IL138827A0 - Process for preparing 4-substituted-1h-indole-3-glyoxamides - Google Patents

Process for preparing 4-substituted-1h-indole-3-glyoxamides

Info

Publication number
IL138827A0
IL138827A0 IL13882799A IL13882799A IL138827A0 IL 138827 A0 IL138827 A0 IL 138827A0 IL 13882799 A IL13882799 A IL 13882799A IL 13882799 A IL13882799 A IL 13882799A IL 138827 A0 IL138827 A0 IL 138827A0
Authority
IL
Israel
Prior art keywords
glyoxamides
indole
substituted
preparing
Prior art date
Application number
IL13882799A
Other languages
English (en)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL138827A0 publication Critical patent/IL138827A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/22Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an aralkyl radical attached to the ring nitrogen atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL13882799A 1998-04-17 1999-04-15 Process for preparing 4-substituted-1h-indole-3-glyoxamides IL138827A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8211098P 1998-04-17 1998-04-17
PCT/US1999/008332 WO1999054300A1 (en) 1998-04-17 1999-04-15 Process for preparing 4-substituted-1h-indole-3-glyoxamides

Publications (1)

Publication Number Publication Date
IL138827A0 true IL138827A0 (en) 2001-10-31

Family

ID=22169126

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13882799A IL138827A0 (en) 1998-04-17 1999-04-15 Process for preparing 4-substituted-1h-indole-3-glyoxamides

Country Status (27)

Country Link
US (1) US6265591B1 (de)
EP (1) EP1071663A4 (de)
JP (1) JP2002512225A (de)
KR (1) KR20010042741A (de)
CN (1) CN1305459A (de)
AR (1) AR015767A1 (de)
AU (1) AU750368B2 (de)
BR (1) BR9909697A (de)
CA (1) CA2326515A1 (de)
CO (1) CO5080803A1 (de)
DZ (1) DZ2770A1 (de)
EA (1) EA003582B1 (de)
EG (1) EG22139A (de)
HK (1) HK1039120A1 (de)
HR (1) HRP20000685A2 (de)
HU (1) HUP0101344A3 (de)
ID (1) ID26021A (de)
IL (1) IL138827A0 (de)
NO (1) NO20005148L (de)
NZ (1) NZ507175A (de)
PE (1) PE20000430A1 (de)
PL (1) PL343487A1 (de)
SK (1) SK15372000A3 (de)
SV (1) SV1999000043A (de)
TR (1) TR200002999T2 (de)
WO (1) WO1999054300A1 (de)
ZA (1) ZA200005294B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6407261B1 (en) 1998-04-17 2002-06-18 Eli Lilly And Company Process for preparing 4-hdyroxy indole, indazole and carbazole compounds
JP2002512222A (ja) * 1998-04-17 2002-04-23 イーライ・リリー・アンド・カンパニー 4−ヒドロキシインドール、インダゾール、及び、カルバゾール化合物の製造方法
DE19962300A1 (de) * 1999-12-23 2001-06-28 Asta Medica Ag Substituierte N-Benzyl-Indol-3-yl-glyoxylsäure-Derivate mit Antitumorwirkung
US20030225149A1 (en) * 2002-04-30 2003-12-04 Blazecka Peter G. Process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids
MY198422A (en) 2009-04-29 2023-08-29 Amarin Pharmaceuticals Ie Ltd Pharmaceutical compositions comprising epa and a cardiovascular agent and methods of using the same
AR088377A1 (es) 2011-10-20 2014-05-28 Siena Biotech Spa Proceso para la preparacion de 6-cloro-2,3,4,9-tetrahidro-1h-carbazol-1-carboxamida y compuestos intermedios de esta

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL180523B1 (pl) * 1994-04-01 2001-02-28 Eli Lilly & Co Nowy zwiazek, pochodna 1H-indolo-3-glioksylamidu i srodek farmaceutyczny PL PL PL PL PL PL PL PL PL PL
JP2002512222A (ja) * 1998-04-17 2002-04-23 イーライ・リリー・アンド・カンパニー 4−ヒドロキシインドール、インダゾール、及び、カルバゾール化合物の製造方法

Also Published As

Publication number Publication date
PL343487A1 (en) 2001-08-27
EA200001076A1 (ru) 2001-04-23
CO5080803A1 (es) 2001-09-25
NO20005148D0 (no) 2000-10-13
AU3564899A (en) 1999-11-08
AU750368B2 (en) 2002-07-18
HUP0101344A2 (hu) 2001-09-28
BR9909697A (pt) 2000-12-19
HUP0101344A3 (en) 2002-12-28
SK15372000A3 (sk) 2001-08-06
KR20010042741A (ko) 2001-05-25
CA2326515A1 (en) 1999-10-28
TR200002999T2 (tr) 2001-01-22
NO20005148L (no) 2000-11-09
ZA200005294B (en) 2001-10-01
SV1999000043A (es) 2000-05-02
CN1305459A (zh) 2001-07-25
DZ2770A1 (fr) 2003-12-01
NZ507175A (en) 2002-12-20
EP1071663A1 (de) 2001-01-31
HK1039120A1 (zh) 2002-04-12
HRP20000685A2 (en) 2001-10-31
US6265591B1 (en) 2001-07-24
AR015767A1 (es) 2001-05-16
EA003582B1 (ru) 2003-06-26
EP1071663A4 (de) 2002-06-19
WO1999054300A1 (en) 1999-10-28
JP2002512225A (ja) 2002-04-23
ID26021A (id) 2000-11-16
PE20000430A1 (es) 2000-05-24
EG22139A (en) 2002-08-30

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