IE51657B1 - Lh-rh antagonists - Google Patents

Lh-rh antagonists

Info

Publication number
IE51657B1
IE51657B1 IE1213/81A IE121381A IE51657B1 IE 51657 B1 IE51657 B1 IE 51657B1 IE 1213/81 A IE1213/81 A IE 1213/81A IE 121381 A IE121381 A IE 121381A IE 51657 B1 IE51657 B1 IE 51657B1
Authority
IE
Ireland
Prior art keywords
phe
compound
trp
formula
peptide
Prior art date
Application number
IE1213/81A
Other languages
English (en)
Other versions
IE811213L (en
Original Assignee
Schally Andrew Victor
Coy David Howard
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/155,249 external-priority patent/US4317815A/en
Application filed by Schally Andrew Victor, Coy David Howard filed Critical Schally Andrew Victor
Publication of IE811213L publication Critical patent/IE811213L/xx
Publication of IE51657B1 publication Critical patent/IE51657B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IE1213/81A 1980-06-02 1981-06-02 Lh-rh antagonists IE51657B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/155,249 US4317815A (en) 1979-06-13 1980-06-02 LH-RH Antagonists

Publications (2)

Publication Number Publication Date
IE811213L IE811213L (en) 1981-12-02
IE51657B1 true IE51657B1 (en) 1987-02-04

Family

ID=22554652

Family Applications (1)

Application Number Title Priority Date Filing Date
IE1213/81A IE51657B1 (en) 1980-06-02 1981-06-02 Lh-rh antagonists

Country Status (13)

Country Link
EP (1) EP0041286B1 (el)
JP (1) JPS5714568A (el)
AT (1) ATE8988T1 (el)
AU (1) AU7125381A (el)
DE (1) DE3165535D1 (el)
DK (1) DK239781A (el)
ES (1) ES8207511A1 (el)
FI (1) FI811682L (el)
GR (1) GR75673B (el)
HU (1) HU185427B (el)
IE (1) IE51657B1 (el)
PT (1) PT73105B (el)
ZA (1) ZA813356B (el)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU9102582A (en) * 1981-12-10 1983-06-16 David Howard Coy Lh-rh antagonists
US4444759A (en) * 1982-07-26 1984-04-24 The Salk Institute For Biological Studies GnRH Antagonists II
IL70888A0 (en) * 1983-03-10 1984-05-31 Salk Inst For Biological Studi Gn rh antagonist peptides and pharmaceutical compositions containing them
EP0145032B1 (en) * 1983-08-16 1987-11-04 Akzo N.V. Lh- rh antagonists
US4547370A (en) * 1983-11-29 1985-10-15 The Salk Institute For Biological Studies GnRH Antagonists
IL74827A (en) * 1984-05-21 1989-06-30 Salk Inst For Biological Studi Peptides active as gnrh antagonists and pharmaceutical compositions containing them
JP2673025B2 (ja) * 1988-02-10 1997-11-05 タツプ・フアーマシユーテイカルズ・インコーポレイテツド 小さいサイズのｌｈｒｈ類似体
US5140009A (en) * 1988-02-10 1992-08-18 Tap Pharmaceuticals, Inc. Octapeptide LHRH antagonists
DE69330838T2 (de) * 1992-12-18 2002-04-25 Abbott Laboratories, Abbott Park Lhrh antagonisten mit modifizierten aminoacylresten an den positionen 5 und 6
DE10040700A1 (de) * 2000-08-17 2002-02-28 Asta Medica Ag Salze von biologisch aktiven Peptiden, ihre Herstellung und Verwendung

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4211769A (en) * 1977-08-24 1980-07-08 Takeda Chemical Industries, Ltd. Preparations for vaginal administration
NZ188987A (en) * 1977-11-30 1982-02-23 Salk Inst For Biological Studi Peptide analogues of luteinizing hormone releasing factor

Also Published As

Publication number Publication date
DK239781A (da) 1981-12-03
HU185427B (en) 1985-02-28
JPS5714568A (en) 1982-01-25
ATE8988T1 (de) 1984-09-15
GR75673B (el) 1984-08-02
EP0041286B1 (en) 1984-08-15
PT73105B (en) 1982-07-05
ES502688A0 (es) 1982-10-01
IE811213L (en) 1981-12-02
EP0041286A1 (en) 1981-12-09
FI811682L (fi) 1981-12-03
ES8207511A1 (es) 1982-10-01
ZA813356B (en) 1982-06-30
PT73105A (en) 1981-06-01
AU7125381A (en) 1981-12-10
DE3165535D1 (en) 1984-09-20

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