IL128917A - Heteroaryloxyethylamines as 5-ht1a receptor ligands, a process for their preparation and pharmaceutical compositions containing them - Google Patents

Heteroaryloxyethylamines as 5-ht1a receptor ligands, a process for their preparation and pharmaceutical compositions containing them

Info

Publication number
IL128917A
IL128917A IL12891797A IL12891797A IL128917A IL 128917 A IL128917 A IL 128917A IL 12891797 A IL12891797 A IL 12891797A IL 12891797 A IL12891797 A IL 12891797A IL 128917 A IL128917 A IL 128917A
Authority
IL
Israel
Prior art keywords
heteroaryloxyethylamines
preparation
pharmaceutical compositions
compositions containing
receptor ligands
Prior art date
Application number
IL12891797A
Other languages
English (en)
Other versions
IL128917A0 (en
Original Assignee
Scras
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scras filed Critical Scras
Publication of IL128917A0 publication Critical patent/IL128917A0/xx
Publication of IL128917A publication Critical patent/IL128917A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/24Oxygen atoms attached in position 8
    • C07D215/26Alcohols; Ethers thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/24Oxygen atoms attached in position 8
    • C07D215/26Alcohols; Ethers thereof
    • C07D215/28Alcohols; Ethers thereof with halogen atoms or nitro radicals in positions 5, 6 or 7

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
IL12891797A 1996-09-27 1997-09-26 Heteroaryloxyethylamines as 5-ht1a receptor ligands, a process for their preparation and pharmaceutical compositions containing them IL128917A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9611798A FR2753968B1 (fr) 1996-09-27 1996-09-27 Nouvelles heteroaryloxyethylamines, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
PCT/FR1997/001691 WO1998013349A2 (fr) 1996-09-27 1997-09-26 Heteroaryloxyethylamines en tant que ligands 5-ht¿1a?

Publications (2)

Publication Number Publication Date
IL128917A0 IL128917A0 (en) 2000-02-17
IL128917A true IL128917A (en) 2003-10-31

Family

ID=9496126

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12891797A IL128917A (en) 1996-09-27 1997-09-26 Heteroaryloxyethylamines as 5-ht1a receptor ligands, a process for their preparation and pharmaceutical compositions containing them

Country Status (21)

Country Link
US (1) US6063784A (xx)
EP (1) EP0929525B1 (xx)
JP (1) JP2001503393A (xx)
AR (1) AR008486A1 (xx)
AT (1) ATE223380T1 (xx)
AU (1) AU731459B2 (xx)
BR (1) BR9711560A (xx)
CA (1) CA2267247C (xx)
DE (1) DE69715223T2 (xx)
DK (1) DK0929525T3 (xx)
ES (1) ES2182120T3 (xx)
FR (1) FR2753968B1 (xx)
HU (1) HUP0001189A3 (xx)
IL (1) IL128917A (xx)
MY (1) MY118992A (xx)
NO (1) NO311935B1 (xx)
NZ (1) NZ334623A (xx)
PL (1) PL190221B1 (xx)
RU (1) RU2176639C2 (xx)
TW (1) TW425390B (xx)
WO (1) WO1998013349A2 (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4507398B2 (ja) * 1999-12-06 2010-07-21 宇部興産株式会社 3−ハロメチルオキセタン化合物の合成方法
US20040147581A1 (en) * 2002-11-18 2004-07-29 Pharmacia Corporation Method of using a Cox-2 inhibitor and a 5-HT1A receptor modulator as a combination therapy

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK203990D0 (da) * 1990-08-24 1990-08-24 Novo Nordisk As Piperazinylderivater
MX9201991A (es) * 1991-05-02 1992-11-01 Jonh Wyeth & Brother Limited Derivados de piperazina y procedimiento para su preparacion.
US5240800A (en) * 1991-07-29 1993-08-31 Eastman Kodak Company Near-infrared radiation sensitive photoelectrographic master and imaging method
GB9507288D0 (en) * 1995-04-07 1995-05-31 Sod Conseils Rech Applic Phenoxyethylamine derivatives with high affinity for 5-HT1A receptors

Also Published As

Publication number Publication date
NZ334623A (en) 1999-09-29
NO991481D0 (no) 1999-03-26
DK0929525T3 (da) 2002-12-02
CA2267247C (fr) 2009-05-05
HUP0001189A3 (en) 2001-12-28
BR9711560A (pt) 1999-08-24
FR2753968B1 (fr) 1998-11-27
FR2753968A1 (fr) 1998-04-03
WO1998013349A3 (fr) 1998-11-05
PL190221B1 (pl) 2005-11-30
NO311935B1 (no) 2002-02-18
ATE223380T1 (de) 2002-09-15
WO1998013349A2 (fr) 1998-04-02
AR008486A1 (es) 2000-01-19
AU4463797A (en) 1998-04-17
TW425390B (en) 2001-03-11
RU2176639C2 (ru) 2001-12-10
IL128917A0 (en) 2000-02-17
MY118992A (en) 2005-02-28
US6063784A (en) 2000-05-16
ES2182120T3 (es) 2003-03-01
CA2267247A1 (fr) 1998-04-02
JP2001503393A (ja) 2001-03-13
AU731459B2 (en) 2001-03-29
EP0929525B1 (fr) 2002-09-04
EP0929525A2 (fr) 1999-07-21
PL332480A1 (en) 1999-09-13
HUP0001189A2 (hu) 2000-10-28
DE69715223T2 (de) 2003-04-30
NO991481L (no) 1999-03-26
DE69715223D1 (de) 2002-10-10

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees