IL27126A - 4,3,2,1-Tetrahydro-6-sulfamyl-H) -43) Coinazolinones and the process for their preparation - Google Patents

4,3,2,1-Tetrahydro-6-sulfamyl-H) -43) Coinazolinones and the process for their preparation

Info

Publication number
IL27126A
IL27126A IL27126A IL2712666A IL27126A IL 27126 A IL27126 A IL 27126A IL 27126 A IL27126 A IL 27126A IL 2712666 A IL2712666 A IL 2712666A IL 27126 A IL27126 A IL 27126A
Authority
IL
Israel
Prior art keywords
lower alkyl
hydrogen
methyl
sulfamyl
chloro
Prior art date
Application number
IL27126A
Other languages
English (en)
Hebrew (he)
Original Assignee
Vichness I
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vichness I filed Critical Vichness I
Publication of IL27126A publication Critical patent/IL27126A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL27126A 1966-01-03 1966-12-22 4,3,2,1-Tetrahydro-6-sulfamyl-H) -43) Coinazolinones and the process for their preparation IL27126A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US517995A US3360518A (en) 1966-01-03 1966-01-03 Tetrahydro-halo-sulfamyl quinazolinones

Publications (1)

Publication Number Publication Date
IL27126A true IL27126A (en) 1972-01-27

Family

ID=24062092

Family Applications (1)

Application Number Title Priority Date Filing Date
IL27126A IL27126A (en) 1966-01-03 1966-12-22 4,3,2,1-Tetrahydro-6-sulfamyl-H) -43) Coinazolinones and the process for their preparation

Country Status (14)

Country Link
US (1) US3360518A (fr)
AT (2) AT286989B (fr)
BE (1) BE692082A (fr)
BR (1) BR6785894D0 (fr)
CH (1) CH515910A (fr)
DE (1) DE1620740C3 (fr)
DK (1) DK134113B (fr)
ES (1) ES334560A1 (fr)
FI (1) FI51350C (fr)
FR (1) FR6844M (fr)
GB (1) GB1170790A (fr)
IL (1) IL27126A (fr)
NL (1) NL149493B (fr)
SE (1) SE390969B (fr)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3458513A (en) * 1967-11-02 1969-07-29 Wallace & Tiernan Inc 2-substituted-tetrahydro-halosulfamyl-quinazolinones
US3452020A (en) * 1967-11-09 1969-06-24 Wallace & Tiernan Inc 2-alkenyl and 2-alkynyl substituted - tetrahydro - halo-sulfamyl-quinazolinones
US3452019A (en) * 1967-11-16 1969-06-24 Wallace & Tiernan Inc 1-phenylalkyl-tetrahydro-halo-sulfamyl-quinazolinone
US3518267A (en) * 1968-02-23 1970-06-30 Pennwalt Corp 1-aminoalkyl and 1-hydroxyalkyl-tetrahydro-halo-sulfamyl-quinazolinone
US3549629A (en) * 1968-02-29 1970-12-22 Pennwalt Corp 2 - substituted or unsubstituted carboxy tetrahydro - halo - sulfamyl-quinazolinones
US3549636A (en) * 1968-02-29 1970-12-22 Pennwalt Corp 2-alkanoyl,alkanoylalkyl,alkanoyloxyalkyl,and hydroxyalkyl substituted tetrahydro - halo - sulfamyl- quinazolinones
US3549634A (en) * 1968-03-28 1970-12-22 Pennwalt Corp 8,5 - amino - substituted - tetrahydrohalo-sulfamyl-quinazolinones
US3541096A (en) * 1968-12-24 1970-11-17 Pennwalt Corp 2-aryl-substituted-tetrahydro-halo-sulfamyl-quinazolinones
ZA732937B (en) * 1972-05-05 1974-03-27 Maggioni & C Spa Non mercurial diuretics
EP0057763A1 (fr) * 1981-01-26 1982-08-18 Pennwalt Corporation Procédé de préparation de 2-méthyl-4-(o-toluyl)-7-chloro-1,2,3,4-tétrahydro-4-oxo-6-quinazolinesulfonamide
US4522818A (en) * 1982-10-14 1985-06-11 Pennwalt Corporation Diuretic/antihypertensive compositions
US4517179A (en) * 1983-04-29 1985-05-14 Pennwalt Corporation Rapid dissolving, uniform drug compositions and their preparation
US5264439A (en) * 1990-02-13 1993-11-23 Merck & Co., Inc. Quinazolinone, triazolinone and pyrimidinone angiotensin II antagonists incorporating a substituted benzyl element
US5633240A (en) * 1994-09-01 1997-05-27 Academic Pharmaceuticals Parenteral solutions containing metolazone
IT1288123B1 (it) * 1996-09-04 1998-09-10 Nicox Sa Uso di nitroderivati per l'incontinenza urinaria
HUP0400553A3 (en) * 2000-11-21 2010-03-29 Daiichi Sankyo Company Pharmaceutical compositions
CN1681495B (zh) 2002-08-19 2010-05-12 辉瑞产品公司 用于治疗过度增生性疾病的组合物
JP2008520578A (ja) * 2004-11-15 2008-06-19 ニトロメッド インコーポレーティッド 複素環式の酸化窒素供与体基を含む利尿化合物、組成物および使用方法
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
CN101663262B (zh) 2006-12-01 2014-03-26 百时美施贵宝公司 用于治疗动脉粥样硬化和心血管疾病的作为cetp抑制剂的n-(3-苄基)-2,2-(二苯基)-丙-1胺衍生物
WO2014170786A1 (fr) 2013-04-17 2014-10-23 Pfizer Inc. Dérivés de n-pipéridin-3-ylbenzamide dans le traitement des maladies cardiovasculaires
ES2847904T3 (es) 2013-07-23 2021-08-04 Daiichi Sankyo Co Ltd Medicamento para la prevención o el tratamiento de la hipertensión
WO2016055901A1 (fr) 2014-10-08 2016-04-14 Pfizer Inc. Composés d'amide substitué
CN113574055A (zh) 2019-01-18 2021-10-29 阿斯利康(瑞典)有限公司 Pcsk9抑制剂及其使用方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2976289A (en) * 1961-03-21 X-tetrahydro -
GB1464445A (en) * 1973-02-19 1977-02-16 Mitsubishi Electric Corp Apparatus for making a printing master
DE3266655D1 (en) * 1982-06-04 1985-11-07 Hell Rudolf Dr Ing Gmbh Process to avoid image defects in multicolour printing caused by non coincident printing of the colour separations
GB8410860D0 (en) * 1984-04-27 1984-06-06 Crosfield Electronics Ltd Image modification

Also Published As

Publication number Publication date
BR6785894D0 (pt) 1973-12-27
GB1170790A (en) 1969-11-19
US3360518A (en) 1967-12-26
BE692082A (fr) 1967-06-16
ES334560A1 (es) 1967-11-01
FR6844M (fr) 1969-04-08
DK134113B (da) 1976-09-13
AT291269B (de) 1971-07-12
DE1620740A1 (de) 1970-05-21
FI51350B (fr) 1976-08-31
AT286989B (de) 1971-01-11
NL149493B (nl) 1976-05-17
NL6700083A (fr) 1967-07-04
SE390969B (sv) 1977-01-31
FI51350C (fi) 1976-12-10
DK134113C (fr) 1977-02-14
DE1620740C3 (de) 1979-05-10
DE1620740B2 (de) 1978-09-14
CH515910A (de) 1971-11-30

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