent/ES2059551T3/es not_active Expired - Lifetime
- 1988-08-26 CA CA000575843A patent/CA1310638C/en not_active Expired - Fee Related
- 1988-08-29 MX MX012857A patent/MX173421B/es unknown
-
1992
- 1992-01-16 RU SU925010559A patent/RU2041225C1/ru active
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