IL40060A - Compositions for controlling plant pathogenic organisms containing s-triazole(4,3-alpha)quinoline derivatives and cetain 4,5-dohydro-s-triazolo(4,3-alpha)quinolines rtain 4,5-dihydro-s-triazolo(4,3-alpha)quinolines - Google Patents

Compositions for controlling plant pathogenic organisms containing s-triazole(4,3-alpha)quinoline derivatives and cetain 4,5-dohydro-s-triazolo(4,3-alpha)quinolines rtain 4,5-dihydro-s-triazolo(4,3-alpha)quinolines

Info

Publication number
IL40060A
IL40060A IL40060A IL4006072A IL40060A IL 40060 A IL40060 A IL 40060A IL 40060 A IL40060 A IL 40060A IL 4006072 A IL4006072 A IL 4006072A IL 40060 A IL40060 A IL 40060A
Authority
IL
Israel
Prior art keywords
triazolo
hydrogen
formula
dihydro
alpha
Prior art date
Application number
IL40060A
Other languages
Hebrew (he)
Other versions
IL40060A0 (en
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL40060A0 publication Critical patent/IL40060A0/en
Publication of IL40060A publication Critical patent/IL40060A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

1374369 s-Triazoloquinoline derivatives ELI LILLY & CO 15 Aug 1972 [16 Aug 1971] 37989/72 Heading C2C Novel s-triazoloquinoline derivatives having the formula and known s-triazoloquinoline derivatives of the formula wherein R is hydrogen, halogen, (C 1 -C 3 ) alkyl, (C 1 -C 3 ) alkoxy, formyl, cyano, -CF 3 or substituted methyl radical of the formula -CH 2 Y wherein Y is amino, (C 1 -C 3 ) alkylamino, cyano, hydroxy, halogen or (C 1 -C 3 ) alkoxy; R<SP>2</SP> is hydrogen, (C 1 -C 5 ) alkyl, vinyl, (C 3 -C 6 ) cycloalkyl, hydroxy, (C 1 -C 3 ) alkoxy, mercapto, (C 1 -C 3 ) alkylthio, benzylthio, halogen, amino, (C 1 -C 3 ) alkylamino, di-(C 1 -C 3 ) alkylamino, carbamoyl, thiocyanato, acetamido, -CF 3 , a radical of the formula -COOR<SP>4</SP> wherein R<SP>4</SP> is Na, K or (C 1 -C 3 ) alkyl, or a substituted methyl radical of the formula -CH 2 Y<SP>1</SP> wherein Y<SP>1</SP> is amino, (C 1 -C 3 ) alkylamino, cyano, halogen, (C 1 -C 3 ) alkoxy, (C 1 -C 2 ) alkoxymethyl or halomethyl; and R<SP>3</SP> is hydrogen, (C 1 -C 3 ) alkyl, or halogen, provided that (i) not more than two R<SP>3</SP> groups represent halogen or alkyl, (ii) in the second formula, not more than three of the groups represented by R<SP>1</SP> and R<SP>2</SP> are moieties other than hydrogen, (iii) in the first formula, not more than three of R<SP>1</SP>, R<SP>2</SP> and R<SP>3</SP> represent a moiety other than hydrogen, and (iv) in both formulµ, at least one of R<SP>2</SP> and R<SP>1</SP> at the 9th position represents hydrogen; as well as the phytologically-acceptable mineral acid addition salts thereof, are useful as controllants for plant-pathogenic organisms. [GB1374369A]

Claims (6)

