IL277496B2 - Melanocortin receptor-specific peptide formulations and methods for specific administration to the gastrointestinal tract - Google Patents
Melanocortin receptor-specific peptide formulations and methods for specific administration to the gastrointestinal tractInfo
- Publication number
- IL277496B2 IL277496B2 IL277496A IL27749620A IL277496B2 IL 277496 B2 IL277496 B2 IL 277496B2 IL 277496 A IL277496 A IL 277496A IL 27749620 A IL27749620 A IL 27749620A IL 277496 B2 IL277496 B2 IL 277496B2
- Authority
- IL
- Israel
- Prior art keywords
- eudragit
- average
- pharmaceutically acceptable
- peptide
- acceptable salt
- Prior art date
Links
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- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/64—Cyclic peptides containing only normal peptide links
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Zoology (AREA)
- Endocrinology (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862647000P | 2018-03-23 | 2018-03-23 | |
| PCT/US2019/023575 WO2019183472A1 (en) | 2018-03-23 | 2019-03-22 | Melanocortin receptor-specific peptide formulations and methods for gastrointestinal tract-specific delivery |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| IL277496A IL277496A (en) | 2020-11-30 |
| IL277496B1 IL277496B1 (en) | 2024-09-01 |
| IL277496B2 true IL277496B2 (en) | 2025-01-01 |
Family
ID=67988087
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL277496A IL277496B2 (en) | 2018-03-23 | 2019-03-22 | Melanocortin receptor-specific peptide formulations and methods for specific administration to the gastrointestinal tract |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20220088146A1 (https=) |
| EP (1) | EP3768245A4 (https=) |
| JP (1) | JP2021523931A (https=) |
| KR (1) | KR102743821B1 (https=) |
| CN (1) | CN112188888A (https=) |
| AU (2) | AU2019239300A1 (https=) |
| BR (1) | BR112020019128A2 (https=) |
| CA (1) | CA3095036A1 (https=) |
| EA (1) | EA202092275A1 (https=) |
| IL (1) | IL277496B2 (https=) |
| MX (1) | MX2020009900A (https=) |
| PH (1) | PH12020551596A1 (https=) |
| WO (1) | WO2019183472A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20220137043A (ko) * | 2020-02-03 | 2022-10-11 | 팔라틴 테크놀로지스 인코포레이티드 | 디아민-연결 수용체-특이적 고리형 펩티드 |
| JPWO2024143501A1 (https=) * | 2022-12-28 | 2024-07-04 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20130023576A1 (en) * | 2011-01-24 | 2013-01-24 | Boehringer Ingelheim International Gmbh | Pyrazole Compounds as CRTH2 Antagonists |
| US20140357575A1 (en) * | 2009-06-08 | 2014-12-04 | Palatin Technologies, Inc. | Melanocortin Receptor-Specific Heptapeptides |
| US20170266117A1 (en) * | 2012-04-30 | 2017-09-21 | Tillotts Phharma AG | Delayed release drug formulation |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7645459B2 (en) * | 2004-05-24 | 2010-01-12 | The Procter & Gamble Company | Dosage forms of bisphosphonates |
| FR2937868B1 (fr) * | 2008-11-04 | 2010-11-05 | Galderma Res & Dev | Composes antagonistes des recepteurs de la melanocortine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique |
| WO2010144341A2 (en) * | 2009-06-08 | 2010-12-16 | Palatin Technologies, Inc. | Lactam-bridged melanocortin receptor-specific peptides |
| WO2011063366A1 (en) * | 2009-11-23 | 2011-05-26 | Palatin Technologies, Inc. | Melanocortin-1 receptor-specific cyclic peptides |
| CA2833676C (en) * | 2011-06-14 | 2019-04-23 | Ipsen Pharma S.A.S. | A sustained-release composition containing peptides as active ingredient |
| UA119335C2 (uk) * | 2013-12-11 | 2019-06-10 | Айронвуд Фармасьютикалз, Інк. | Композиції лінаклотиду з затриманим вивільненням |
| US20150307754A1 (en) * | 2014-04-28 | 2015-10-29 | Celanese Acetate Llc | Adhesives that include highly-plasticized cellulose esters and methods and articles relating thereto |
| US10588864B2 (en) * | 2016-03-11 | 2020-03-17 | Gateway Pharmaceuticals LLC | Pharmaceutical compositions for colon-specific delivery |
-
2019
- 2019-03-22 EP EP19771187.2A patent/EP3768245A4/en active Pending
- 2019-03-22 CA CA3095036A patent/CA3095036A1/en active Pending
- 2019-03-22 AU AU2019239300A patent/AU2019239300A1/en not_active Abandoned
- 2019-03-22 CN CN201980034318.2A patent/CN112188888A/zh active Pending
- 2019-03-22 KR KR1020207030569A patent/KR102743821B1/ko active Active
- 2019-03-22 EA EA202092275A patent/EA202092275A1/ru unknown
- 2019-03-22 MX MX2020009900A patent/MX2020009900A/es unknown
- 2019-03-22 IL IL277496A patent/IL277496B2/en unknown
- 2019-03-22 BR BR112020019128-0A patent/BR112020019128A2/pt not_active Application Discontinuation
- 2019-03-22 JP JP2021500503A patent/JP2021523931A/ja active Pending
- 2019-03-22 WO PCT/US2019/023575 patent/WO2019183472A1/en not_active Ceased
-
2020
- 2020-09-22 PH PH12020551596A patent/PH12020551596A1/en unknown
- 2020-09-22 US US17/028,437 patent/US20220088146A1/en not_active Abandoned
-
2025
- 2025-02-19 AU AU2025201154A patent/AU2025201154A1/en active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20140357575A1 (en) * | 2009-06-08 | 2014-12-04 | Palatin Technologies, Inc. | Melanocortin Receptor-Specific Heptapeptides |
| US20130023576A1 (en) * | 2011-01-24 | 2013-01-24 | Boehringer Ingelheim International Gmbh | Pyrazole Compounds as CRTH2 Antagonists |
| US20170266117A1 (en) * | 2012-04-30 | 2017-09-21 | Tillotts Phharma AG | Delayed release drug formulation |
Non-Patent Citations (1)
| Title |
|---|
| PATEL, MP ET AL., LOOP SWAPPED CHIMERAS OF THE AGOUTI-RELATED PROTEIN (AGRP) AND THE AGOUTI SIGNALING PROTEIN (ASIP) IDENTIFY CONTACTS REQUIRED FOR MELANOCORTIN 1 RECEPTOR (MC1R) SELECTIVITY AND ANTAGONISM., 19 November 2010 (2010-11-19) * |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2021523931A (ja) | 2021-09-09 |
| BR112020019128A2 (pt) | 2021-01-12 |
| EP3768245A1 (en) | 2021-01-27 |
| PH12020551596A1 (en) | 2021-08-16 |
| IL277496A (en) | 2020-11-30 |
| IL277496B1 (en) | 2024-09-01 |
| CN112188888A (zh) | 2021-01-05 |
| US20220088146A1 (en) | 2022-03-24 |
| KR102743821B1 (ko) | 2024-12-18 |
| WO2019183472A1 (en) | 2019-09-26 |
| MX2020009900A (es) | 2021-01-08 |
| KR20210003759A (ko) | 2021-01-12 |
| CA3095036A1 (en) | 2019-09-26 |
| EP3768245A4 (en) | 2023-10-18 |
| AU2025201154A1 (en) | 2025-03-13 |
| AU2019239300A1 (en) | 2020-11-19 |
| EA202092275A1 (ru) | 2021-02-09 |
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