IE43791B1 - 1,2-dihydro-4h-imidazo/1,2-a/ /1,4/benzodiazepin-1-ones,prcess for their preparation,and compositions incorporating them - Google Patents

1,2-dihydro-4h-imidazo/1,2-a/ /1,4/benzodiazepin-1-ones,prcess for their preparation,and compositions incorporating them

Info

Publication number
IE43791B1
IE43791B1 IE298/76A IE29876A IE43791B1 IE 43791 B1 IE43791 B1 IE 43791B1 IE 298/76 A IE298/76 A IE 298/76A IE 29876 A IE29876 A IE 29876A IE 43791 B1 IE43791 B1 IE 43791B1
Authority
IE
Ireland
Prior art keywords
radical
piperazin
dihydro
imidazo
benzodiazepin
Prior art date
Application number
IE298/76A
Other languages
English (en)
Other versions
IE43791L (en
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB6509/75A external-priority patent/GB1496426A/en
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IE43791L publication Critical patent/IE43791L/xx
Publication of IE43791B1 publication Critical patent/IE43791B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IE298/76A 1975-02-15 1976-02-13 1,2-dihydro-4h-imidazo/1,2-a/ /1,4/benzodiazepin-1-ones,prcess for their preparation,and compositions incorporating them IE43791B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB6509/75A GB1496426A (en) 1975-02-15 1975-02-15 1,2-dihydro-4h-imidazo(1,2-alpha)(1,4)benzodiazepin-1-ones processes for their preparation and compositions incorporating them
GB4580075 1975-11-04

Publications (2)

Publication Number Publication Date
IE43791L IE43791L (en) 1976-08-15
IE43791B1 true IE43791B1 (en) 1981-06-03

Family

ID=26240753

Family Applications (1)

Application Number Title Priority Date Filing Date
IE298/76A IE43791B1 (en) 1975-02-15 1976-02-13 1,2-dihydro-4h-imidazo/1,2-a/ /1,4/benzodiazepin-1-ones,prcess for their preparation,and compositions incorporating them

Country Status (26)

Country Link
JP (1) JPS5914034B2 (enrdf_load_stackoverflow)
AR (1) AR225721A1 (enrdf_load_stackoverflow)
AT (1) AT351030B (enrdf_load_stackoverflow)
CA (1) CA1073454A (enrdf_load_stackoverflow)
CH (2) CH613706A5 (enrdf_load_stackoverflow)
DE (1) DE2605652A1 (enrdf_load_stackoverflow)
DK (1) DK141250B (enrdf_load_stackoverflow)
EG (1) EG12462A (enrdf_load_stackoverflow)
ES (1) ES445188A1 (enrdf_load_stackoverflow)
FI (1) FI62090C (enrdf_load_stackoverflow)
FR (1) FR2300569A1 (enrdf_load_stackoverflow)
GR (1) GR60028B (enrdf_load_stackoverflow)
HK (1) HK47379A (enrdf_load_stackoverflow)
HU (1) HU173109B (enrdf_load_stackoverflow)
IE (1) IE43791B1 (enrdf_load_stackoverflow)
IL (1) IL48888A (enrdf_load_stackoverflow)
IT (1) IT8047823A0 (enrdf_load_stackoverflow)
LU (1) LU74341A1 (enrdf_load_stackoverflow)
MX (1) MX3327E (enrdf_load_stackoverflow)
NL (1) NL171585C (enrdf_load_stackoverflow)
NO (1) NO146201C (enrdf_load_stackoverflow)
NZ (1) NZ179990A (enrdf_load_stackoverflow)
PH (3) PH14669A (enrdf_load_stackoverflow)
PT (1) PT64796B (enrdf_load_stackoverflow)
SE (1) SE422686B (enrdf_load_stackoverflow)
YU (1) YU42471B (enrdf_load_stackoverflow)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2479818A1 (en) * 1980-04-03 1981-10-09 Roussel Uclaf 2-Substd. phenyl 7-nitro 3H 1,4-benzodiazepinyl aminoacid derivs. - are anxiolytics, tranquillisers, sedatives and anticonvulsants, prepd. by reacting aminoacid or peptide with benzodiazepin-2-thione
FR2502621B1 (enrdf_load_stackoverflow) * 1981-03-27 1983-10-28 Roussel Uclaf

Also Published As

Publication number Publication date
CH613706A5 (en) 1979-10-15
DK141250B (da) 1980-02-11
AR225721A1 (es) 1982-04-30
NL171585B (nl) 1982-11-16
MX3327E (es) 1980-09-29
DE2605652A1 (de) 1976-09-02
NO760468L (enrdf_load_stackoverflow) 1976-08-17
IL48888A (en) 1979-03-12
YU42471B (en) 1988-10-31
FR2300569A1 (fr) 1976-09-10
SE7601592L (sv) 1976-08-16
NO146201B (no) 1982-05-10
YU34576A (en) 1984-12-31
EG12462A (en) 1979-06-30
NO146201C (no) 1982-08-18
GR60028B (en) 1978-03-31
DE2605652C2 (enrdf_load_stackoverflow) 1987-08-20
AU1113776A (en) 1977-08-25
CH618171A5 (en) 1980-07-15
NZ179990A (en) 1978-06-02
LU74341A1 (enrdf_load_stackoverflow) 1976-12-31
HU173109B (hu) 1979-02-28
FI760347A7 (enrdf_load_stackoverflow) 1976-08-16
PT64796B (fr) 1978-02-06
SE422686B (sv) 1982-03-22
PH16286A (en) 1983-09-02
ATA107376A (de) 1978-12-15
DK141250C (enrdf_load_stackoverflow) 1980-08-04
IL48888A0 (en) 1976-03-31
HK47379A (en) 1979-07-20
DK58776A (enrdf_load_stackoverflow) 1976-08-16
CA1073454A (en) 1980-03-11
FI62090C (fi) 1982-11-10
PH14669A (en) 1981-10-30
PT64796A (fr) 1976-03-01
IE43791L (en) 1976-08-15
ES445188A1 (es) 1977-09-16
NL171585C (nl) 1983-04-18
FI62090B (fi) 1982-07-30
AT351030B (de) 1979-07-10
JPS5914034B2 (ja) 1984-04-02
PH15282A (en) 1982-11-02
IT8047823A0 (it) 1980-02-06
JPS51105098A (enrdf_load_stackoverflow) 1976-09-17
FR2300569B1 (enrdf_load_stackoverflow) 1979-09-21
NL7601492A (nl) 1976-08-17

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Legal Events

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MK9A Patent expired