ES405899A1 - Triazoloquinoline derivatives and their use as agents for the control of plant-pathogenic organisms - Google Patents

Triazoloquinoline derivatives and their use as agents for the control of plant-pathogenic organisms

Info

Publication number
ES405899A1
ES405899A1 ES405899A ES405899A ES405899A1 ES 405899 A1 ES405899 A1 ES 405899A1 ES 405899 A ES405899 A ES 405899A ES 405899 A ES405899 A ES 405899A ES 405899 A1 ES405899 A1 ES 405899A1
Authority
ES
Spain
Prior art keywords
formula
lower alkyl
halogen
amino
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES405899A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES405899A1 publication Critical patent/ES405899A1/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Abstract

A procedure for the preparation of new s-triazolo (4,3-a) quinoline compounds of the formula **(See formula)** and its addition salts with phytologically acceptable mineral acids, where each group independently represents hydrogen, halogen, C1-C3 lower alkyl, C1-C3 lower alkoxy, formyl, cyano, trifluoromethyl or substituted methyl of the formula -CH2Y, where Y represents amino, C1-C3 lower alkyl), cyano, hydroxy, halogen or C1-C3 lower alkoxy; R2 represents hydrogen, C1C5 lower alkyl, vinyl, C3-C6 cycloalkyl, hydroxy, C1-C3 lower alkoxy, mercapto, C1-C3 lower alkylthio, benzylthio, halogen, amino, C1-C3 lower alkyl, dialkyl (lower C1-C3) amino, carbamoyl, thiocyanate, acetamido, trifluoromethyl, a radical of formula (see formula), where it represents sodium, potassium, or C1-C3 lower alkyl or a radical of formula -CH2Y', where Y' represents amino, C1-C3 lower alkyl, cyano, halogen, C1-C3 lower alkoxy, C1-C2 lower alkoxy methyl or halomethyl; and each group independently represents hydrogen, C1-C3 lower alkyl, or halogen, subject to the limitation that no more than two R3 groups represent halogen or lower alkyl as defined; the above definitions being subject to the following additional limitations: (1) no more than three of the groups r1, R2 and R3 represent a radical other than hydrogen and (2) at least one of the groups R2 and the substituent R1 in the Position 9 represent hydrogen, characterized by the following stages: 1) condense 3,4-dihydro-2-hydrazinoquinoline: **(See formula)** with an acid of formula R2-COOH or a suitable ester thereof; 2) react 3,4-dihydro-2-hydrazinoquinoline of formula: **(See formula)** with a formula orthoester R2-C (O-alkyl) 3 where R2 represents hydrogen, lower alkyl or cycloalkyl; 3) when R2 represents -OH or -SH, the same precursor 2-hydrazino compounds described above as starting materials are reacted with a phenyl isocyanate or a phenyl isothiocyanate; and 4) react 3,4-dihydro-2-hydrazinoquinoline with cyanogen bromide, when R2 is amino. (Machine-translation by Google Translate, not legally binding)
ES405899A 1971-08-16 1971-08-16 Triazoloquinoline derivatives and their use as agents for the control of plant-pathogenic organisms Expired ES405899A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17231771A 1971-08-16 1971-08-16

Publications (1)

Publication Number Publication Date
ES405899A1 true ES405899A1 (en) 1975-08-01

Family

ID=22627199

Family Applications (1)

Application Number Title Priority Date Filing Date
ES405899A Expired ES405899A1 (en) 1971-08-16 1971-08-16 Triazoloquinoline derivatives and their use as agents for the control of plant-pathogenic organisms

Country Status (31)

Country Link
JP (1) JPS5760321B2 (en)
KR (1) KR790000421B1 (en)
AR (2) AR195289A1 (en)
AT (1) AT324767B (en)
AU (1) AU461057B2 (en)
BE (1) BE787536A (en)
BG (3) BG19623A1 (en)
CA (1) CA997766A (en)
CH (2) CH564016A5 (en)
CS (1) CS190371B2 (en)
DD (2) DD107462A5 (en)
DE (1) DE2239892A1 (en)
DK (1) DK139832B (en)
EG (1) EG10668A (en)
ES (1) ES405899A1 (en)
FR (1) FR2149467B1 (en)
GB (1) GB1374369A (en)
GT (1) GT197225694A (en)
HU (1) HU167272B (en)
IE (1) IE36916B1 (en)
IL (1) IL40060A (en)
IT (1) IT962096B (en)
MY (1) MY7800200A (en)
NL (1) NL177173C (en)
PH (1) PH10204A (en)
PL (1) PL94442B1 (en)
RO (2) RO63409A (en)
SE (2) SE405313B (en)
SU (1) SU554815A3 (en)
YU (1) YU36937B (en)
ZA (1) ZA725365B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2385389A1 (en) * 1977-03-29 1978-10-27 Capsugel Ag NOCKED CAPSULE FILLED WITH A VISCOUS MATERIAL SUCH AS, IN PARTICULAR, A LIQUID PHARMACEUTICAL PREPARATION
JPS61186648U (en) * 1984-12-29 1986-11-20
AT393764B (en) * 1986-09-02 1991-12-10 System Elektrotechnik Gotthold JUMPER CABLES
JPS63166228U (en) * 1987-04-21 1988-10-28
WO2005030774A1 (en) * 2003-09-26 2005-04-07 Rigel Pharmaceuticals, Inc. Hcv inhibitors and methods of using them
WO2005121138A2 (en) * 2004-06-03 2005-12-22 Rigel Pharmaceuticals, Inc. Heterotricyclic compounds for use as hcv inhibitors
EP1978966A4 (en) * 2006-01-23 2010-11-10 Amira Pharmaceuticals Inc Tricyclic inhibitors of 5-lipoxygenase

Also Published As

Publication number Publication date
YU36937B (en) 1984-08-31
SE7507384L (en) 1975-06-27
EG10668A (en) 1976-03-31
ZA725365B (en) 1974-03-27
DE2239892A1 (en) 1973-03-01
JPS4828642A (en) 1973-04-16
AR195289A1 (en) 1973-09-28
BG19623A1 (en) 1975-10-10
IE36916B1 (en) 1977-03-30
AU461057B2 (en) 1975-05-15
IT962096B (en) 1973-12-20
RO79165A (en) 1982-06-25
KR790000421B1 (en) 1979-05-14
GB1374369A (en) 1974-11-20
IL40060A0 (en) 1972-10-29
IL40060A (en) 1976-08-31
CH552942A (en) 1974-08-30
NL7210957A (en) 1973-02-20
DD107462A5 (en) 1974-08-05
GT197225694A (en) 1974-02-05
NL177173B (en) 1985-03-18
RO63409A (en) 1978-09-15
MY7800200A (en) 1978-12-31
BG20354A3 (en) 1975-11-05
BE787536A (en) 1973-02-14
YU204372A (en) 1982-06-18
SE405313B (en) 1978-12-04
PH10204A (en) 1976-09-27
NL177173C (en) 1985-08-16
AR215825A1 (en) 1979-11-15
PL94442B1 (en) 1977-08-31
CH564016A5 (en) 1975-07-15
CS190371B2 (en) 1979-05-31
AU4539772A (en) 1974-02-14
BG24409A3 (en) 1978-02-10
DK139832B (en) 1979-04-30
SU554815A3 (en) 1977-04-15
AT324767B (en) 1975-09-25
CA997766A (en) 1976-09-28
DD104176A5 (en) 1974-03-05
IE36916L (en) 1973-02-16
DK139832C (en) 1979-10-08
JPS5760321B2 (en) 1982-12-18
FR2149467B1 (en) 1976-10-29
HU167272B (en) 1975-09-27
FR2149467A1 (en) 1973-03-30
SE422059B (en) 1982-02-15

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