IL78250A - 1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL78250A
IL78250A IL78250A IL7825086A IL78250A IL 78250 A IL78250 A IL 78250A IL 78250 A IL78250 A IL 78250A IL 7825086 A IL7825086 A IL 7825086A IL 78250 A IL78250 A IL 78250A
Authority
IL
Israel
Prior art keywords
halo
alkyl
benzisothiazol
benzisoxazol
derivatives
Prior art date
Application number
IL78250A
Other languages
English (en)
Other versions
IL78250A0 (en
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24880589&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL78250(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of IL78250A0 publication Critical patent/IL78250A0/xx
Publication of IL78250A publication Critical patent/IL78250A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
IL78250A 1985-03-27 1986-03-25 1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them IL78250A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US71706785A 1985-03-27 1985-03-27

Publications (2)

Publication Number Publication Date
IL78250A0 IL78250A0 (en) 1986-07-31
IL78250A true IL78250A (en) 1991-05-12

Family

ID=24880589

Family Applications (1)

Application Number Title Priority Date Filing Date
IL78250A IL78250A (en) 1985-03-27 1986-03-25 1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them

Country Status (13)

Country Link
KR (1) KR910000165B1 (xx)
AT (1) ATE79379T1 (xx)
DE (1) DE3686341T2 (xx)
ES (1) ES8705881A1 (xx)
FI (1) FI81800C (xx)
GR (1) GR860800B (xx)
HU (1) HU195793B (xx)
IL (1) IL78250A (xx)
NO (2) NO162765C (xx)
NZ (1) NZ215462A (xx)
PH (1) PH24016A (xx)
PT (1) PT82254B (xx)
ZA (1) ZA862279B (xx)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2050069B1 (es) * 1992-07-10 1994-12-16 Vita Invest Sa Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-il)piperidino)etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido(1,2-a) pirimidin-4-ona.
ES2085234B1 (es) * 1994-02-24 1997-01-16 Vita Invest Sa Agente activo sobre el sistema nervioso central, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.
HUP0402163A2 (en) * 2004-10-25 2006-05-29 Richter Gedeon Vegyeszet Process for the preparation of risperidone

Also Published As

Publication number Publication date
FI861328A0 (fi) 1986-03-26
PH24016A (en) 1990-02-09
HU195793B (en) 1988-07-28
NO162765B (no) 1989-11-06
HUT42461A (en) 1987-07-28
KR910000165B1 (ko) 1991-01-21
FI861328A (fi) 1986-09-28
ES553419A0 (es) 1987-05-16
KR860007247A (ko) 1986-10-10
DE3686341D1 (de) 1992-09-17
NO1994021I1 (no) 1994-11-03
PT82254B (pt) 1988-04-21
PT82254A (en) 1986-04-01
DE3686341T2 (de) 1993-01-14
ZA862279B (en) 1987-11-25
FI81800C (fi) 1990-12-10
GR860800B (en) 1986-07-21
NZ215462A (en) 1988-09-29
IL78250A0 (en) 1986-07-31
FI81800B (fi) 1990-08-31
NO162765C (no) 1990-02-14
ATE79379T1 (de) 1992-08-15
NO861230L (no) 1986-09-29
ES8705881A1 (es) 1987-05-16

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