1. CLAIMS 1. Compositions for controlling plant- pathogenic organisms which comprise,-- as the active agent a¾ least one compound selected from the s_-trlazolo ( ,3-a)quinoline compounds- of the formulae 20 and the phytologlcally-acceptable mineral acid addition · salts thereof, wherein each R1 independently represents hydrogen, halo, loweralkyl of C^-C-j, loweralkoxy of C-^-C^, *8.72 X R2 represents hydrogen, loweralkyl of C-^-C^, vinyl, cyclo-. alkyl of C^-Cg, hydroxy, loweralkoxy of C-^-C-,, mercapto, loweralkylthio of O^-C^, benzylthio, halo, amino (loweralkyl of amino, carbamoyl, acetamido, trifluoromethyl, a radical of the formula wherein R4 represents sodium, potassium, or loweralkyl of C^-C-j, or a radical of the .72 formula -CHp-Y' wherein Y' represents loweralkoxy of C ' of halo, subject to the limitation that no more than two groups represent halo or loweralk l as defined the foregoing definitions being subject to the further limitations (1) that in Formula X not more than three of B1 and R2 are other than hydrogen; (2) that in Formula IX 1 2 3 not more than three of R , R and R^ are other than hydrogen; and (3) that in both Formulae X and II at least one of the 2 1 R and the R substituents at the 9-position represents hydrogen.
2. , A composition according to Claim 1 which contains a surface active dispersing agent and an inert finely divided solid. 3· The composition of Claim 2 wherein the active agent is l^methyl-s.-triazolo(4,3-a)qulnoline. 4. The composition of Claim 2 wherein the active agent is l-chloro-s-triazolo(4,3-a)qulnoline. 5. The composition of Claim 2 wherein the active agent is 9-chloro-s-triazolo(4,3-a)qulnoline. 6. The composition of Claim 2 wherein the active agent is 9-methyl-s-trlazolo(4,3-a)qulnoline. 7. The compositon of Claim 2 wherein the active agent is 4» 5-dihydro-s-triazolo(4,3-a)qulnoline. 8. The composition of Claim 2 wherein the active agent is 4, 5-dihydro-l-methyl^s-triazolo(4»3-a)qulnoline. 40060/ 4 10. The composition of Claim 2 wherein the active agent is 4 , 5-dihydro-9-methyl-s-tria olo( , 3-a)quinoline . 11. s-Triazolo(4, 3-a)quinoline compounds of the formula and. the phytologlcall -acceptable mineral acid addition salts thereof, wherein R1 is hydrogen, halogen, or lower- alkyl, and R2 is hydrogen, lower alkyl or trifluoromethyl ; provided that (l) not more than three of R1 and R2 are othe than hydrogen, and (2) that at least one of R2 and the substituent R1 at the 9-position represent hydrogen. 12. 4, 5-Dihydro-s-triazolo(4,3-a)quinoline. 1
3. 4, 5-Dihydro-l-methyl-s-triazolo ;(4,3-a)quinoline". 1
4. 9-Chloro-4 , 5-dihydro-s-triazolo (4 , 3-a)quinoline . 1
5. 4, 5-Dihydro-9-methyl-s-triazol6'( , quinoline. 1
6. A process for controlling plant-'pathc-genic organisms which comprises applying to a locus of the organism an effective amount of a composition according tocany of Claims 1 to, 9L P md
IL40060A 1971-08-16 1972-08-07 Compositions for controlling plant pathogenic organisms containing s-triazole(4,3-alpha)quinoline derivatives and cetain 4,5-dohydro-s-triazolo(4,3-alpha)quinolines rtain 4,5-dihydro-s-triazolo(4,3-alpha)quinolines IL40060A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17231771A 1971-08-16 1971-08-16

Publications (2)

Publication Number Publication Date
IL40060A0 IL40060A0 (en) 1972-10-29
IL40060A true IL40060A (en) 1976-08-31

Family

ID=22627199

Family Applications (1)

Application Number Title Priority Date Filing Date
IL40060A IL40060A (en) 1971-08-16 1972-08-07 Compositions for controlling plant pathogenic organisms containing s-triazole(4,3-alpha)quinoline derivatives and cetain 4,5-dohydro-s-triazolo(4,3-alpha)quinolines rtain 4,5-dihydro-s-triazolo(4,3-alpha)quinolines

Country Status (31)

