IL160944A0 - Neurotensin active 2,3-diaryl-pyrazolidine derivatives - Google Patents

Neurotensin active 2,3-diaryl-pyrazolidine derivatives

Info

Publication number
IL160944A0
IL160944A0 IL16094403A IL16094403A IL160944A0 IL 160944 A0 IL160944 A0 IL 160944A0 IL 16094403 A IL16094403 A IL 16094403A IL 16094403 A IL16094403 A IL 16094403A IL 160944 A0 IL160944 A0 IL 160944A0
Authority
IL
Israel
Prior art keywords
neurotensin
diaryl
active
pyrazolidine derivatives
pyrazolidine
Prior art date
Application number
IL16094403A
Other languages
English (en)
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Publication of IL160944A0 publication Critical patent/IL160944A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/04—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL16094403A 2002-03-18 2003-03-17 Neurotensin active 2,3-diaryl-pyrazolidine derivatives IL160944A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02076482 2002-03-18
PCT/EP2003/050064 WO2003078400A1 (en) 2002-03-18 2003-03-17 Neurotensin active 2,3-diaryl-pyrazolidine derivatives

Publications (1)

Publication Number Publication Date
IL160944A0 true IL160944A0 (en) 2004-08-31

Family

ID=27838122

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16094403A IL160944A0 (en) 2002-03-18 2003-03-17 Neurotensin active 2,3-diaryl-pyrazolidine derivatives

Country Status (25)

Country Link
US (1) US7186741B2 (es)
EP (1) EP1487802B1 (es)
JP (1) JP4484525B2 (es)
KR (1) KR20040106290A (es)
CN (1) CN100509788C (es)
AR (1) AR038967A1 (es)
AT (1) ATE493390T1 (es)
AU (1) AU2003219165B2 (es)
BR (1) BR0306149A (es)
CA (1) CA2462694C (es)
DE (1) DE60335525D1 (es)
DK (1) DK1487802T3 (es)
ES (1) ES2358894T3 (es)
HK (1) HK1070646A1 (es)
HR (1) HRP20040275A2 (es)
IL (1) IL160944A0 (es)
MX (1) MXPA04004743A (es)
NO (1) NO20044405L (es)
PL (1) PL371440A1 (es)
PT (1) PT1487802E (es)
RU (1) RU2304578C2 (es)
SI (1) SI1487802T1 (es)
UA (1) UA77775C2 (es)
WO (1) WO2003078400A1 (es)
ZA (1) ZA200404741B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1801098A1 (en) 2005-12-16 2007-06-27 Merck Sante 2-Adamantylurea derivatives as selective 11B-HSD1 inhibitors
CN102241678B (zh) 2011-04-26 2014-10-29 辽宁利锋科技开发有限公司 含有脂环结构化合物的抗肿瘤作用与应用
US10377718B2 (en) 2014-06-06 2019-08-13 Research Triangle Institute Apelin receptor (APJ) agonists and uses thereof
EP3386976A1 (en) 2015-12-09 2018-10-17 Research Triangle Institute, International Improved apelin receptor (apj) agonists and uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3712365A1 (de) 1987-04-11 1988-10-27 Hoechst Ag Neue 2-acylpyrrolidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel sowie deren verwendung
PH27357A (en) * 1989-09-22 1993-06-21 Fujisawa Pharmaceutical Co Pyrazole derivatives and pharmaceutical compositions comprising the same
FR2665898B1 (fr) * 1990-08-20 1994-03-11 Sanofi Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2711140B1 (fr) * 1993-10-12 1996-01-05 Sanofi Sa 1-Naphtylpyrazole-3-carboxamides substitués actifs sur la neurotensine, leur préparation, les compositions pharmaceutiques en contenant.

Also Published As

Publication number Publication date
MXPA04004743A (es) 2004-08-02
CA2462694A1 (en) 2003-09-25
CN100509788C (zh) 2009-07-08
NO20044405L (no) 2004-10-15
PT1487802E (pt) 2011-03-11
AU2003219165B2 (en) 2008-03-13
ES2358894T3 (es) 2011-05-16
JP2005527528A (ja) 2005-09-15
CN1592742A (zh) 2005-03-09
RU2304578C2 (ru) 2007-08-20
BR0306149A (pt) 2004-10-19
EP1487802B1 (en) 2010-12-29
DE60335525D1 (de) 2011-02-10
EP1487802A1 (en) 2004-12-22
AU2003219165A1 (en) 2003-09-29
HK1070646A1 (en) 2005-06-24
AR038967A1 (es) 2005-02-02
CA2462694C (en) 2010-08-10
ZA200404741B (en) 2005-08-29
PL371440A1 (en) 2005-06-13
HRP20040275A2 (en) 2004-08-31
JP4484525B2 (ja) 2010-06-16
SI1487802T1 (sl) 2011-04-29
DK1487802T3 (da) 2011-04-04
UA77775C2 (en) 2007-01-15
US20040242493A1 (en) 2004-12-02
US7186741B2 (en) 2007-03-06
ATE493390T1 (de) 2011-01-15
KR20040106290A (ko) 2004-12-17
WO2003078400A1 (en) 2003-09-25
RU2004114262A (ru) 2005-09-20

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