IE831933L - Derivatives of omega-amino acids - Google Patents
Derivatives of omega-amino acidsInfo
- Publication number
- IE831933L IE831933L IE831933A IE193383A IE831933L IE 831933 L IE831933 L IE 831933L IE 831933 A IE831933 A IE 831933A IE 193383 A IE193383 A IE 193383A IE 831933 L IE831933 L IE 831933L
- Authority
- IE
- Ireland
- Prior art keywords
- branched
- linear
- substituted
- radicals
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C221/00—Preparation of compounds containing amino groups and doubly-bound oxygen atoms bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Compounds of the formula I <IMAGE> for use in treating epilepsy, depression, dyskinesias such as Parkinson's disease, muscular spasms of nervous origin, hypertension, hypotension, sleeping troubles, memory defects, and as anthelminthic and analgesic agents wherein R represents:- a linear or branched C2 to C12 alkyl radical a linear or branched C2 to C4 alkyl radical substituted by a phenyl or phenoxy nucleus which may be substituted by one or two linear or branched C1 to C4 alkyl radicals by one or two linear or branched C1 to C4 alkoxy radicals or by one or two halogen atoms a linear or branched C2 to C6 acyl radical substituted by a phenyl nucleus which may be substituted by one or two linear or branched C1 to C4 alkyl radicals by one or two linear or branched C1 to C4 alkoxy radicals or by one or two halogen atoms. R1 represents hydrogen, a linear or branched C2 to C11 acyl radical a linear or branched C2 to C6 acyl radical substituted by a phenyl nucleus which may be substituted by one or two linear or branched C1 to C4 alkyl radicals by one or two linear or branched C1 to C4 alkoxy radicals or by one or two atoms of halogen, such as fluorine, chlorine or bromine, R2 represents:- a hydroxyl group an alkoxy group R3O- in which R3 is a linear or branched C1 to C3 alkyl radical; an amino group; and n is 3, 4 or 5; or a pharmaceutically or veterinarily acceptable salt thereof.
[GB2126224A]
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| LU84343 | 1982-08-20 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE831933L true IE831933L (en) | 1984-02-20 |
| IE55872B1 IE55872B1 (en) | 1991-02-14 |
Family
ID=19729937
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE1933/83A IE55872B1 (en) | 1982-08-20 | 1983-08-18 | Derivatives of omega-amino acids,the preparation and utilisation thereof,and the compositions containing these derivatives |
Country Status (24)
| Country | Link |
|---|---|
| JP (1) | JPS5962555A (en) |
| KR (1) | KR870000980B1 (en) |
| AU (2) | AU1814083A (en) |
| BE (1) | BE897566A (en) |
| CA (1) | CA1256899A (en) |
| CH (1) | CH659466A5 (en) |
| DE (2) | DE3329628A1 (en) |
| DK (1) | DK373383A (en) |
| ES (2) | ES8602608A1 (en) |
| FI (1) | FI832935A (en) |
| FR (1) | FR2531950B1 (en) |
| GB (1) | GB2126224B (en) |
| GR (1) | GR77444B (en) |
| IE (1) | IE55872B1 (en) |
| IL (1) | IL69543A (en) |
| IT (1) | IT1169767B (en) |
| MA (1) | MA19882A1 (en) |
| MX (1) | MX156348A (en) |
| NL (1) | NL8302916A (en) |
| NO (1) | NO163770C (en) |
| OA (1) | OA07525A (en) |
