IL33582A - Basic aryloxyacetamides,their preparation and pharmaceutical compositions containing them - Google Patents

Basic aryloxyacetamides,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL33582A
IL33582A IL33582A IL3358269A IL33582A IL 33582 A IL33582 A IL 33582A IL 33582 A IL33582 A IL 33582A IL 3358269 A IL3358269 A IL 3358269A IL 33582 A IL33582 A IL 33582A
Authority
IL
Israel
Prior art keywords
compound
formula
halogen
preparation
compounds according
Prior art date
Application number
IL33582A
Other languages
English (en)
Original Assignee
Cerpha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cerpha filed Critical Cerpha
Publication of IL33582A publication Critical patent/IL33582A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL33582A 1968-12-26 1969-12-22 Basic aryloxyacetamides,their preparation and pharmaceutical compositions containing them IL33582A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR180720A FR8120M (de) 1968-12-26 1968-12-26

Publications (1)

Publication Number Publication Date
IL33582A true IL33582A (en) 1973-02-28

Family

ID=8659084

Family Applications (1)

Application Number Title Priority Date Filing Date
IL33582A IL33582A (en) 1968-12-26 1969-12-22 Basic aryloxyacetamides,their preparation and pharmaceutical compositions containing them

Country Status (15)

Country Link
US (1) US3818021A (de)
JP (1) JPS4837258B1 (de)
AT (1) AT293367B (de)
BE (1) BE743077A (de)
BR (1) BR6915166D0 (de)
CA (1) CA930738A (de)
CH (1) CH518267A (de)
DE (1) DE1964712C3 (de)
DK (1) DK127106B (de)
ES (1) ES374922A1 (de)
FR (1) FR8120M (de)
GB (1) GB1282600A (de)
IL (1) IL33582A (de)
NL (1) NL148591B (de)
SE (1) SE380009B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2623228C3 (de) * 1976-05-24 1981-09-10 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren N-Acyl-substituierte Benzamide, Verfahren zu ihrer Herstellung und Arzneimittel, enthaltend solche Benzamide
US4073940A (en) * 1976-10-28 1978-02-14 Centre Europeen De Recherches Pharmacologiques C.E.R.P.H.A. Method for treating cardiac arhythmia by administration of basic aryloxyacetamide
FR2618149B1 (fr) * 1987-07-16 1989-09-22 Synthelabo Derives de n-aminoalkyl n-phenyl arylamides, leur preparation et leur application en therapeutique
MXPA05001958A (es) 2002-08-19 2005-04-28 Pfizer Prod Inc Terapia de combinacion para enfermedades hiperproliferativas.
US20050037063A1 (en) * 2003-07-21 2005-02-17 Bolton Anthony E. Combined therapies
US20060063803A1 (en) * 2004-09-23 2006-03-23 Pfizer Inc 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
CN101663262B (zh) 2006-12-01 2014-03-26 百时美施贵宝公司 用于治疗动脉粥样硬化和心血管疾病的作为cetp抑制剂的n-(3-苄基)-2,2-(二苯基)-丙-1胺衍生物
WO2012112958A2 (en) * 2011-02-19 2012-08-23 The Broad Institute, Inc High-throughput assays to probe leukemia within the stromal niche
CN105143203A (zh) 2013-04-17 2015-12-09 辉瑞大药厂 用于治疗心血管疾病的n-哌啶-3-基苯甲酰胺衍生物
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
CN113574055B (zh) 2019-01-18 2024-07-23 阿斯利康(瑞典)有限公司 Pcsk9抑制剂及其使用方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2428978A (en) * 1943-07-30 1947-10-14 Geigy Ag J R Basic derivatives of alpha-substituted aryloxy acetic acids and a process for their manufacture
US2437545A (en) * 1944-06-02 1948-03-09 Geigy Ag J R Basic amides of 1-aryl-cycloalkyl-1-carboxylic acids
US2715645A (en) * 1952-07-16 1955-08-16 Searle & Co N-aryl and n-aralkyl derivatives of n-dialkylaminoalkyl-aryloxyalkanoamides and methods for their production
US2948954A (en) * 1956-03-08 1960-08-16 Alexander P Ramsa Small sized helixes and method of their fabrication
FR1455055A (fr) * 1965-02-02 1966-04-01 Centre Nat Rech Scient Procédé de préparation d'amides d'acides carboxyliques

Also Published As

Publication number Publication date
CH518267A (fr) 1972-01-31
NL148591B (nl) 1976-02-16
DK127106B (da) 1973-09-24
AT293367B (de) 1971-10-11
DE1964712A1 (de) 1970-07-02
FR8120M (de) 1970-08-03
NL6919276A (de) 1970-06-30
SE380009B (de) 1975-10-27
BR6915166D0 (pt) 1973-02-13
DE1964712B2 (de) 1974-05-30
BE743077A (de) 1970-05-14
DE1964712C3 (de) 1975-02-27
ES374922A1 (es) 1972-02-16
CA930738A (en) 1973-07-24
US3818021A (en) 1974-06-18
GB1282600A (en) 1972-07-19
JPS4837258B1 (de) 1973-11-09

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