IL172585A0 - Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile - Google Patents

Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile

Info

Publication number
IL172585A0
IL172585A0 IL172585A IL17258505A IL172585A0 IL 172585 A0 IL172585 A0 IL 172585A0 IL 172585 A IL172585 A IL 172585A IL 17258505 A IL17258505 A IL 17258505A IL 172585 A0 IL172585 A0 IL 172585A0
Authority
IL
Israel
Prior art keywords
trifluoromethyl
polymorphs
carbonitrile
sulfinyl
pyrazole
Prior art date
Application number
IL172585A
Original Assignee
Maktheshim Chemical Works Ltd
Sharona Zamir
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Maktheshim Chemical Works Ltd, Sharona Zamir filed Critical Maktheshim Chemical Works Ltd
Priority to IL172585A priority Critical patent/IL172585A0/en
Publication of IL172585A0 publication Critical patent/IL172585A0/en
Priority to AU2006324854A priority patent/AU2006324854B8/en
Priority to KR1020087015581A priority patent/KR20080077650A/en
Priority to PCT/IL2006/001441 priority patent/WO2007069254A2/en
Priority to BRPI0620687A priority patent/BRPI0620687A8/en
Priority to KR1020147019887A priority patent/KR20140096396A/en
Priority to US12/097,615 priority patent/US8440709B2/en
Priority to JP2008545252A priority patent/JP5396085B2/en
Priority to EP06832241A priority patent/EP1968578A4/en
Priority to CA2808259A priority patent/CA2808259A1/en
Priority to CA2808257A priority patent/CA2808257A1/en
Priority to CA2630849A priority patent/CA2630849C/en
Priority to IL191856A priority patent/IL191856A/en
Priority to US13/095,829 priority patent/US8691862B2/en
Priority to JP2013010305A priority patent/JP2013144678A/en
Priority to US13/893,045 priority patent/US9023884B2/en
Priority to IL227951A priority patent/IL227951A0/en
Priority to IL227950A priority patent/IL227950A0/en
Priority to US14/230,702 priority patent/US9215873B2/en
Priority to US14/940,201 priority patent/US9580389B2/en
Priority to US15/416,146 priority patent/US9822079B2/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28—Two oxygen or sulfur atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL172585A 2005-12-14 2005-12-14 Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile IL172585A0 (en)

Priority Applications (21)

Application Number Priority Date Filing Date Title
IL172585A IL172585A0 (en) 2005-12-14 2005-12-14 Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile
CA2630849A CA2630849C (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
EP06832241A EP1968578A4 (en) 2005-12-14 2006-12-14 POLYMORPHS AND AMORPHOUS FORMS OF 5-AMINO-l-[2,6- DICHLORO-4-(TRIFLUOROMETHYL)PHENYL]-4- [(TRIFLUOROMETHYL)SULFINYL]-IH-PYRAZOLE-3-CARBONITRILE
CA2808257A CA2808257A1 (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
PCT/IL2006/001441 WO2007069254A2 (en) 2005-12-14 2006-12-14 POLYMORPHS AND AMORPHOUS FORMS OF 5-AMINO-l-[2,6- DICHLORO-4-(TRIFLUOROMETHYL)PHENYL]-4- [(TRIFLUOROMETHYL)SULFINYL]-IH-PYRAZOLE-3-CARBONITRILE
BRPI0620687A BRPI0620687A8 (en) 2005-12-14 2006-12-14 CRYSTALLINE POLYMORPH, PSEUDOMORPH IN HEMISOLVATE, AMORPHOUS COMPOUND, POLYMORPHIC MIXTURE, PROCESS FOR PREPARING A CRYSTALLINE POLYMORPH, PROCESS FOR PREPARING A PSEUDOMORPH OF 5-AMINO-1-[2,6-DICHLORO-4-(TRIFLUOROMETYL) PHENYL] -4- [(TRIFLUOROMETHYL) SULFINIL] -1H- PYRAZOL-3-CARBONITRILE, PROCESS FOR THE PREPARATION OF THE AMORPHOUS FORM OF 5-AMINO-1-[2,6-DICHLORO-4-(TRIFLUOROMETHYL) PHENYL] -4 - [TRIFLUOROMETHYL)SULFINIL]-1H-PYRAZOL-3-CARBONITRILE, PESTICIDE COMPOSITION AND METHOD FOR PEST CONTROL IN A SITE
KR1020147019887A KR20140096396A (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
US12/097,615 US8440709B2 (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
JP2008545252A JP5396085B2 (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1- [2,6-dichloro-4- (trifluoromethyl) phenyl] -4-[(trifluoromethyl) sulfinyl] -1H-pyrazole-3-carbonitrile
AU2006324854A AU2006324854B8 (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6- dichloro-4-(trifluoromethyl)phenyl]-4- [(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
CA2808259A CA2808259A1 (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
KR1020087015581A KR20080077650A (en) 2005-12-14 2006-12-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
IL191856A IL191856A (en) 2005-12-14 2008-06-01 Crystalline forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile, mixtures thereof, process for their preparation and compositions thereof for use as pesticides
US13/095,829 US8691862B2 (en) 2005-12-14 2011-04-27 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
JP2013010305A JP2013144678A (en) 2005-12-14 2013-01-23 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
US13/893,045 US9023884B2 (en) 2005-12-14 2013-05-13 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
IL227951A IL227951A0 (en) 2005-12-14 2013-08-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
IL227950A IL227950A0 (en) 2005-12-14 2013-08-14 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
US14/230,702 US9215873B2 (en) 2005-12-14 2014-03-31 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
US14/940,201 US9580389B2 (en) 2005-12-14 2015-11-13 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
US15/416,146 US9822079B2 (en) 2005-12-14 2017-01-26 Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IL172585A IL172585A0 (en) 2005-12-14 2005-12-14 Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile

Publications (1)

Publication Number Publication Date
IL172585A0 true IL172585A0 (en) 2006-04-10

Family

ID=42331702

Family Applications (1)

Application Number Title Priority Date Filing Date
IL172585A IL172585A0 (en) 2005-12-14 2005-12-14 Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile

Country Status (4)

Country Link
KR (1) KR20140096396A (en)
BR (1) BRPI0620687A8 (en)
CA (2) CA2808259A1 (en)
IL (1) IL172585A0 (en)

Also Published As

Publication number Publication date
KR20140096396A (en) 2014-08-05
BRPI0620687A2 (en) 2011-11-22
CA2808257A1 (en) 2007-06-21
CA2808259A1 (en) 2007-06-21
BRPI0620687A8 (en) 2017-04-11

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