| PT (1) | PT77226B (en) |
| SE (1) | SE8304513L (en) |
| ZA (1) | ZA836130B (en) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3476197D1 (en) * | 1983-08-01 | 1989-02-23 | Mclean Hospital Corp | Gaba esters and gaba analogue esters |
| DE3445816C1 (en) | 1984-12-15 | 1986-06-12 | Behringwerke Ag, 3550 Marburg | Flat diagnostic agent |
| GB8813185D0 (en) * | 1988-06-03 | 1988-07-06 | Wyeth John & Brother Ltd | New method & amines used therein |
| CA2028782C (en) * | 1989-11-07 | 2003-10-14 | Christian T. Goralski | Process for the production of vinyl-gaba |
| US5585358A (en) * | 1993-07-06 | 1996-12-17 | Yissum Research Development Corporation Of The Hebrew University Of Jerusalem | Derivatives of valproic acid amides and 2-valproenoic acid amides, method of making and use thereof as anticonvulsant agents |
| KR100491282B1 (en) | 1996-07-24 | 2005-05-24 | 워너-램버트 캄파니 엘엘씨 | Isobutylgaba and Its Derivatives for the Treatment of Pain |
| FR2753967B1 (en) * | 1996-09-27 | 1998-11-27 | Sod Conseils Rech Applic | NOVEL PHENOXYETHYLAMINE DERIVATIVES, THEIR PREPARATION PROCESS, THEIR USE AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| UA59384C2 (en) | 1996-12-20 | 2003-09-15 | Пфайзер, Інк. | Preventing bone mass loss and recovery thereof by means of prostaglandin agonists |
| UA67754C2 (en) | 1997-10-10 | 2004-07-15 | Пфайзер, Інк. | Prostaglandin agonists and use thereof for the treatment of bone disorders |
| KR100843703B1 (en) | 2000-07-21 | 2008-07-04 | 이섬 리서치 디벨러프먼트 컴파니 오브 더 히브루 유니버시티 오브 예루살렘 | Use of derivatives of valproic acid and 2-valproenic acid amides for the treatment of mania in bipolar disorder |
| DE60134337D1 (en) | 2000-11-21 | 2008-07-17 | Ucb Pharma Sa | N-ALKYLATED GABA COMPOUNDS, METHODS THEREOF |
| EP1675822A2 (en) * | 2003-10-16 | 2006-07-05 | Cara Therapeutics, Inc. | Amide or thioamide derivatives and their use in the treatment of pain |
| FR3018076B1 (en) | 2014-03-03 | 2016-02-19 | Arkema France | PROCESS FOR PREPARING DERIVATIVES OF 11-AMINOUNDECANOIC ACID AND 12-AMINODODECANOIC ACID |
| WO2020031201A1 (en) * | 2018-08-04 | 2020-02-13 | Msn Laboratories Private Limited, R&D Center | Improved process for the preparation of 6-aminohexanoic acid |
| CN109593044B (en) * | 2018-12-06 | 2021-05-14 | 盐城工学院 | Alkyl fatty acid amine and preparation method thereof |
| CN115636761B (en) * | 2021-07-20 | 2024-07-05 | 中国石油天然气股份有限公司 | Oil-soluble surfactant, oil displacement agent and application thereof |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE636245A (en) * | ||||
| GB586645A (en) * | 1944-07-19 | 1947-03-26 | Burroughs Wellcome Co | Improvements relating to the synthesis of amino acid derivatives and salts thereof |
| GB775364A (en) * | 1954-05-05 | 1957-05-22 | Unilever Ltd | Improvements in soap compositions |
| US2851345A (en) * | 1955-02-02 | 1958-09-09 | Armour & Co | Fuel oil compositions |
| DE1189556B (en) * | 1962-05-29 | 1965-03-25 | Sandoz Ag | Process for the preparation of 3-diaethylaminobutyric acid-N-methylanilide |
| BE647556A (en) * | 1964-05-06 | 1964-08-31 | ||
