IL304974A - תכשירים של תצורה iv טהורה בעיקר של n–((r)–3,2–דיהידרוקסיפרופוקסי)–4,3–דיפלואורו–2–(2–פלואורו–4–יודופנילאמינו)–בנזאמיד ושימושים שלהם - Google Patents
תכשירים של תצורה iv טהורה בעיקר של n–((r)–3,2–דיהידרוקסיפרופוקסי)–4,3–דיפלואורו–2–(2–פלואורו–4–יודופנילאמינו)–בנזאמיד ושימושים שלהםInfo
- Publication number
- IL304974A IL304974A IL304974A IL30497423A IL304974A IL 304974 A IL304974 A IL 304974A IL 304974 A IL304974 A IL 304974A IL 30497423 A IL30497423 A IL 30497423A IL 304974 A IL304974 A IL 304974A
- Authority
- IL
- Israel
- Prior art keywords
- fluoro
- dihydroxypropoxy
- difluoro
- benzamide
- iodo
- Prior art date
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Inorganic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US2021/018378 WO2022177556A1 (en) | 2021-02-17 | 2021-02-17 | Compositions of essentially pure form iv of n-((r)-2,3- dihydroxypropoxy)-3,4-difluoro-2- (2-fluoro-4-iodophenylamino)- benzamide and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL304974A true IL304974A (he) | 2023-10-01 |
Family
ID=74860567
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL304974A IL304974A (he) | 2021-02-17 | 2021-02-17 | תכשירים של תצורה iv טהורה בעיקר של n–((r)–3,2–דיהידרוקסיפרופוקסי)–4,3–דיפלואורו–2–(2–פלואורו–4–יודופנילאמינו)–בנזאמיד ושימושים שלהם |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP4294789A1 (he) |
| JP (1) | JP2024507822A (he) |
| KR (1) | KR20230148177A (he) |
| CN (1) | CN117500781A (he) |
| AR (1) | AR124907A1 (he) |
| AU (1) | AU2021428932A1 (he) |
| CA (1) | CA3211395A1 (he) |
| IL (1) | IL304974A (he) |
| TW (1) | TW202245746A (he) |
| WO (1) | WO2022177556A1 (he) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2023223205A1 (en) | 2022-05-17 | 2023-11-23 | Teva Pharmaceuticals International Gmbh | Solid state forms of mirdametinib and process for preparation thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1301472T3 (da) | 2000-07-19 | 2014-04-07 | Warner Lambert Co | Oxygenerede estere af 4-iod-phenylamino-benzhydroxamsyrer |
| NZ546011A (en) | 2003-10-21 | 2009-09-25 | Warner Lambert Co | Polymorphic form of N-[(R)-2,3-dihydroxy-propoxy]-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-benzamide |
| WO2006134469A1 (en) | 2005-06-14 | 2006-12-21 | Warner-Lambert Company Llc | Methods of preparing mek inhibitor |
-
2021
- 2021-02-17 AU AU2021428932A patent/AU2021428932A1/en active Pending
- 2021-02-17 WO PCT/US2021/018378 patent/WO2022177556A1/en active Application Filing
- 2021-02-17 JP JP2023549999A patent/JP2024507822A/ja active Pending
- 2021-02-17 CN CN202180095226.2A patent/CN117500781A/zh active Pending
- 2021-02-17 KR KR1020237030268A patent/KR20230148177A/ko unknown
- 2021-02-17 IL IL304974A patent/IL304974A/he unknown
- 2021-02-17 CA CA3211395A patent/CA3211395A1/en active Pending
- 2021-02-17 EP EP21710827.3A patent/EP4294789A1/en active Pending
-
2022
- 2022-02-17 AR ARP220100332A patent/AR124907A1/es unknown
- 2022-02-17 TW TW111105793A patent/TW202245746A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW202245746A (zh) | 2022-12-01 |
| WO2022177556A1 (en) | 2022-08-25 |
| AR124907A1 (es) | 2023-05-17 |
| EP4294789A1 (en) | 2023-12-27 |
| KR20230148177A (ko) | 2023-10-24 |
| JP2024507822A (ja) | 2024-02-21 |
| CN117500781A (zh) | 2024-02-02 |
| CA3211395A1 (en) | 2022-08-25 |
| AU2021428932A1 (en) | 2023-09-21 |
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