Country Link
JP (1) JPS5760321B2 (en)
KR (1) KR790000421B1 (en)
AR (2) AR195289A1 (en)
AT (1) AT324767B (en)
AU (1) AU461057B2 (en)
BE (1) BE787536A (en)
BG (3) BG24409A3 (en)
CA (1) CA997766A (en)
CH (2) CH564016A5 (en)
CS (1) CS190371B2 (en)
DD (2) DD107462A5 (en)
DE (1) DE2239892A1 (en)
DK (1) DK139832B (en)
EG (1) EG10668A (en)
ES (1) ES405899A1 (en)
FR (1) FR2149467B1 (en)
GB (1) GB1374369A (en)
GT (1) GT197225694A (en)
HU (1) HU167272B (en)
IE (1) IE36916B1 (en)
IL (1) IL40060A (en)
IT (1) IT962096B (en)
MY (1) MY7800200A (en)
NL (1) NL177173C (en)
PH (1) PH10204A (en)
PL (1) PL94442B1 (en)
RO (2) RO79165A (en)
SE (2) SE405313B (en)
SU (1) SU554815A3 (en)
YU (1) YU36937B (en)
ZA (1) ZA725365B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1102524B (en) * 1977-03-29 1985-10-07 Capsugel Ag CONTAINMENT CAPSULE FOR VISCOUS MATERIALS IN PARTICULAR A LIQUID PHARMACEUTICAL PREPARATION AND PROCEDURE FOR ITS PRODUCTION
JPS61186648U (en) * 1984-12-29 1986-11-20
AT393764B (en) * 1986-09-02 1991-12-10 System Elektrotechnik Gotthold JUMPER CABLES
JPS63166228U (en) * 1987-04-21 1988-10-28
JP2007506788A (en) * 2003-09-26 2007-03-22 ライジェル ファーマシューティカルズ, インコーポレイテッド HCV infection inhibitors and uses thereof
WO2005121138A2 (en) * 2004-06-03 2005-12-22 Rigel Pharmaceuticals, Inc. Heterotricyclic compounds for use as hcv inhibitors
WO2007087250A2 (en) * 2006-01-23 2007-08-02 Amira Pharmaceuticals, Inc. Tricyclic inhibitors of 5-lipoxygenase

Also Published As

Publication number Publication date
RO63409A (en) 1978-09-15
IT962096B (en) 1973-12-20
PH10204A (en) 1976-09-27
KR790000421B1 (en) 1979-05-14
CH552942A (en) 1974-08-30
ZA725365B (en) 1974-03-27
YU36937B (en) 1984-08-31
ES405899A1 (en) 1975-08-01
CH564016A5 (en) 1975-07-15
DD104176A5 (en) 1974-03-05
AT324767B (en) 1975-09-25
CA997766A (en) 1976-09-28
BG20354A3 (en) 1975-11-05
AU461057B2 (en) 1975-05-15
DK139832B (en) 1979-04-30
SE7507384L (en) 1975-06-27
IE36916B1 (en) 1977-03-30
EG10668A (en) 1976-03-31
AU4539772A (en) 1974-02-14
BG19623A1 (en) 1975-10-10
DE2239892A1 (en) 1973-03-01
PL94442B1 (en) 1977-08-31
FR2149467A1 (en) 1973-03-30
AR195289A1 (en) 1973-09-28
CS190371B2 (en) 1979-05-31
HU167272B (en) 1975-09-27
SU554815A3 (en) 1977-04-15
DK139832C (en) 1979-10-08
YU204372A (en) 1982-06-18
BE787536A (en) 1973-02-14
NL177173C (en) 1985-08-16
NL7210957A (en) 1973-02-20
RO79165A (en) 1982-06-25
IE36916L (en) 1973-02-16
GT197225694A (en) 1974-02-05
JPS4828642A (en) 1973-04-16
BG24409A3 (en) 1978-02-10
FR2149467B1 (en) 1976-10-29
NL177173B (en) 1985-03-18
DD107462A5 (en) 1974-08-05
SE422059B (en) 1982-02-15
JPS5760321B2 (en) 1982-12-18
SE405313B (en) 1978-12-04
MY7800200A (en) 1978-12-31
AR215825A1 (en) 1979-11-15
GB1374369A (en) 1974-11-20
IL40060A0 (en) 1972-10-29

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