| IE33790B1 (en) * | 1968-06-04 | 1974-10-30 | Beecham Group Ltd | Derivatives of n-acylaminoacid amides |
| US3954778A (en) * | 1970-03-03 | 1976-05-04 | Zambon S.P.A. | Aminoacetyl derivatives of 2,3-diphenyl cyclopropyl amine |
| GB1369247A (en) * | 1970-08-07 | 1974-10-02 | Pfizer | Amines the preparation thereof and their use in pharmaceutical compositions |
| DE2234399A1 (en) * | 1972-07-17 | 1974-01-31 | Thomae Gmbh Dr K | SKIN PROTECTION PRODUCTS |
| US3947579A (en) * | 1974-06-03 | 1976-03-30 | Nelson Research & Development Company | Method and composition for potentiating neuroleptic drugs |
| GB1538207A (en) * | 1975-12-09 | 1979-01-10 | Mitsubishi Chem Ind | N2-arylsulphonyl-l-argininamides and the pharmaceutically acceptable salts thereof |
| LU78804A1 (en) * | 1977-12-30 | 1979-07-20 | Byk Gulden Lomberg Chem Fab | N-SUBSTITUTED W-AMINOALKANOYL-W-AMINOALKANIC ACIDS, THEIR USE AND METHOD FOR THE PRODUCTION THEREOF, AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS |
| LU78805A1 (en) * | 1977-12-30 | 1979-07-20 | Byk Gulden Lomberg Chem Fab | ACYLHYDROCARBYLAMINO ALKANIC ACIDS, THEIR PRODUCTION AND USE AND THE MEDICINAL PRODUCTS CONTAINING THEM |
| DE3050800C2 (en) * | 1979-03-22 | 1989-06-22 | Continental Pharma Inc., Bruessel/Bruxelles, Be |
-
1983
- 1983-08-16 DK DK373383A patent/DK373383A/en not_active Application Discontinuation
- 1983-08-16 FI FI832935A patent/FI832935A/en not_active Application Discontinuation
- 1983-08-17 DE DE19833329628 patent/DE3329628A1/en active Granted
- 1983-08-17 CA CA000434769A patent/CA1256899A/en not_active Expired
- 1983-08-17 DE DE3347867A patent/DE3347867C2/de not_active Expired
- 1983-08-18 IE IE1933/83A patent/IE55872B1/en unknown
- 1983-08-18 GR GR72245A patent/GR77444B/el unknown
- 1983-08-18 GB GB08322245A patent/GB2126224B/en not_active Expired
- 1983-08-18 NO NO832965A patent/NO163770C/en unknown
- 1983-08-19 AU AU18140/83A patent/AU1814083A/en not_active Abandoned
- 1983-08-19 OA OA58092A patent/OA07525A/en unknown
- 1983-08-19 SE SE8304513A patent/SE8304513L/en not_active Application Discontinuation
- 1983-08-19 MX MX198462A patent/MX156348A/en unknown
- 1983-08-19 BE BE0/211380A patent/BE897566A/en not_active IP Right Cessation
- 1983-08-19 IT IT22591/83A patent/IT1169767B/en active
- 1983-08-19 ZA ZA836130A patent/ZA836130B/en unknown
- 1983-08-19 NL NL8302916A patent/NL8302916A/en not_active Application Discontinuation
- 1983-08-19 FR FR8313490A patent/FR2531950B1/en not_active Expired
- 1983-08-19 PT PT77226A patent/PT77226B/en not_active IP Right Cessation
- 1983-08-19 CH CH4544/83A patent/CH659466A5/en not_active IP Right Cessation
- 1983-08-19 ES ES525031A patent/ES8602608A1/en not_active Expired
- 1983-08-20 KR KR1019830003898A patent/KR870000980B1/en not_active IP Right Cessation
- 1983-08-20 MA MA20104A patent/MA19882A1/en unknown
- 1983-08-20 JP JP58150964A patent/JPS5962555A/en active Granted
- 1983-08-22 IL IL69543A patent/IL69543A/en unknown
-
1985
- 1985-09-02 ES ES546625A patent/ES8800658A1/en not_active Expired
-
1988
- 1988-04-18 AU AU14727/88A patent/AU1472788A/en not_active Abandoned
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